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Naing Aay
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San Mateo, CA, US
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Patents Grants
last 30 patents
Information
Patent Grant
Substituted pyrazolopyrazines, imidazopyrazines and [1,2,4]triazolo...
Patent number
11,739,093
Issue date
Aug 29, 2023
Revolution Medicines, Inc.
Brian R. Blank
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyridine, pyrazine, and triazine compounds as allosteric SHP2 inhib...
Patent number
11,702,411
Issue date
Jul 18, 2023
Revolution Medicines, Inc.
Jie Jack Li
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Ras inhibitors
Patent number
11,690,915
Issue date
Jul 4, 2023
Revolution Medicines, Inc.
Naing Aay
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyridine compounds as allosteric SHP2 inhibitors
Patent number
11,673,896
Issue date
Jun 13, 2023
Revolution Medicines, Inc.
Adrian Gill
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Polycyclic compounds as allosteric SHP2 inhibitors
Patent number
11,673,901
Issue date
Jun 13, 2023
Revolution Medicines, Inc.
Elena S. Koltun
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2,5-disubstituted 3-methyl pyrazines and 2,5,6-trisubstituted 3-met...
Patent number
11,661,401
Issue date
May 30, 2023
Revolution Medicines, Inc.
Elena S. Koltun
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Polycyclic compounds as allosteric SHP2 inhibitors
Patent number
11,634,435
Issue date
Apr 25, 2023
Revolution Medicines, Inc.
Elena S. Koltun
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
MEK inhibitors and methods of their use
Patent number
11,597,699
Issue date
Mar 7, 2023
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic heteroaryl compounds and uses thereof
Patent number
11,168,102
Issue date
Nov 9, 2021
Revolution Medicines, Inc.
Adrian L. Gill
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2,5-disubstituted 3-methyl pyrazines and 2,5,6-trisubstituted 3-met...
Patent number
10,590,090
Issue date
Mar 17, 2020
Revolution Medicines, Inc.
Elena S. Koltun
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzoxazepines as inhibitors of PI3K/mTOR and methods of their use...
Patent number
8,637,499
Issue date
Jan 28, 2014
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4-aryl-2-amino-pyrimidines or 4-aryl-2-aminoalkyl-pyrimidines as JA...
Patent number
8,440,663
Issue date
May 14, 2013
Exelixis, Inc.
Grace Mann
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Azetidines as MEK inhibitors for the treatment of proliferative dis...
Patent number
8,362,002
Issue date
Jan 29, 2013
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrimidinones as casein kinase II (CK2) modulators
Patent number
8,324,231
Issue date
Dec 4, 2012
Exelixis, Inc.
Elena S. Koltun
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-phenylpyrimidinones as PIM modulators
Patent number
8,242,129
Issue date
Aug 14, 2012
Exelixis, Inc.
Amy L. Tsuhako
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tropane compounds
Patent number
8,012,956
Issue date
Sep 6, 2011
Exelixis, Inc.
Kenneth D. Rice
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Azetidines as MEK inhibitors for the treatment of proliferative dis...
Patent number
7,915,250
Issue date
Mar 29, 2011
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Azetidines as MEK inhibitors for the treatment of proliferative dis...
Patent number
7,803,839
Issue date
Sep 28, 2010
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
BICYCLIC COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
Publication number
20240199616
Publication date
Jun 20, 2024
Revolution Medicines, Inc.
Brian R. BLANK
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2,5-DISUBSTITUTED 3-METHYL PYRAZINES AND 2,5,6-TRISUBSTITUTED 3-MET...
Publication number
20240116878
Publication date
Apr 11, 2024
Revolution Medicines, Inc.
Elena S. KOLTUN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
POLYCYCLIC COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
Publication number
20240101577
Publication date
Mar 28, 2024
Revolution Medicines, Inc.
Elena S. KOLTUN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDINE COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
Publication number
20240092795
Publication date
Mar 21, 2024
Revolution Medicines, Inc.
Adrian GILL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDINE, PYRAZINE, AND TRIAZINE COMPOUNDS AS ALLOSTERIC SHP2 INHIB...
Publication number
20240067636
Publication date
Feb 29, 2024
Revolution Medicines, Inc.
Jie Jack LI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
RAS INHIBITORS
Publication number
20230374035
Publication date
Nov 23, 2023
Revolution Medicines, Inc.
