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Stephen P. Raillard
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Mountain View, CA, US
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Patents Grants
last 30 patents
Information
Patent Grant
Methods of synthesizing a levodopa ester prodrug
Patent number
9,533,941
Issue date
Jan 3, 2017
XenoPort, Inc.
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
Patent number
9,353,057
Issue date
May 31, 2016
XenoPort, Inc.
Mark A. Gallop
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Method of making monomethyl fumarate
Patent number
9,302,977
Issue date
Apr 5, 2016
XenoPort, Inc.
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of synthesizing a levodopa ester prodrug
Patent number
9,290,445
Issue date
Mar 22, 2016
XenoPort, Inc.
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Anhydrous and hemihydrate crystalline forms of an (R)-baclofen prod...
Patent number
9,265,748
Issue date
Feb 23, 2016
XenoPort, Inc.
Stephen P. Raillard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Crystalline form of γ-aminobutyric acid analog
Patent number
9,150,503
Issue date
Oct 6, 2015
XenoPort, Inc.
Tono Estrada
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Anhydrous and hemihydrate crystalline forms of an (R)-baclofen prod...
Patent number
9,139,517
Issue date
Sep 22, 2015
XenoPort, Inc.
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Crystalline form of γ-aminobutyric acid analog
Patent number
8,686,034
Issue date
Apr 1, 2014
XenoPort, Inc.
Tono Estrada
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Anhydrous and hemihydrate crystalline forms of an (R)-baclofen prod...
Patent number
8,580,850
Issue date
Nov 12, 2013
XenoPort, Inc.
Stephen P. Raillard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
Patent number
8,378,137
Issue date
Feb 19, 2013
XenoPort, Inc.
Mark A. Gallop
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of synthesizing 1-(acyloxy)-alkyl carbamate prodrugs
Patent number
8,299,291
Issue date
Oct 30, 2012
XenoPort, Inc.
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Enantiomerically resolving acyloxyalkyl thiocarbonates used in synt...
Patent number
8,062,870
Issue date
Nov 22, 2011
XenoPort, Inc.
Mark A. Gallop
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Crystalline form of γ-aminobutyric acid analog
Patent number
8,026,279
Issue date
Sep 27, 2011
XenoPort, Inc.
Tono Estrada
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
Patent number
8,003,809
Issue date
Aug 23, 2011
XenoPort, Inc.
Mark A. Gallop
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of synthesizing N-hydroxysuccinimidyl carbonates
Patent number
7,989,641
Issue date
Aug 2, 2011
XenoPort, Inc.
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
Patent number
7,511,158
Issue date
Mar 31, 2009
XenoPort, Inc.
Mark A. Gallop
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods for synthesis of acyloxyalkyl derivatives of GABA analogs
Patent number
7,423,169
Issue date
Sep 9, 2008
XenoPort, Inc.
Stephen P. Raillard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Methods for synthesis of acyloxyalkyl derivatives of GABA analogs
Patent number
7,232,924
Issue date
Jun 19, 2007
XenoPort, Inc.
Stephen P. Raillard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
Patent number
7,227,028
Issue date
Jun 5, 2007
XenoPort, Inc.
Mark A. Gallop
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
CRYSTALLINE FORM OF y-AMINOBUTYRIC ACID ANALOG
Publication number
20170183296
Publication date
Jun 29, 2017
Xenoport, Inc.
Tono Estrada
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHODS OF SYNTHESIZING A LEVODOPA ESTER PRODRUG
Publication number
20160176804
Publication date
Jun 23, 2016
Xenoport, Inc.
STEPHEN P. RAILLARD
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CRYSTALLINE FORM OF y-AMINOBUTYRIC ACID ANALOG
Publication number
20150353483
Publication date
Dec 10, 2015
Xenoport, Inc.
Tono Estrada
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ANHYDROUS AND HEMIHYDRATE CRYSTALLINE FORMS OF AN (R)-BACLOFEN PROD...
Publication number
20150313865
Publication date
Nov 5, 2015
Xenoport, Inc.
Stephen P. Raillard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
METHOD OF MAKING 1-(ACYLOXY)-ALKYL CARBAMATE COMPOUNDS
Publication number
20150158809
Publication date
Jun 11, 2015
Xenoport, Inc.
