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Susana Conde-Ceide
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Toledo, ES
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last 30 patents
Information
Patent Grant
6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one compounds and their use...
Patent number
10,668,065
Issue date
Jun 2, 2020
JANSSEN PHARMACEUTICA NV
Susana Conde-Ceide
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
6,7-dihydropyrazolo[1,5-α]pyrazin-4(5H)-one compounds and their use...
Patent number
10,519,162
Issue date
Dec 31, 2019
JANSSEN PHARMACEUTICA NV
Sergio-Alvar Alonso-de Diego
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6,7-dihydropyrazolo[1,5-a]pyrazin-4(5H)-one compounds and their use...
Patent number
10,220,032
Issue date
Mar 5, 2019
JANSSEN PHARMACEUTICA NV
Susana Conde-Ceide
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6,7-dihydropyrazolo[1,5-α]pyrazin-4(5H)-one compounds and their use...
Patent number
10,017,514
Issue date
Jul 10, 2018
JANSSEN PHARMACEUTICA NV
Susana Conde-Ceide
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted 6,7-dihydropyrazolo[1,5-a] pyrazines as negative allost...
Patent number
10,005,785
Issue date
Jun 26, 2018
Janssen Pharmaceutica N.V.
Sergio-Alvar Alonso-de Diego
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Inhibitors of phosphodiesterase 10 enzyme
Patent number
9,550,784
Issue date
Jan 24, 2017
Beerse Pharmaceutica NV
Laurent Christian L. Leclercq
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazolo[1,5-a]pyrazines as mGluR5 receptor modulators
Patent number
9,255,103
Issue date
Feb 9, 2016
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic oxazole and thiazole compounds and their use as allosteric...
Patent number
9,090,632
Issue date
Jul 28, 2015
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic thiazoles as allosteric modulators of mGluR5 receptors
Patent number
9,040,707
Issue date
May 26, 2015
JANSSEN PHARMACEUTICA NV
Gregor James MacDonald
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted bicyclic alkoxy pyrazole analogs as allosteric modulato...
Patent number
9,029,366
Issue date
May 12, 2015
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted bicyclic alkoxy pyrazole analogs as allosteric modulato...
Patent number
8,901,125
Issue date
Dec 2, 2014
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted imidazopyrimidin-5(6H)-ones as allosteric modulators of...
Patent number
8,865,725
Issue date
Oct 21, 2014
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo[1,2-a]pyrazine derivatives and their use for the prevention...
Patent number
8,859,543
Issue date
Oct 14, 2014
JANSSEN PHARMACEUTICA NV
José Manuel Bartolomé-Nebreda
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Naphthyridinone analogs as mGluR5 positive allosteric modulators
Patent number
8,853,237
Issue date
Oct 7, 2014
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Imidazo[1,2-b]pyridazine derivatives and their use as PDE10 inhibitors
Patent number
8,716,282
Issue date
May 6, 2014
JANSSEN PHARMACEUTICA NV
Joaquin Pastor-Fernández
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dihydronaphthyridinyl(organo)methanone analogs as positive alloster...
Patent number
8,710,074
Issue date
Apr 29, 2014
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazolo[1,5-A]pyrazine compounds as allosteric modulat...
Patent number
8,703,946
Issue date
Apr 22, 2014
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic triazole and pyrazole lactams as allosteric modulators of...
Patent number
8,592,422
Issue date
Nov 26, 2013
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted 6-(1-piperazinyl)-pyridazines as 5-HT6 receptor antagon...
Patent number
8,530,474
Issue date
Sep 10, 2013
JANSSEN PHARMACEUTICA NV
José Manuel Bartolomé-Nebreda
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
OGA INHIBITOR COMPOUNDS
Publication number
20210277015
Publication date
Sep 9, 2021
Janssen Pharmaceutica N.V.
José Manuel Bartolomé-Nebreda
C07 - ORGANIC CHEMISTRY
Information
Patent Application
OGA INHIBITOR COMPOUNDS
Publication number
20210122763
Publication date
Apr 29, 2021
Janssen Pharmaceutica N.V.
José Manuel Bartolomé-Nebreda
C07 - ORGANIC CHEMISTRY
Information
Patent Application
OGA INHIBITOR COMPOUNDS
Publication number
20210115040
Publication date
Apr 22, 2021
Janssen Pharmaceutica N.V.
José Manuel Bartolomé-Nebreda
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE...
Publication number
20200261450
Publication date
Aug 20, 2020
Janssen Pharmaceutica N.V.
Susana Conde-Ceide
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE...
