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last 30 patents
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Patent Grant
4-amino-6-phenyl-5,6-dihydroimidazo[1,5-A]pyrazine derivatives as i...
Patent number
9,580,433
Issue date
Feb 28, 2017
JANSSEN PHARMACEUTICA NV
Daniel Oehlrich
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzimidazole cannabinoid agonists bearing a substituted heterocycl...
Patent number
9,284,303
Issue date
Mar 15, 2016
JANSSEN PHARMACEUTICA NV
Henricus Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted triazole derivatives as gamma secretase modulators
Patent number
9,079,886
Issue date
Jul 14, 2015
Janssen Pharmaceuticals, Inc.
Sven Franciscus Anna Van Brandt
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted bicyclic heterocyclic compounds as gamma secretase modu...
Patent number
8,946,426
Issue date
Feb 3, 2015
Janssen Pharmaceuticals, Inc.
Henricus Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted triazole and imidazole derivatives as gamma secretase m...
Patent number
8,946,266
Issue date
Feb 3, 2015
Janssen Pharmaceuticals, Inc.
Tongfei Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted benzoxazole, benzimidazole, oxazolopyridine and imidazo...
Patent number
8,772,504
Issue date
Jul 8, 2014
Janssen Pharmaceuticals, Inc.
Henricus Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzimidazole cannabinoid agonists bearing a substituted heterocycl...
Patent number
8,524,757
Issue date
Sep 3, 2013
JANSSEN PHARMACEUTICA NV
Henricus Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidi...
Patent number
8,318,742
Issue date
Nov 27, 2012
Janssen Pharmaceutica, N.V.
Jean-Paul René Marie André Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzimidazole cannabinoid agonists
Patent number
8,193,369
Issue date
Jun 5, 2012
JANSSEN PHARMACEUTICA NV
Henricus Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic benzamides of 3-or 4-substituted 4-(aminomethyl)-piperidin...
Patent number
8,063,070
Issue date
Nov 22, 2011
Janssen Pharmaceutica, N.V.
Jean-Paul René Marie André Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidi...
Patent number
7,790,750
Issue date
Sep 7, 2010
JANSSEN PHARMACEUTICA NV
Jean-Paul René Marie André Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic benzamides of 3-or 4-substituted 4-(aminomethyl)-piperidin...
Patent number
RE40793
Issue date
Jun 23, 2009
Janssen Pharmaceutica, N.V.
Jean-Paul Renë Marie Andrë Bosmans
514 - Drug, bio-affecting and body treating compositions
Information
Patent Grant
Gastrokinetic monocyclic benzamides of 3-or 4-substituted 4-(aminoe...
Patent number
6,750,349
Issue date
Jun 15, 2004
Janssen Pharmaceutics, N.V.
Jean-Paul René Marie André Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidi...
Patent number
6,635,643
Issue date
Oct 21, 2003
Janssen Pharmaceutica, N.V.
Jean-Paul René Marie André Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Gastrokinetic monocyclic benzamides of 3- or 4-substituted 4-(amino...
Patent number
6,452,013
Issue date
Sep 17, 2002
JANSSEN PHARMACEUTICA NV
Jean-Paul René Marie André Bosmans
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
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Patent Application
MACROCYCLIC 2-ALLYLTETRAHYDROFURANS AS INHIBITORS OF MCL-1
Publication number
20240239812
Publication date
Jul 18, 2024
Janssen Pharmaceutica N.V.
Frederik Jan Rita ROMBOUTS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC BRANCHED 3-FLUORO-BUT-3-ENAMIDES AS INHIBITORS OF MCL-1
Publication number
20240083890
Publication date
Mar 14, 2024
Janssen Pharmaceutica N.V.
Meng-Yang HSIAO
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC SPIROCYCLE DERIVATIVES AS MCL-1 INHIBITORS
Publication number
20240067660
Publication date
Feb 29, 2024
Janssen Pharmaceutica N.V.
Frederik Jan Rita ROMBOUTS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYCLIC-2-AMINO-3-FLUORO-BUT-3-ENAMIDES AS INHIBITORS OF MCL-1
Publication number
20230219906
Publication date
Jul 13, 2023
Janssen Pharmaceutica N.V.
