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Theodore M. Kamenecka
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Palm Beach Gardens, FL, US
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Patents Grants
last 30 patents
Information
Patent Grant
Halo-substituted piperidines as orexin receptor modulators
Patent number
12,084,437
Issue date
Sep 10, 2024
Astrazeneca AB
Theodore M. Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Nonmuscle myosin II inhibitors for substance use relapse
Patent number
11,649,234
Issue date
May 16, 2023
The University of Florida Research Foundation, Inc.
Courtney Miller
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Halo-substituted piperidines as orexin receptor modulators
Patent number
11,434,236
Issue date
Sep 6, 2022
Astrazeneca AB
Theodore M. Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Chemical uncouplers of respiration and methods of use thereof
Patent number
11,365,177
Issue date
Jun 21, 2022
Dana-Farber Cancer Institute, Inc.
Bruce M. Spiegelman
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Selective inhibition of gluconeogenic activity
Patent number
11,247,970
Issue date
Feb 15, 2022
Dana-Farber Cancer Institute, Inc.
Pere Puigserver
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Halo-substituted piperidines as orexin receptor modulators
Patent number
10,894,789
Issue date
Jan 19, 2021
Astrazeneca AB
Theodore M. Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Small molecule analogs of the nemo binding peptide
Patent number
10,758,522
Issue date
Sep 1, 2020
The Scripps Research Institute
Paul Robbins
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
PPARG modulators for the treatment of osteoporosis
Patent number
10,744,117
Issue date
Aug 18, 2020
The Scripps Research Institute
Patrick R. Griffin
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Difluoropyrrolidines as orexin receptor modulators
Patent number
10,221,170
Issue date
Mar 5, 2019
Eolas Therapeutics, Inc.
Theodore M. Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
PPARG modulators for treatment of osteoporosis
Patent number
10,016,394
Issue date
Jul 10, 2018
The Scripps Research Institute
Patrick R. Griffin
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted prolines/piperidines as orexin receptor antagonists
Patent number
9,896,452
Issue date
Feb 20, 2018
Eolas Therapeutics, Inc.
Theodore M. Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Modulators of the nuclear hormone receptor ROR
Patent number
9,586,928
Issue date
Mar 7, 2017
The Scripps Research Institute
Theodore Mark Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted prolines / piperidines as orexin receptor antagonists
Patent number
9,499,517
Issue date
Nov 22, 2016
Eolas Therapeutics, Inc.
Theodore M. Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted prolines/piperidines as orexin receptor antagonists
Patent number
9,440,982
Issue date
Sep 13, 2016
Eolas Therapeutics, Inc.
Theodore M. Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
N-biphenylmethylbenzimidazole modulators of PPARG
Patent number
9,309,227
Issue date
Apr 12, 2016
The Scripps Research Institute
Theodore Mark Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
N-benzylindole modulators of PPARG
Patent number
9,051,265
Issue date
Jun 9, 2015
The Scripps Research Institute
Theodore Mark Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrimidinyl-amines as protein kinase inhibitors
Patent number
9,018,205
Issue date
Apr 28, 2015
The Scripps Research Institute
Theodore Mark Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
N-biphenylmethylindole modulators of PPARG
Patent number
8,957,093
Issue date
Feb 17, 2015
The Scripps Research Institute
Theodore Mark Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrimidinyl-amines as protein kinase inhibitors
Patent number
8,530,480
Issue date
Sep 10, 2013
The Scripps Research Institute
Theodore Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzazole potentiators of metabotropic glutamate receptors
Patent number
7,960,417
Issue date
Jun 14, 2011
Merck Sharp & Dohme Corp.
Steven P. Govek
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzoxazinyl-amidocyclopentyl-heterocyclic modulators of chemokine...
Patent number
7,700,591
Issue date
Apr 20, 2010
Merck & Co., Inc.
Stephen D. Goble
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-arylsulfonyl-proline derivatives as potent cell adhes...
Patent number
6,943,180
Issue date
Sep 13, 2005
Merck & Co., Inc.
George Doherty
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
HALO-SUBSTITUTED PIPERIDINES AS OREXIN RECEPTOR MODULATORS
Publication number
20240400550
Publication date
Dec 5, 2024
AstraZeneca AB
Theodore M. Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PPARG Modulators for the Treatment of Osteoporosis
Publication number
20240009169
Publication date
Jan 11, 2024
University of Florida Research Foundation, Incorporated
Patrick R. Griffin
C07 - ORGANIC CHEMISTRY
Information
Patent Application
REV-ERB AGONISTS FOR THE TREATMENT OF TH17-MEDIATED INFLAMMATORY DI...
Publication number
20230339886
Publication date
Oct 26, 2023
University of Florida Research Foundation, Incorporated
Theodore Mark Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Application
THERAPEUTIC USES OF GLUCOCORTICOIDS WITH ANABOLIC EFFECTS IN SKELET...
Publication number
20230263808
Publication date
Aug 24, 2023
University of Florida Research Foundation, Incorporated
Kendall Nettles
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NONMUSCLE MYOSIN II INHIBITORS
Publication number
20230227452
Publication date
Jul 20, 2023
The University of Florida Research Foundation, Inc.