Huan Wang
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHOD OF MAKING MONOMETHYL FUMARATE
Publication number
20140364604
Publication date
Dec 11, 2014
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHOD OF MAKING 1-(ACYLOXY)-ALKYL CARBAMATE COMPOUNDS
Publication number
20140243544
Publication date
Aug 28, 2014
Xenoport, Inc.
Huan Wang
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CRYSTALLINE FORM OF y-AMINOBUTYRIC ACID ANALOG
Publication number
20140235710
Publication date
Aug 21, 2014
Xenoport, Inc.
Tono Estrada
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Anhydrous and Hemihydrate Crystalline Forms of an (R)-Baclofen Prod...
Publication number
20140066501
Publication date
Mar 6, 2014
Xenoport, Inc.
Stephen P. Raillard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SYNTHESIS OF ACYLOXYALKYL CARBAMATE PRODRUGS AND INTERMEDIATES THEREOF
Publication number
20130131355
Publication date
May 23, 2013
Xenoport, Inc.
Mark A. Gallop
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ANHYDROUS AND HEMIHYDRATE CRYSTALLINE FORMS OF AN (R)-BACLOFEN PROD...
Publication number
20130041026
Publication date
Feb 14, 2013
Xenoport, Inc.
Stephen P. Raillard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SYNTHESIS OF ACYLOXYALKYL CARBAMATE PRODRUGS AND INTERMEDIATES THEREOF
Publication number
20120010425
Publication date
Jan 12, 2012
Xenoport, Inc.
Mark A. Gallop
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CRYSTALLINE FORM OF y-AMINOBUTYRIC ACID ANALOG
Publication number
20110313036
Publication date
Dec 22, 2011
Xenoport, Inc.
Tono Estrada
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CRYSTALLINE FORM OF y-AMINOBUTYRIC ACID ANALOG
Publication number
20110021628
Publication date
Jan 27, 2011
Xenoport, Inc.
Tono Estrada
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Methods of Synthesizing a Levodopa Ester Prodrug
Publication number
20100099907
Publication date
Apr 22, 2010
XenoPort, Inc.
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHODS OF SYNTHESIZING 1-(ACYLOXY)-ALKYL CARBAMATE PRODRUGS
Publication number
20100087667
Publication date
Apr 8, 2010
Xenoport, Inc.
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHODS OF SYNTHESIZING N-HYDROXYSUCCINIMIDYL CARBONATES
Publication number
20100081830
Publication date
Apr 1, 2010
Xenoport, Inc.
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CRYSTALLINE FORM OF y-AMINOBUTYRIC ACID ANALOG
Publication number
20100056632
Publication date
Mar 4, 2010
Xenoport, Inc.
Tono Estrada
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Synthesis of Acyloxyalkyl Carbamate Prodrugs and Intermediates Thereof
Publication number
20090216037
Publication date
Aug 27, 2009
Xenoport, Inc.
Mark A. Gallop
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ENANTIOMERICALLY RESOLVING ACYLOXYALKYL THIOCARBONATES USED IN SYNT...
Publication number
20090192325
Publication date
Jul 30, 2009
Xenoport, Inc.
Mark A. Gallop
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Methods for Synthesis of Acyloxyalkyl Derivatives of GABA Analogs
Publication number
20080058546
Publication date
Mar 6, 2008
XenoPort, Inc.
Stephen P. Raillard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Synthesis of Acyloxyalkyl Carbamate Prodrugs and Intermediates Thereof
Publication number
20070244331
Publication date
Oct 18, 2007
XenoPort, Inc.
Mark A. GALLOP
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
Publication number
20070037988
Publication date
Feb 15, 2007
XenoPort, Inc.
Mark A. Gallop
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Methods for synthesis of acyloxyalkyl derivatives of GABA analogs
Publication number
20060287250
Publication date
Dec 21, 2006
XenoPort, Inc.
Stephen P. Raillard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Synthesis of acyloxyalkyl carbamate prodrugs and intermediates thereof
Publication number
20050222431
Publication date
Oct 6, 2005
XenoPort, Inc.
Mark A. Gallop
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Crystalline form of y-aminobutyric acid analog
Publication number
20050154057
Publication date
Jul 14, 2005
Tono Estrada
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Methods for synthesis of acyloxyalkyl derivatives of GABA analogs
Publication number
20040014940
Publication date
Jan 22, 2004
Stephen P. Raillard
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Fast scale-up using solid phase chemistry
Publication number
20020028466
Publication date
Mar 7, 2002
Stephen P. Raillard
C07 - ORGANIC CHEMISTRY