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Michael O'Donnell
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Abingdon, GB
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Patents Grants
last 30 patents
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
12,187,731
Issue date
Jan 7, 2025
Vertex Pharmaceuticals Incorporated
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-(hydroxyalkyl (hetero)aryl) tetrahydrofuran carboxamides as modul...
Patent number
11,827,627
Issue date
Nov 28, 2023
Vertex Pharmaceuticals Incorporated
Elizabeth Mary Beck
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
11,370,798
Issue date
Jun 28, 2022
Vertex Pharmaceuticals Incorporated
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
11,117,900
Issue date
Sep 14, 2021
Vertex Pharmaceuticals Incorporated
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazines as ATR kinase inhibitors
Patent number
10,961,232
Issue date
Mar 30, 2021
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
10,787,452
Issue date
Sep 29, 2020
Vertex Pharmaceuticals Incorporated
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazin-2-amines as inhibitors of ATR kinase
Patent number
10,479,784
Issue date
Nov 19, 2019
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
10,392,391
Issue date
Aug 27, 2019
Vertex Pharmaceuticals Incorporated
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of regioselective synthesis of 2,4-disubstituted pyrimidines
Patent number
10,005,737
Issue date
Jun 26, 2018
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
9,718,827
Issue date
Aug 1, 2017
Vertex Pharmaceuticals Incorporated
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazines as ATR kinase inhibitors
Patent number
9,701,674
Issue date
Jul 11, 2017
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
9,650,381
Issue date
May 16, 2017
Vertex Pharmaceuticals Incorporated
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
9,630,956
Issue date
Apr 25, 2017
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of regioselective synthesis of 2,4-disubstituted pyrimidines
Patent number
9,533,959
Issue date
Jan 3, 2017
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazin-2-amines as inhibitors of ATR kinase
Patent number
9,365,557
Issue date
Jun 14, 2016
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
9,340,546
Issue date
May 17, 2016
Vertex Pharmaceuticals Incorporated
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of regioselective synthesis of 2,4-disubstituted pyrimidines
Patent number
9,296,727
Issue date
Mar 29, 2016
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
8,969,360
Issue date
Mar 3, 2015
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
5-cyano-4- (pyrrolo [2,3B] pyridine-3-yl) -pyrimidine derivatives u...
Patent number
8,962,642
Issue date
Feb 24, 2015
Vertex Pharmaceuticals Incorporated
Michael Mortimore
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aminopyrazines as ATR kinase inhibitors
Patent number
8,877,759
Issue date
Nov 4, 2014
Vertex Pharnaceuticals Incorporated
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
8,841,450
Issue date
Sep 23, 2014
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazin-2-amines useful as inhibitors of ATR kinase
Patent number
8,841,308
Issue date
Sep 23, 2014
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aminopyrimidines useful as kinase inhibitors
Patent number
8,637,511
Issue date
Jan 28, 2014
Vertex Pharmaceuticals Incorporated
Hayley Binch
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods for preparing pyrimidine derivatives useful as protein kina...
Patent number
8,592,577
Issue date
Nov 26, 2013
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
5-cyano-4-(pyrrolo [2,3B] pyridine-3-yl)-pyrimidine derivatives use...
Patent number
8,530,489
Issue date
Sep 10, 2013
Vertex Pharmaceuticals Incorporated
Michael Mortimore
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds useful as inhibitors of ATR kinase
Patent number
8,410,112
Issue date
Apr 2, 2013
Vertex Pharmaceuticals Incorporated
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
5-cyano-4-(pyrrolo [2,3B] pyridine-3-yl)-pyrimidine derivatives use...
Patent number
8,247,421
Issue date
Aug 21, 2012
Vertex Pharmaceuticals Incorporated
Michael Mortimore
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aminopyrimidines useful as kinase inhibitors
Patent number
8,129,399
Issue date
Mar 6, 2012
Vertex Pharmaceuticals Incorporated
Hayley Binch
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aminopyrimidines useful as kinase inhibitors
Patent number
7,767,672
Issue date
Aug 3, 2010
Vertex Pharmaceuticals Incorporated
Hayley Binch
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Caspase inhibitors and uses thereof
Patent number
7,652,153
Issue date
Jan 26, 2010
Vertex Pharmaceuticals Incorporated
Jean Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
N-(HYDROXYALKYL (HETERO)ARYL) TETRAHYDROFURAN CARBOXAMIDE ANALOGS A...