Courtney Anne MILLER
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PPARG Modulators for the Treatment of Osteoporosis
Publication number
20230072933
Publication date
Mar 9, 2023
The Scripps Research Institute
Patrick R. Griffin
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HALO-SUBSTITUTED PIPERIDINES AS OREXIN RECEPTOR MODULATORS
Publication number
20220380359
Publication date
Dec 1, 2022
AstraZeneca AB
Theodore M. Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NONMUSCLE MYOSIN II INHIBITORS FOR SUBSTANCE USE RELAPSE
Publication number
20210317117
Publication date
Oct 14, 2021
The Scripps Research Institute
Courtney Miller
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HALO-SUBSTITUTED PIPERIDINES AS OREXIN RECEPTOR MODULATORS
Publication number
20210214348
Publication date
Jul 15, 2021
AstraZeneca AB
Theodore M. Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SELECTIVE INHIBITION OF GLUCONEOGENIC ACTIVITY
Publication number
20200317620
Publication date
Oct 8, 2020
Dana-Farber Cancer Institute, Inc.
Pere PUIGSERVER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CHEMICAL UNCOUPLERS OF RESPIRATION AND METHODS OF USE THEREOF
Publication number
20200317613
Publication date
Oct 8, 2020
Dana-Farber Cancer Institute, Inc.
Bruce M. Spiegelman
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HALO-SUBSTITUTED PIPERIDINES AS OREXIN RECEPTOR MODULATORS
Publication number
20190135800
Publication date
May 9, 2019
AstraZeneca AB
Theodore M. Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PPARG Modulators for the Treatment of Osteoporosis
Publication number
20180369196
Publication date
Dec 27, 2018
The Scripps Research Institute
Patrick R. Griffin
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Small Molecule Analogs of the Nemo Binding Peptide
Publication number
20180169078
Publication date
Jun 21, 2018
The Scripps Research Institute
Paul Robbins
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
DIFLUOROPYRROLIDINES AS OREXIN RECEPTOR MODULATORS
Publication number
20170226103
Publication date
Aug 10, 2017
Eolas Therapeutics, Inc.
Theodore M. Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PROLINES / PIPERIDINES AS OREXIN RECEPTOR ANTAGONISTS
Publication number
20170101410
Publication date
Apr 13, 2017
Eolas Therapeutics, Inc.
Theodore M. Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PPARG MODULATORS FOR TREATMENT OF OSTEOPOROSIS
Publication number
20170035730
Publication date
Feb 9, 2017
The Scripps Research Institute
Patrick R. Griffin
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRIMIDINYL-AMINES AS PROTEIN KINASE INHIBITORS
Publication number
20150232429
Publication date
Aug 20, 2015
The Scripps Research Institute
Theodore Mark Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-BIPHENYLMETHYLBENZIMIDAZOLE MODULATORS OF PPARG
Publication number
20150141464
Publication date
May 21, 2015
Theodore Mark Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PROLINES / PIPERIDINES AS OREXIN RECEPTOR ANTAGONISTS
Publication number
20140364433
Publication date
Dec 11, 2014
Theodore M. KAMENECKA
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PROLINES / PIPERIDINES AS OREXIN RECEPTOR ANTAGONISTS
Publication number
20140364432
Publication date
Dec 11, 2014
Theodore M. KAMENECKA
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
N-ARYLYLMETHYLINDAZOLE MODULATORS OF PPARG
Publication number
20140288090
Publication date
Sep 25, 2014
Theodore Mark Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
N-BENZYLBENZIMIDAZOLE MODULATORS OF PPARG
Publication number
20140249196
Publication date
Sep 4, 2014
Theodore Mark Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MODULATORS OF THE NUCLEAR HORMONE RECEPTOR ROR
Publication number
20140187554
Publication date
Jul 3, 2014
The Scripps Research Institute
Theodore Mark Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRIMIDINYL-AMINES AS PROTEIN KINASE INHIBITORS
Publication number
20130231336
Publication date
Sep 5, 2013
The Scripps Research Institute
Theodore Mark Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-BENZYLINDOLE MODULATORS OF PPARG
Publication number
20120309769
Publication date
Dec 6, 2012
SCRIPPS RESEARCH INSTITUTE, THE
Theodore Mark Kamenecka
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
N-BIPHENYLMETHYLINDOLE MODULATORS OF PPARG
Publication number
20120309757
Publication date
Dec 6, 2012
SCRIPPS RESEARCH INSTITUTE, THE
Theodore Mark Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRIMIDINYL-AMINES AS PROTEIN KINASE INHIBITORS
Publication number
20100298312
Publication date
Nov 25, 2010
The Scripps Research Institute
Theodore M. Kamenecka
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Indanone Potentiators of Metabotropic Glutamate Receptors
Publication number
20080312286
Publication date
Dec 18, 2008
Anthony B. Pinkerton
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Heterocyclic Acetophenone Potentiators of Metabotropic Glutamate Re...
Publication number
20080293684
Publication date
Nov 27, 2008
Anthony B Pinkerton
C07 - ORGANIC CHEMISTRY