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Paul E. Fleming
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Wellesley, MA, US
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Patents Grants
last 30 patents
Information
Patent Grant
Substituted pyrrolopyridines as inhibitors of activin receptor-like...
Patent number
11,236,086
Issue date
Feb 1, 2022
Blueprint Medicines Corporation
Jason D. Brubaker
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2-(pyridin-3-yl)-pyrimidine derivatives as RET inhibitors
Patent number
10,774,070
Issue date
Sep 15, 2020
Blueprint Medicines Corporation
Natasja Brooijmans
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heteroaryls and uses thereof
Patent number
10,538,533
Issue date
Jan 21, 2020
Millennium Pharmaceuticals, Inc.
Indu T. Bharathan
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Inhibitors of activin receptor-like kinase
Patent number
10,233,186
Issue date
Mar 19, 2019
Blueprint Medicines Corporation
Natasja Brooijmans
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds useful for treating disorders related to RET
Patent number
10,227,329
Issue date
Mar 12, 2019
Blueprint Medicines Corporation
Jason D. Brubaker
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2-(pyridin-3-yl)-pyrimidine derivatives as RET inhibitors
Patent number
10,202,365
Issue date
Feb 12, 2019
Blueprint Medicines Corporation
Natasja Brooijmans
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme
Patent number
10,202,389
Issue date
Feb 12, 2019
Millennium Pharmaceuticals, Inc.
Roushan Afroze
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Derivatives of 1-amino-2-cyclobutylethylboronic acid
Patent number
10,035,811
Issue date
Jul 31, 2018
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heteroaryls and uses thereof
Patent number
9,802,960
Issue date
Oct 31, 2017
Millennium Pharmaceuticals, Inc.
Indu T. Bharathan
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme
Patent number
9,796,725
Issue date
Oct 24, 2017
Millennium Pharmaceuticals, Inc.
Roushan Afroze
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Derivatives of 1-amino-2-cyclobutylethylboronic acid
Patent number
9,771,381
Issue date
Sep 26, 2017
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heteroaryls and uses thereof
Patent number
9,751,854
Issue date
Sep 5, 2017
Millennium Pharmaceuticals, Inc.
Indu T. Bharathan
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme
Patent number
9,663,525
Issue date
May 30, 2017
Millennium Pharmaceuticals, Inc.
Roushan Afroze
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolopyrimidinyl inhibitors of ubiquitin-activating enzyme
Patent number
9,290,500
Issue date
Mar 22, 2016
Millennium Pharmaceuticals, Inc.
Roushan Afroze
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
CCR9 inhibitors and methods of use thereof
Patent number
9,035,096
Issue date
May 19, 2015
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Derivatives of 1-amino-2-cyclopropylethylboronic acid
Patent number
9,023,832
Issue date
May 5, 2015
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Derivatives of 1-amino-2-cyclopropylethylboronic acid
Patent number
8,703,743
Issue date
Apr 22, 2014
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Derivatives of 1-amino-2-cyclobutylethylboronic acid
Patent number
8,664,200
Issue date
Mar 4, 2014
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
CCR9 inhibitors and methods of use thereof
Patent number
8,569,543
Issue date
Oct 29, 2013
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Derivatives of 1-amino-2-cyclopropylethylboronic acid
Patent number
8,513,218
Issue date
Aug 20, 2013
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2-(amino-substituted)-4-aryl pyrimidines and related compounds usef...
Patent number
8,268,822
Issue date
Sep 18, 2012
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
CCR9 inhibitors and methods of use thereof
Patent number
8,030,517
Issue date
Oct 4, 2011
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
CCR9 inhibitors and methods of use thereof
Patent number
7,999,109
Issue date
Aug 16, 2011
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Beta-carbolines useful for treating inflammatory disease
Patent number
7,951,801
Issue date
May 31, 2011
Millennium Pharmaceuticals, Inc.
Michael E. Hepperle
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
CCR9 inhibitors and methods of use thereof
Patent number
7,820,717
Issue date
Oct 26, 2010
Millennium Pharmaceuticals, Inc.
Paul Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2-(amino-substituted)-4-aryl pyrimidines and related compounds usef...
Patent number
7,732,444
Issue date
Jun 8, 2010
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Beta-carbolines useful for treating inflammatory disease
Patent number
7,727,985
Issue date
Jun 1, 2010
Millennium Pharmaceuticals, Inc.
Michael E. Hepperle
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
CCR9 inhibitors and methods of use thereof
Patent number
7,659,272
Issue date
Feb 9, 2010
Millennium Pharmaceuticals, Inc.
Paul Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
CCR9 inhibitors and methods of use thereof
Patent number
7,282,502
Issue date
Oct 16, 2007
Millennium Pharmaceuticals, Inc.
Paul Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
CCR9 inhibitors and methods of use thereof
Patent number
7,238,717
Issue date
Jul 3, 2007
Millennium Pharmaceuticals, Inc.
Paul Fleming
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
INHIBITORS OF ACTIVIN RECEPTOR-LIKE KINASE
Publication number
20220315585
Publication date
Oct 6, 2022
BLUEPRINT MEDICINES CORPORATION
Natasja Brooijmans
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRROLOPYRIDINES AS INHIBITORS OF ACTIVIN RECEPTOR-LIKE...
Publication number
20200331908
Publication date
Oct 22, 2020
BLUEPRINT MEDICINES CORPORATION
Jason D. Brubaker
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2-(PYRIDIN-3-YL)-PYRIMIDINE DERIVATIVES AS RET INHIBITORS
Publication number
20190359591
Publication date
Nov 28, 2019
BLUEPRINT MEDICINES CORPORATION
Natasja Brooijmans
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROARYLS AND USES THEREOF
Publication number
20180118762
Publication date
May 3, 2018
Millennium Pharmaceuticals, Inc.