Soufyan JERHAOUI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC HETEROCYCLE DERIVATIVES HAVING SELECTIVE BACE1 INHIBITORY...
Publication number
20210261561
Publication date
Aug 26, 2021
Shionogi & Co., Ltd.
Tatsuhiko UENO
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
4-AMINO-6-PHENYL-5,6-DIHYDROIMIDAZO[1,5-A]PYRAZINE DERIVATIVES AS I...
Publication number
20160115170
Publication date
Apr 28, 2016
Janssen Pharmaceutica N.V.
Daniel Oehlrich
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL SUBSTITUTED BICYCLIC HETEROCYCLIC COMPOUNDS AS GAMMA SECRETAS...
Publication number
20150094311
Publication date
Apr 2, 2015
CELLZOME LIMITED
HENRICUS JACOBUS MARIA GIJSEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-DIFLUOROMETHYL-5,6-DIHYDRO-2H-[1,4]OXAZIN-3-AMINE DERIVATIVES
Publication number
20140343048
Publication date
Nov 20, 2014
Andrés Avelino Trabanco-Suárez
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZIMIDAZOLE CANNABINOID AGONISTS BEARING A SUBSTITUTED HETEROCYCL...
Publication number
20130324529
Publication date
Dec 5, 2013
Janssen Pharmaceutica N.V.
Henricus Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL SUBSTITUTED TRIAZOLE DERIVATIVES AS GAMMA SECRETASE MODULATORS
Publication number
20120295891
Publication date
Nov 22, 2012
Sven Franciscus Anna Van Brandt
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL SUBSTITUTED TRIAZOLE AND IMIDAZOLE DERIVATIVES AS GAMMA SECRE...
Publication number
20120135981
Publication date
May 31, 2012
Tongfei Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic Benzamides of 3-Or-4-Substituted 4-(Aminomethyl)-Piperidin...
Publication number
20120028987
Publication date
Feb 2, 2012
Janssen Pharmaceutica N.V.
Jean-Paul René Marie André Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL SUBSTITUTED BENZOXAZOLE, BENZIMIDAZOLE, OXAZOLOPYRIDINE AND I...
Publication number
20120022090
Publication date
Jan 26, 2012
Henricu Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL SUBSTITUTED BICYCLIC HETEROCYCLIC COMPOUNDS AS GAMMA SECRETAS...
Publication number
20110281881
Publication date
Nov 17, 2011
Henricus, Jacobus, Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FLUORO ALKYL SUBSTITUTED BENZIMIDAZOLE CANNABINOID AGONISTS
Publication number
20100273831
Publication date
Oct 28, 2010
Henricus Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic Benzamides of 3-or 4-Substituted 4-(Aminomethyl)-Piperidin...
Publication number
20100210657
Publication date
Aug 19, 2010
Janssen Pharmaceutica N.V.
Jean-Paul René Marie André Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZIMIDAZOLE CANNABINOID AGONISTS
Publication number
20100041702
Publication date
Feb 18, 2010
Henricus Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZIMIDAZOLE CANNABINOID AGONISTS BEARING A SUBSTITUTED HETEROCYCL...
Publication number
20090312339
Publication date
Dec 17, 2009
Janssen Pharmaceutica N.V.
Henricus Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidi...
Publication number
20070037850
Publication date
Feb 15, 2007
Jean-Paul Rene Marie Andre Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidi...
Publication number
20060142342
Publication date
Jun 29, 2006
Jean-Paul Rene Marie Andre Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidi...
Publication number
20060142341
Publication date
Jun 29, 2006
Jean-Paul Rene Marie Andre Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidi...
Publication number
20040058958
Publication date
Mar 25, 2004
Jean-Paul Rene Marie Andre Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Monocyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperi...
Publication number
20030078427
Publication date
Apr 24, 2003
Jean-Paul Rene Marie Andre Bosmans
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic benzamides of 3- or 4-substituted 4-(aminomethyl)-piperidi...
Publication number
20020086879
Publication date
Jul 4, 2002
Jean-Paul Rene Marie Andre Bosmans
C07 - ORGANIC CHEMISTRY