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Michael Eissenstat
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Frederick, MD, US
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Patents Grants
last 30 patents
Information
Patent Grant
Compositions and methods for inhibiting cytochrome P450
Patent number
9,849,107
Issue date
Dec 26, 2017
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compositions and methods for inhibiting cytochrome P450 2D6
Patent number
9,604,952
Issue date
Mar 28, 2017
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Diamide inhibitors of cytochrome P450
Patent number
9,540,354
Issue date
Jan 10, 2017
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzofuran-containing amino acid inhibitors of cytochrome P450
Patent number
9,403,789
Issue date
Aug 2, 2016
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compositions and methods for inhibiting cytochrome P450
Patent number
9,233,952
Issue date
Jan 12, 2016
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Methods for inhibiting drug degradation
Patent number
8,952,056
Issue date
Feb 10, 2015
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Diamide inhibitors of cytochrome P450
Patent number
8,906,647
Issue date
Dec 9, 2014
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
5-substituted benzofurans as inhibitors of cytochrome P450 2D6
Patent number
8,791,157
Issue date
Jul 29, 2014
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
HCV protease inhibitors
Patent number
8,765,667
Issue date
Jul 1, 2014
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bimacrocylic HCV NS3 protease inhibitors
Patent number
8,703,700
Issue date
Apr 22, 2014
Sequoia Pharmaceuticals, Inc.
Pavel Majer
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
HIV protease inhibitor and cytochrome p450 inhibitor combinations
Patent number
8,673,970
Issue date
Mar 18, 2014
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
5-substituted benzofurans as inhibitors of cytochrome P450 2D6
Patent number
8,569,364
Issue date
Oct 29, 2013
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compositions and methods for inhibiting cytochrome P450
Patent number
8,481,520
Issue date
Jul 9, 2013
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzofuran derived HIV protease inhibitors
Patent number
8,389,571
Issue date
Mar 5, 2013
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compositions and methods for inhibiting cytochrome P450
Patent number
8,048,871
Issue date
Nov 1, 2011
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzofuran derived HIV protease inhibitors
Patent number
7,981,929
Issue date
Jul 19, 2011
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Resistance-repellent retroviral protease inhibitors
Patent number
7,807,845
Issue date
Oct 5, 2010
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Resistance-repellent retroviral protease inhibitors
Patent number
7,507,763
Issue date
Mar 24, 2009
Sequoia Pharmaceuticals
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Small molecule entry inhibitors
Patent number
7,429,677
Issue date
Sep 30, 2008
Tibotec Pharmaceuticals Ltd.
Marie-Pierre T. M. M. G De Bethune
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Resistance-repellent retroviral protease inhibitors
Patent number
7,378,441
Issue date
May 27, 2008
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Resistance-repellent retroviral protease inhibitors
Patent number
7,285,566
Issue date
Oct 23, 2007
John W. Erickson
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Grant
Hexahydrofuro[2,3-B]furan-3-YL-N-{3-[(1,3-benzodioxol-5-ylsulfonyl)...
Patent number
7,157,495
Issue date
Jan 2, 2007
Tibotec Pharmaceuticals, Ltd.
Guangyang Wang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aspartic protease inhibitors
Patent number
7,132,420
Issue date
Nov 7, 2006
The United States of America as represented by the Department of Health and H...
Ramnarayan S. Randad
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Resistance-repellent retroviral protease inhibitors
Patent number
7,109,230
Issue date
Sep 19, 2006
Sequoia Pharmaceuticals, Inc.
John W. Erickson
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Grant
Hexahydrofuro[2,3-B]furan-3-yl-n{3[...
Patent number
6,649,651
Issue date
Nov 18, 2003
Tibotec Pharmaceuticals LTD
Piet T. B. P. Wigerinck
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aspartic protease inhibitors
Patent number
6,613,764
Issue date
Sep 2, 2003
The United States of America as represented by the Department of Health and H...
Ramnarayan S. Randad
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2-(pyrazol-5-yl-oxymethyl)-1,2-benzisothiazol-3 (2H)-One 1, 1-dioxi...
Patent number
5,750,550
Issue date
May 12, 1998
Sanofi
Michael A. Eissenstat
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
COMPOSITIONS AND METHODS FOR INHIBITING CYTOCHROME P450
Publication number
20160361287
Publication date
Dec 15, 2016
SEQUOIA PHARMACEUTICALS, INC.
Michael EISSENSTAT
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
METHODS FOR INHIBITING DRUG DEGRADATION
Publication number
20150284352
Publication date
Oct 8, 2015
SEQUOIA PHARMACEUTICALS, INC.