Indu T. Bharathan
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS USEFUL FOR TREATING DISORDERS RELATED TO RET
Publication number
20180022732
Publication date
Jan 25, 2018
BLUEPRINT MEDICINES CORPORATION
JASON D. BRUBAKER
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2-(PYRIDIN-3-YL)-PYRIMIDINE DERIVATIVES AS RET INHIBITORS
Publication number
20180022731
Publication date
Jan 25, 2018
BLUEPRINT MEDICINES CORPORATION
Natasja Brooijmans
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLOPYRIMIDINYL INHIBITORS OF UBIQUITIN-ACTIVATING ENZYME
Publication number
20170369499
Publication date
Dec 28, 2017
Millennium Pharmaceuticals, Inc.
Roushan Afroze
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DERIVATIVES OF 1-AMINO-2-CYCLOBUTYLETHYLBORONIC ACID
Publication number
20170349611
Publication date
Dec 7, 2017
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INHIBITORS OF ACTIVIN RECEPTOR-LIKE KINASE
Publication number
20170298069
Publication date
Oct 19, 2017
BLUEPRINT MEDICINES CORPORATION
Natasja Brooijmans
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLOPYRIMIDINYL INHIBITORS OF UBIQUITIN-ACTIVATING ENZYME
Publication number
20170217968
Publication date
Aug 3, 2017
Millennium Pharmaceuticals, Inc.
Roushan AFROZE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROARYLS AND USES THEREOF
Publication number
20170073326
Publication date
Mar 16, 2017
Millennium Pharmaceuticals, Inc.
Indu T. BHARATHAN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLOPYRIMIDINYL INHIBITORS OF UBIQUITIN-ACTIVATING ENZYME
Publication number
20160244455
Publication date
Aug 25, 2016
Millennium Pharmaceuticals, Inc.
Roushan AFROZE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CCR9 INHIBITORS AND METHODS OF USE THEREOF
Publication number
20160068479
Publication date
Mar 10, 2016
Millennium Pharmeceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROARYLS AND USES THEREOF
Publication number
20150225422
Publication date
Aug 13, 2015
Millennium Pharmaceuticals, Inc.
Indu T. Bharathan
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
DERIVATIVES OF 1-AMINO-2-CYCLOBUTYLETHYLBORONIC ACID
Publication number
20140194387
Publication date
Jul 10, 2014
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DERIVATIVES OF 1-AMINO-2-CYCLOPROPYLETHYLBORONIC ACID
Publication number
20140179631
Publication date
Jun 26, 2014
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CCR9 INHIBITORS AND METHODS OF USE THEREOF
Publication number
20140107160
Publication date
Apr 17, 2014
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLOPYRIMIDINYL INHIBITORS OF UBIQUITIN-ACTIVATING ENZYME
Publication number
20140088096
Publication date
Mar 27, 2014
Millennium Pharmaceuticals, Inc.
Roushan Afroze
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DERIVATIVES OF 1-AMINO-2-CYCLOPROPYLETHYLBORONIC ACID
Publication number
20140011998
Publication date
Jan 9, 2014
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLOPYRIMIDINYL INHIBITORS OF UBIQUITIN-ACTIVATING ENZYME
Publication number
20130217682
Publication date
Aug 22, 2013
Millennium Pharmaceuticals, Inc.
Roushan Afroze
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CCR9 INHIBITORS AND METHODS OF USE THEREOF
Publication number
20110313000
Publication date
Dec 22, 2011
Millennium Pharmaceuticals, Inc.
Paul Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DERIVATIVES OF 1-AMINO-2-CYCLOPROPYLETHYLBORONIC ACID
Publication number
20110245203
Publication date
Oct 6, 2011
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2-(AMINO-SUBSTITUTED)-4-ARYL PYRIMIDINES AND RELATED COMPOUNDS USEF...
Publication number
20110071134
Publication date
Mar 24, 2011
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CCR9 INHIBITORS AND METHODS OF USE THEREOF
Publication number
20100324093
Publication date
Dec 23, 2010
Millennium Pharmaceuticals, Inc.
Paul Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CCR9 INHIBITORS AND METHODS OF USE THEREOF
Publication number
20100280074
Publication date
Nov 4, 2010
Millennium Pharmaceuticals, Inc.
Paul Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BETA-CARBOLINES USEFUL FOR TREATING INFLAMMATORY DISEASE
Publication number
20100093713
Publication date
Apr 15, 2010
Millennium Pharmaceuticals, Inc.
Michael E. Hepperle
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CCR9 INHIBITORS AND METHODS OF USE THEREOF
Publication number
20100093802
Publication date
Apr 15, 2010
Millennnium Pharmaceuticals, Inc.
Paul Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Derivatives of 1-amino-2-cyclobutylethylboronic acid
Publication number
20100081633
Publication date
Apr 1, 2010
Millennium Pharmaceuticals, Inc.
Paul E. Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CCR9 inhibitors and methods of use thereof
Publication number
20090054495
Publication date
Feb 26, 2009
Millennium Pharmaceuticals, Inc.
Paul Fleming
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CCR9 inhibitors and methods of use thereof
Publication number
20080103180
Publication date
May 1, 2008
Millennium Pharmaceuticals, Inc.
Paul Fleming
C07 - ORGANIC CHEMISTRY