Membership
Tour
Register
Log in
Michael Alistair O'Brien
Follow
Person
Welwyn Garden City, GB
People
Overview
Industries
Organizations
People
Information
Impact
Patents Grants
last 30 patents
Information
Patent Grant
CGRP antagonist compounds
Patent number
12,227,521
Issue date
Feb 18, 2025
Nxera Pharma UK Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor
Patent number
10,961,225
Issue date
Mar 30, 2021
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic aza compounds as muscarinic M1 receptor and/or M4 receptor
Patent number
10,689,368
Issue date
Jun 23, 2020
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic aza compounds as muscarnic M1 receptor and/or M4 receptor...
Patent number
10,385,039
Issue date
Aug 20, 2019
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic aza compounds as muscarinic M1 receptor and/or M4 receptor...
Patent number
10,196,380
Issue date
Feb 5, 2019
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperidin-1-yl and azepin-1-yl carboxylates as muscarinic M4 recept...
Patent number
10,030,012
Issue date
Jul 24, 2018
Heptares Therapeutics Limited
David Livermore
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor...
Patent number
9,926,297
Issue date
Mar 27, 2018
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Hydroxybenzamide derivatives and their use as inhibitors of HSP90
Patent number
9,914,719
Issue date
Mar 13, 2018
Astex Therapeutics Ltd.
Gianni Chessari
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic AZA compounds as muscarinic M1 receptor and/or M4 receptor...
Patent number
9,670,183
Issue date
Jun 6, 2017
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperidin-1-yl and azepin-1-yl carboxylates as muscarinic M4 recept...
Patent number
9,593,106
Issue date
Mar 14, 2017
Heptares Therapeutics Limited
David Livermore
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
9,051,278
Issue date
Jun 9, 2015
Astex Therapeutics, Ltd.
Valerio Berdini
C04 - CEMENTS CONCRETE ARTIFICIAL STONE CERAMICS REFRACTORIES
Information
Patent Grant
Bicyclic heterocyclic compounds as FGFR inhibitors
Patent number
8,895,745
Issue date
Nov 25, 2014
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pharmaceutical compounds
Patent number
8,779,132
Issue date
Jul 15, 2014
Astex Therapeutics Limited
Miles Stuart Congreve
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
8,779,147
Issue date
Jul 15, 2014
Astex Therapeutics, Ltd.
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Therapeutic combinations of hydroxybenzamide derivatives as inhibit...
Patent number
8,530,469
Issue date
Sep 10, 2013
Astex Therapeutics Ltd.
Gianni Chessari
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo[1,2-a]pyridine compounds for use in treating cancer
Patent number
8,513,276
Issue date
Aug 20, 2013
Astex Therapeutics Limited
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dihydroxyphenyl isoindolylmethanones
Patent number
8,106,057
Issue date
Jan 31, 2012
Astex Therapeutics, Ltd.
Gianni Chessari
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Hydroxybenzamide derivatives and their use as inhibitors of HSP90
Patent number
8,101,648
Issue date
Jan 24, 2012
Astex Therapeutics, Ltd.
Gianni Chessari
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
8,080,666
Issue date
Dec 20, 2011
Astex Therapeutics, Ltd.
Valerio Berdini
C04 - CEMENTS CONCRETE ARTIFICIAL STONE CERAMICS REFRACTORIES
Information
Patent Grant
Benzimidazole derivatives and their use as protein kinase inhibitors
Patent number
7,977,477
Issue date
Jul 12, 2011
Astex Therapeutics, Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
7,825,140
Issue date
Nov 2, 2010
Astex Therapeutics, Ltd.
Valerio Berdini
C04 - CEMENTS CONCRETE ARTIFICIAL STONE CERAMICS REFRACTORIES
Information
Patent Grant
Dihydroxyphenyl isoindolymethanones
Patent number
7,754,725
Issue date
Jul 13, 2010
Astex Therapeutics Ltd.
Gianni Chessari
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
7,745,638
Issue date
Jun 29, 2010
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
7,385,059
Issue date
Jun 10, 2008
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
GPR52 MODULATOR COMPOUNDS
Publication number
20240376070
Publication date
Nov 14, 2024
NXERA PHARMA UK LIMITED
Stephen Paul WATSON
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
GPR52 MODULATOR COMPOUNDS
Publication number
20240254101
Publication date
Aug 1, 2024
Heptares Therapeutics Limited
Sarah Joanne BUCKNELL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
GPR52 MODULATOR COMPOUNDS
Publication number
20230348416
Publication date
Nov 2, 2023
Heptares Therapeutics Limited
Sarah Joanne BUCKNELL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
GPR52 MODULATOR COMPOUNDS
Publication number
20230002374
Publication date
Jan 5, 2023
Heptares Therapeutics Limited
Sarah Joanne Bucknell
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CGRP ANTAGONIST COMPOUNDS
Publication number
20220306651
Publication date
Sep 29, 2022
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CGRP ANTAGONIST COMPOUNDS
Publication number
20220251110
Publication date
Aug 11, 2022
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC AZA COMPOUNDS AS MUSCARINIC M1 RECEPTOR AND/OR M4 RECEPTOR
Publication number
20200325118
Publication date
Oct 15, 2020
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC AZA COMPOUNDS AS MUSCARINIC M1 RECEPTOR AND/OR M4 RECEPTOR
Publication number
20190337925
Publication date
Nov 7, 2019
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC AZA COMPOUNDS AS MUSCARNIC M1 RECEPTOR AND/OR M4 RECEPTOR...