Publication number
20190160061
Publication date
May 30, 2019
Susana Conde-Ceide
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE...
Publication number
20180258096
Publication date
Sep 13, 2018
Janssen Pharmaceutica N.V.
Sergio-Alvar Alonso-de Diego
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE...
Publication number
20170273976
Publication date
Sep 28, 2017
Janssen Pharmaceutica N.V.
Susana Conde-Ceide
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE...
Publication number
20170267682
Publication date
Sep 21, 2017
Janssen Pharmaceutica N.V.
Susana Conde-Ceide
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE...
Publication number
20170217971
Publication date
Aug 3, 2017
Janssen Pharmaceutica N.V.
Sergio-Alvar Alonso-de Diego
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED BICYCLIC ALKOXY PYRAZOLE ANALOGS AS ALLOSTERIC MODULATO...
Publication number
20150216863
Publication date
Aug 6, 2015
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INHIBITORS OF PHOSPHODIESTERASE 10 ENZYME
Publication number
20150203498
Publication date
Jul 23, 2015
Janssen Pharmaceutica N.V.
Laurent Christian L. Leclercq
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED IMIDAZOPYRIMIDIN-5(6H)-ONES AS ALLOSTERIC MODULATORS OF...
Publication number
20140329838
Publication date
Nov 6, 2014
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC PYRAZOLE COMPOUNDS AS ALLOSTERIC MODULATORS OF MGLUR5 RECE...
Publication number
20140213593
Publication date
Jul 31, 2014
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BICYCLIC CYCLOALKYL PYRAZOLE LACTAM ANALOGS AS ALLOSTER...
Publication number
20130345204
Publication date
Dec 26, 2013
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BICYCLIC ALKOXY PYRAZOLE ANALOGS AS ALLOSTERIC MODULATO...
Publication number
20130345206
Publication date
Dec 26, 2013
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BICYCLIC ARALKYL PYRAZOLE LACTAM ANALOGS AS ALLOSTERIC...
Publication number
20130345205
Publication date
Dec 26, 2013
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BICYCLIC ALKOXY PYRAZOLE ANALOGS AS ALLOSTERIC MODULATO...
Publication number
20130345203
Publication date
Dec 26, 2013
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC OXAZOLE AND THIAZOLE COMPOUNDS AND THEIR USE AS ALLOSTERIC...
Publication number
20130261107
Publication date
Oct 3, 2013
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC OXAZOLE LACTAMS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS
Publication number
20130252943
Publication date
Sep 26, 2013
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED IMIDAZOPYRIMIDIN-5(6H)-ONES AS ALLOSTERIC MODULATORS OF...
Publication number
20130245043
Publication date
Sep 19, 2013
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZO[1,2-a]PYRAZINE DERIVATIVES AND THEIR USE FOR THE PREVENTION...
Publication number
20120329792
Publication date
Dec 27, 2012
Janssen Pharmaceutica N.V.
José Manuel Bartolomé-Nebreda
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC PYRAZOLE COMPOUNDS AS ALLOSTERIC MODULATORS OF MGLUR5 RECE...
Publication number
20120295913
Publication date
Nov 22, 2012
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC THIAZOLES AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS
Publication number
20120258955
Publication date
Oct 11, 2012
Janssen Pharmaceutica N.V.
Gregor James MacDonald
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC TRIAZOLE AND PYRAZOLE LACTAMS AS ALLOSTERIC MODULATORS OF...
Publication number
20120225844
Publication date
Sep 6, 2012
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AND THEIR USE AS PDE10 INHIBITORS
Publication number
20120220581
Publication date
Aug 30, 2012
Janssen-Cilag, S.A.
Joaquin Pastor-Fernández
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DIHYDRONAPHTHYRIDINYL(ORGANO)METHANONE ANALOGS AS POSITIVE ALLOSTER...
Publication number
20120178776
Publication date
Jul 12, 2012
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NAPHTHYRIDINONE ANALOGS AS MGLUR5 POSITIVE ALLOSTERIC MODULATORS
Publication number
20120172391
Publication date
Jul 5, 2012
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES AND THEIR USE AS PDE10 INHIBITORS
Publication number
20110269752
Publication date
Nov 3, 2011
Joaquin Pastor-Fernández
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED 6-(1-PIPERAZINYL)-PYRIDAZINES AS 5-HT6 RECEPTOR ANTAGON...
Publication number
20110112107
Publication date
May 12, 2011
José Manuel Bartolomé-Nebreda
C07 - ORGANIC CHEMISTRY