Elena S. KOLTUN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC HETEROARYL COMPOUNDS AND USES THEREOF
Publication number
20230365605
Publication date
Nov 16, 2023
Revolution Medicines, Inc.
Adrian L. Gill
C07 - ORGANIC CHEMISTRY
Information
Patent Application
RAS INHIBITORS
Publication number
20230226186
Publication date
Jul 20, 2023
Revolution Medicines, Inc.
Naing AAY
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC HETEROARYL COMPOUNDS AND USES THEREOF
Publication number
20230148450
Publication date
May 11, 2023
Revolution Medicines, Inc.
Andreas BUCKL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC HETEROCYCLYL COMPOUNDS AND USES THEREOF
Publication number
20230096028
Publication date
Mar 30, 2023
Revolution Medicines, Inc.
James Joseph CREGG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC HETEROARYL COMPOUNDS AND USES THEREOF
Publication number
20220135584
Publication date
May 5, 2022
Revolution Medicines, Inc.
Andreas BUCKL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
RAS INHIBITORS
Publication number
20220105185
Publication date
Apr 7, 2022
Revolution Medicines, Inc.
Naing AAY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC HETEROARYL COMPOUNDS AND USES THEREOF
Publication number
20210139517
Publication date
May 13, 2021
Revolution Medicines, Inc.
Adrian L. Gill
C07 - ORGANIC CHEMISTRY
Information
Patent Application
RAS INHIBITORS
Publication number
20210130369
Publication date
May 6, 2021
Revolution Medicines, Inc.
Elena S. KOLTUN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
2,5-DISUBSTITUTED 3-METHYL PYRAZINES AND 2,5,6-TRISUBSTITUTED 3-MET...
Publication number
20210101870
Publication date
Apr 8, 2021
Revolution Medicines, Inc.
Elena S. KOLTUN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
POLYCYCLIC COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
Publication number
20200407372
Publication date
Dec 31, 2020
Revolution Medicines, Inc.
Elena S. KOLTUN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDINE, PYRAZINE, AND TRIAZINE COMPOUNDS AS ALLOSTERIC SHP2 INHIB...
Publication number
20200339552
Publication date
Oct 29, 2020
Revolution Medicines, Inc.
Jie Jack LI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MEK Inhibitors and Methods of Their Use
Publication number
20200283383
Publication date
Sep 10, 2020
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MEK INHIBITORS AND METHODS OF THEIR USE
Publication number
20200031770
Publication date
Jan 30, 2020
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDINE COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
Publication number
20200017517
Publication date
Jan 16, 2020
Revolution Medicines, Inc.
Adrian GILL
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC COMPOUNDS AS ALLOSTERIC SHP2 INHIBITORS
Publication number
20200017511
Publication date
Jan 16, 2020
Revolution Medicines, Inc.
Brian R. BLANK
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2,5-DISUBSTITUTED 3-METHYL PYRAZINES AND 2,5,6-TRISUBSTITUTED 3-MET...
Publication number
20190210977
Publication date
Jul 11, 2019
Revolution Medicines, Inc.
Ashutosh JOGALEKAR
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MEK Inhibitors and Methods of Their Use
Publication number
20190144382
Publication date
May 16, 2019
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MEK Inhibitors And Methods Of Their Use
Publication number
20170166523
Publication date
Jun 15, 2017
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MEK Inhibitors And Methods Of Their Use
Publication number
20150141399
Publication date
May 21, 2015
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Azetidines as MEK Inhibitors for the Treatment of Proliferative Dis...
Publication number
20140275527
Publication date
Sep 18, 2014
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Benzoxazepines as Inhibitors of PI3K/mTOR and Methods of Their Use...
Publication number
20120258953
Publication date
Oct 11, 2012
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Azetidines as MEK Inhibitors for the Treatment of Proliferative Dis...
Publication number
20110263558
Publication date
Oct 27, 2011
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Azetidines as MEK Inhibitors for the Treatment of Proliferative Dis...
Publication number
20100249096
Publication date
Sep 30, 2010
Exelixis, Inc.
Naing Aay
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrimidinones as Casein Kinase II (CK2) Modulators
Publication number
20100144770
Publication date
Jun 10, 2010
Exelixis, Inc.
Elena S. Koltun
C07 - ORGANIC CHEMISTRY