Publication number
20190112294
Publication date
Apr 18, 2019
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC AZA COMPOUNDS AS MUSCARINIC M1 RECEPTOR AND/OR M4 RECEPTOR...
Publication number
20180179184
Publication date
Jun 28, 2018
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC AZA COMPOUNDS AS MUSCARINIC M1 RECEPTOR AND/OR M4 RECEPTOR...
Publication number
20170240530
Publication date
Aug 24, 2017
Heptares Therapeutics Limited
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PIPERIDIN-1 -YL AND AZEPIN-1 -YL CARBOXYLATES AS MUSCARINIC M4 RECE...
Publication number
20170183338
Publication date
Jun 29, 2017
Heptares Therapeutics Limited
David Livermore
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC AZA COMPOUNDS AS MUSCARINIC M1 RECEPTOR AND/OR M4 RECEPTOR...
Publication number
20170015650
Publication date
Jan 19, 2017
HEPTARES THERAPEUTICS LIMITED
Giles Albert Brown
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PIPERIDIN-1 -YL AND AZEPIN-1 -YL CARBOXYLATES AS MUSCARINIC M4 RECE...
Publication number
20150376179
Publication date
Dec 31, 2015
Takeda Pharmaceutical Company Limited
David Livermore
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3,4-DISUBSTITUTED 1H-PYRAZOLE COMPOUNDS AND THEIR USE AS CYCLIN DEP...
Publication number
20140371213
Publication date
Dec 18, 2014
ASTEX THERAPEUTICS, LTD.
Valerio BERDINI
C04 - CEMENTS CONCRETE ARTIFICIAL STONE CERAMICS REFRACTORIES
Information
Patent Application
SUBSTITUTED BENZYLAMINE COMPOUNDS, THEIR USE IN MEDICINE, AND IN PA...
Publication number
20140288040
Publication date
Sep 25, 2014
ASTEX THERAPEUTICS LIMITED
Andrew James Woodhead
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS
Publication number
20140010892
Publication date
Jan 9, 2014
ASTEX THERAPEUTICS LIMITED
Valerio BERDINI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3,4-DISUBSTITUTED 1H-PYRAZOLE COMPOUNDS AND THEIR USE AS CYCLIN DEP...
Publication number
20120213791
Publication date
Aug 23, 2012
ASTEX THERAPEUTICS, LTD.
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS
Publication number
20110224203
Publication date
Sep 15, 2011
ASTEX THERAPEUTICS LIMITED
Valerio BERDINI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3,4-DISUBSTITUTED 1H-PYRAZOLE COMPOUNDS AND THEIR USE AS CYCLIN DEP...
Publication number
20110003799
Publication date
Jan 6, 2011
ASTEX THERAPEUTICS, LTD.
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
DIHYDROXYPHENYL ISOINDOLYLMETHANONES
Publication number
20100286167
Publication date
Nov 11, 2010
Gianni Chessari
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLE DERIVATIVES AS THAT MODULATE THE ACTIVITY OF CDK, GSK AND...
Publication number
20100160324
Publication date
Jun 24, 2010
ASTEX THERAPEUTICS LIMITED
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHARMACEUTICAL COMPOUNDS
Publication number
20100152184
Publication date
Jun 17, 2010
ASTEX THERAPEUTICS LIMITED
Miles Stuart Congreve
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic Heterocyclic Compounds as FGFR Inhibitors
Publication number
20100120761
Publication date
May 13, 2010
ASTEX THERAPEUTICS LIMITED
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Compounds
Publication number
20100093718
Publication date
Apr 15, 2010
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Hydroxybenzamide derivatives and their use as inhibitors of HSP90
Publication number
20090215772
Publication date
Aug 27, 2009
ASTEX THERAPEUTICS LIMITED
Gianni Chessari
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrimidine Derivatives As HSP90 Inhibitors
Publication number
20090215777
Publication date
Aug 27, 2009
Astex Therapeutics Ltd.
Gianni Chessari
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Thiazole And Isothiazole Derivatives That Modulate The Activity Of...
Publication number
20080312223
Publication date
Dec 18, 2008
ASTEX THERAPEUTICS LIMITED
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pharmaceutical Compounds
Publication number
20080306054
Publication date
Dec 11, 2008
ASTEX THERAPEUTICS LIMITED
Gianni Chessari
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrazole Derivatives for the Inhibition of CDK'S and GSK'S
Publication number
20080306069
Publication date
Dec 11, 2008
ASTEX THERAPEUTICS LIMITED
Paul Graham Wyatt
C07 - ORGANIC CHEMISTRY