Publication number
20240400544
Publication date
Dec 5, 2024
VERTEX PHARMACEUTICALS INCORPORATED
Elizabeth Mary BECK
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-(HYDROXYALKYL (HETERO)ARYL) TETRAHYDROFURAN CARBOXAMIDES AS MODUL...
Publication number
20240182455
Publication date
Jun 6, 2024
VERTEX PHARMACEUTICALS INCORPORATED
Elizabeth Mary Beck
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20230271963
Publication date
Aug 31, 2023
VERTEX PHARMACEUTICALS INCORPORATED
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20230030414
Publication date
Feb 2, 2023
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20210047333
Publication date
Feb 18, 2021
VERTEX PHARMACEUTICALS INCORPORATED
Nadia AHMAD
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20200140441
Publication date
May 7, 2020
VERTEX PHARMACEUTICALS INCORPORATED
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20190047995
Publication date
Feb 14, 2019
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien CHARRIER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20180170922
Publication date
Jun 21, 2018
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20180155346
Publication date
Jun 7, 2018
VERTEX PHARMACEUTICALS INCORPORATED
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20180072735
Publication date
Mar 15, 2018
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHODS OF REGIOSELECTIVE SYNTHESIS OF 2,4-DISUBSTITUTED PYRIMIDINES
Publication number
20170073315
Publication date
Mar 16, 2017
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20160347754
Publication date
Dec 1, 2016
VERTEX PHARMACEUTICALS INCORPORATED
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20160311809
Publication date
Oct 27, 2016
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHODS OF REGIOSELECTIVE SYNTHESIS OF 2,4-DISUBSTITUTED PYRIMIDINES
Publication number
20160159749
Publication date
Jun 9, 2016
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20150299205
Publication date
Oct 22, 2015
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHODS OF REGIOSELECTIVE SYNTHESIS OF 2,4-DISUBSTITUTED PYRIMIDINES
Publication number
20150099875
Publication date
Apr 9, 2015
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20150051187
Publication date
Feb 19, 2015
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20150031661
Publication date
Jan 29, 2015
VERTEX PHARMACEUTICALS INCORPORATED
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20140275021
Publication date
Sep 18, 2014
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20140249157
Publication date
Sep 4, 2014
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20140163000
Publication date
Jun 12, 2014
Nadia Ahmad
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20140113005
Publication date
Apr 24, 2014
Vertex Pharmaceuticals Incorporated.
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
5-CYANO-4- (PYRROLO [2,3B] PYRIDINE-3-YL) -PYRIMIDINE DERIVATIVES U...
Publication number
20140045812
Publication date
Feb 13, 2014
Michael Mortimore
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Compounds Useful as Inhibitors of ATR Kinase
Publication number
20130115313
Publication date
May 9, 2013
Vertex Pharmaceuticals Incorporated.
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20130095193
Publication date
Apr 18, 2013
Vertex Pharmaceuticals Incorporated.
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
5-CYANO-4- (PYRROLO [2,3B] PYRIDINE-3-YL) -PYRIMIDINE DERIVATIVES U...
Publication number
20120309963
Publication date
Dec 6, 2012
Vertex Pharmaceuticals Incorporated.
Michael Mortimore
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHODS FOR PREPARING PYRIMIDINE DERIVATIVES USEFUL AS PROTEIN KINA...
Publication number
20120271045
Publication date
Oct 25, 2012
Vertex Pharmaceuticals Incorporated.
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMINOPYRIMIDINES USEFUL AS KINASE INHIBITORS
Publication number
20120142660
Publication date
Jun 7, 2012
Vertex Pharmaceuticals Incorporated.
Hayley Binch
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20120040020
Publication date
Feb 16, 2012
Vertex Pharmaceuticals Incorporated.
Jean-Damien Charrier
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE
Publication number
20120035407
Publication date
Feb 9, 2012
Vertex Pharmaceuticals Incorporated.
Jean-Damien Charrier
C07 - ORGANIC CHEMISTRY