Michael EISSENSTAT
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Diamide Inhibitors of Cytochrome P450
Publication number
20150087676
Publication date
Mar 26, 2015
Michael EISSENSTAT
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOSITIONS AND METHODS FOR INHIBITING CYTOCHROME P450 2D6
Publication number
20140343078
Publication date
Nov 20, 2014
Michael EISSENSTAT
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Application
COMPOSITIONS AND METHODS FOR INHIBITING CYTOCHROME P450
Publication number
20140024671
Publication date
Jan 23, 2014
Michael EISSENSTAT
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOSITIONS AND METHODS FOR INHIBITING CYTOCHROME P450 2D6
Publication number
20130217704
Publication date
Aug 22, 2013
Michael EISSENSTAT
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Application
Bimacrocylic HCV NS3 Protease Inhibitors
Publication number
20120141414
Publication date
Jun 7, 2012
Sequoia Pharmaceuticals, Inc.
Pavel Majer
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOSITIONS AND METHODS FOR INHIBITING CYTOCHROME P450
Publication number
20120053132
Publication date
Mar 1, 2012
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZOFURAN DERIVED HIV PROTEASE INHIBITORS
Publication number
20110281824
Publication date
Nov 17, 2011
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HCV PROTEASE INHIBITORS
Publication number
20110182854
Publication date
Jul 28, 2011
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMINO ACID INHIBITORS OF CYTOCHROME P450
Publication number
20110124578
Publication date
May 26, 2011
Sequoia Pharmaceuticals Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HIV PROTEASE INHIBITOR AND CYTOCHROME P450 INHIBITOR COMBINATIONS
Publication number
20110112137
Publication date
May 12, 2011
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
DIAMIDE INHIBITORS OF CYTOCHROME P450
Publication number
20110098236
Publication date
Apr 28, 2011
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
METHODS FOR INHIBITING DRUG DEGRADATION
Publication number
20110098237
Publication date
Apr 28, 2011
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
RESISTANCE-REPELLENT RETROVIRAL PROTEASE INHIBITORS
Publication number
20100056596
Publication date
Mar 4, 2010
SEQUOIA PHARMACEUTICALS
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
RESISTANCE-REPELLENT RETROVIRAL PROTEASE INHIBITORS
Publication number
20100009935
Publication date
Jan 14, 2010
SEQUOIA PHARMACEUTICALS
John W. Erickson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOSITIONS AND METHODS FOR INHIBITING CYTOCHROME P450 2D6
Publication number
20090143408
Publication date
Jun 4, 2009
Sequoia Pharmaceuticals, Inc.
Michael EISSENSTAT
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZOFURAN DERIVED HIV PROTEASE INHIBITORS
Publication number
20080227744
Publication date
Sep 18, 2008
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOSITIONS AND METHODS FOR INHIBITING CYTOCHROME P450
Publication number
20080113945
Publication date
May 15, 2008
Sequoia Pharmaceuticals, Inc.
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Long Acting Biologically Active Conjugates
Publication number
20070207952
Publication date
Sep 6, 2007
SEQUOIA PHARMACEUTICALS
Abelardo Silva
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Resistant-repellent retroviral protease inhibitors
Publication number
20060293286
Publication date
Dec 28, 2006
Sequoia Pharmaceuticals, Inc.
John W. Erickson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Resistance-repellent retroviral protease inhibitors
Publication number
20060258737
Publication date
Nov 16, 2006
Sequoia Pharmaceuticals, Inc.
John W. Erickson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Resistance-repellent retroviral protease inhibitors
Publication number
20060258627
Publication date
Nov 16, 2006
SEQUOIA PHARMACEUTICALS
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Small molecule entry inhibitors
Publication number
20060025594
Publication date
Feb 2, 2006
TIBOTEC Pharmaceuticals Ltd.
Marie-Pierre T.M.M.G De Bethune
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Resistance-repellent retroviral protease inhibitors
Publication number
20050267074
Publication date
Dec 1, 2005
SEQUOIA PHARMACEUTICALS
Michael Eissenstat
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Hexahydrofuro[2,3-b]furan-3-yl-N-{3-[(1,3-benzodioxol-5-ylsulfonyl)...
Publication number
20050261364
Publication date
Nov 24, 2005
Guangyang Wang
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Resistance-repellent retroviral protease inhibitors
Publication number
20050209301
Publication date
Sep 22, 2005
SEQUOIA PHARMACEUTICALS
Michael Eissenstat
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Resistance-repellent retroviral protease inhibitors
Publication number
20050107342
Publication date
May 19, 2005
John W. Erickson
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Aspartic protease inhibitors
Publication number
20050090546
Publication date
Apr 28, 2005
Government of the U.S.A., represented by the Secretary, Department of Health...
Ramnarayan S. Randad
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Broad spectrum inhibitors
Publication number
20040009890
Publication date
Jan 15, 2004
John W. Erickson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE