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Timothy Paul Burkholder
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Carmel, IN, US
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Patents Grants
last 30 patents
Information
Patent Grant
7-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds as...
Patent number
11,649,247
Issue date
May 16, 2023
Eli Lilly and Company
Renato Alejandro Bauer
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
7-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds as...
Patent number
11,629,156
Issue date
Apr 18, 2023
Eli Lilly and Company
Renato Alejandro Bauer
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
7-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds as...
Patent number
11,001,596
Issue date
May 11, 2021
Eli Lilly and Company
Renato Alejandro Bauer
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Mutant IDH1 inhibitors
Patent number
10,696,665
Issue date
Jun 30, 2020
Eli Lilly and Company
Wenceslao Lumeras Amador
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
7-phenylethylamino-4H-pyrimido[4,5-d][1,3]oxazin-2-one compounds an...
Patent number
10,253,041
Issue date
Apr 9, 2019
Eli Lilly and Company
Renato A. Bauer
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Inhibitor of JAK1 and JAK2
Patent number
9,062,050
Issue date
Jun 23, 2015
Eli Lilly and Company
Timothy Paul Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
AKT inhibitors
Patent number
8,436,002
Issue date
May 7, 2013
Eli Lilly and Company
Douglas Wade Beight
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Purine derivatives as kinase inhibitors
Patent number
8,058,425
Issue date
Nov 15, 2011
Eli Lilly and Company
Thomas Albert Engler
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Amino pyrazole compound
Patent number
7,897,600
Issue date
Mar 1, 2011
Eli Lilly and Company
Timothy Paul Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo[1,2-A]pyridine compounds as VEGF-R2 inhibitors
Patent number
7,666,879
Issue date
Feb 23, 2010
Eli Lilly and Company
David Anthony Barda
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrole-2, 5dione derivatives and their used as GSK-3 inhibitors
Patent number
7,405,305
Issue date
Jul 29, 2008
Eli Lilly and Company
Pamela Ann Albaugh
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds as pharmaceutical agents
Patent number
7,405,299
Issue date
Jul 29, 2008
Eli Lilly and Company
Douglas Wade Beight
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aminoalkylbenzofurans as serotonin (5-HT(2c)) agonists
Patent number
7,045,545
Issue date
May 16, 2006
Eli Lilly and Company
Karin Briner
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzofurylpiperazines and benzofurylhomopiperazines: serotonin agon...
Patent number
6,967,201
Issue date
Nov 22, 2005
Eli Lilly and Company
Karin Briner
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Serotonergic benzofurans
Patent number
6,881,733
Issue date
Apr 19, 2005
Eli Lilly and Company
Karin Briner
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzofurylpiperazine serotonin agonists
Patent number
6,638,936
Issue date
Oct 28, 2003
Eli Lilly and Company
Karin Briner
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted piperidines useful for the treatment of allergic diseases
Patent number
6,329,392
Issue date
Dec 11, 2001
Aventis Pharmaceuticals, Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Carboxy substituted acylic carboxamide derivatives
Patent number
6,316,445
Issue date
Nov 13, 2001
Aventis Pharmaceuticals Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 4-(1H-benzimidazol-2-yl-amino)piperidines useful for th...
Patent number
6,211,199
Issue date
Apr 3, 2001
Aventis Pharmaceuticals Inc.
John M. Kane
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 4-(1H-benzimidazol-2-yl)[1,4]diazepanes...
Patent number
6,194,406
Issue date
Feb 27, 2001
Aventis Pharmaceuticals Inc.
John M. Kane
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Carboxysubstituted cyclic carboxamide derivatives
Patent number
5,977,139
Issue date
Nov 2, 1999
Hoechst Marion Roussel, Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic substituted piperazinone derivatives
Patent number
5,864,045
Issue date
Jan 26, 1999
Hoechst Marion Roussel, Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic substituted pyrrolidine amide derivatives
Patent number
5,861,417
Issue date
Jan 19, 1999
Hoechst Marion Roussel, Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrrolidin-3-yl-alkyl-piperidines
Patent number
5,861,416
Issue date
Jan 19, 1999
Merrell Pharmaceuticals Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic substituted piperazinone derivatives
Patent number
5,840,726
Issue date
Nov 24, 1998
Hoechst Marion Roussel Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrrolidin-3-yl-alkyl-piperidines
Patent number
5,824,690
Issue date
Oct 20, 1998
Hoechst Marion Roussel Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted piperazine derivatives
Patent number
5,672,602
Issue date
Sep 30, 1997
Hoechst Marion Roussel, Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrrolidin-3-yl-alkyl-piperidines
Patent number
5,661,160
Issue date
Aug 26, 1997
Merrell Pharmaceuticals Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrrolidin-3-yl-alkyl-piperidines
Patent number
5,648,366
Issue date
Jul 15, 1997
Merrell Pharmaceuticals Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrrolidin-3-yl-alkyl-piperidines
Patent number
5,635,510
Issue date
Jun 3, 1997
Merrell Pharmaceuticals Inc.
Timothy P. Burkholder
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
7-PHENYLETHYLAMINO-4H-PYRIMIDO[4,5-D][1,3]OXAZIN-2-ONE COMPOUNDS AS...
Publication number
20210230185
Publication date
Jul 29, 2021
Eli Lilly and Company
Renato Alejandro BAUER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
7-PHENYLETHYLAMINO-4H-PYRIMIDO[4,5-D][1,3]OXAZIN-2-ONE COMPOUNDS AS...
Publication number
20210206780
Publication date
Jul 8, 2021
Eli Lilly and Company
Renato Alejandro BAUER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
7-PHENYLETHYLAMINO-4H-PYRIMIDO[4,5-D][1,3]OXAZIN-2-ONE COMPOUNDS AS...
Publication number
20200079791
Publication date
Mar 12, 2020
Eli Lilly and Company
Renato Alejandro BAUER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MUTANT IDH1 INHIBITORS
Publication number
20190292175
Publication date
Sep 26, 2019
Eli Lilly and Company
Wenceslao LUMERAS AMADOR
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
7-PHENYLETHYLAMINO-4H-PYRIMIDO[4,5-D][1,3]OXAZIN-2-ONE COMPOUNDS AN...
Publication number
20180118759
Publication date
May 3, 2018
Eli Lilly and Company
Renato A. Bauer
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL PYRIDYLOXYACETYL TETRAHYDROISOQUINOLINE COMPOUNDS USEFUL AS N...
Publication number
20160229835
Publication date
Aug 11, 2016
Eli Lilly and Company
Timothy Paul Burkholder
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INHIBITOR OF JAK1 AND JAK2
Publication number
20150133490
Publication date
May 14, 2015
Eli Lilly and Company
Timothy Paul Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AKT INHIBITORS
Publication number
20120149684
Publication date
Jun 14, 2012
Eli Lilly and Company
Douglas Wade Beight
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PURINE DERIVATIVES AS KINASE INHIBITORS
Publication number
20110294792
Publication date
Dec 1, 2011
Eli Lilly and Company
Thomas Albert Engler
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PURINE DERIVATIVES AS KINASE INHIBITORS
Publication number
20110207721
Publication date
Aug 25, 2011
Eli Lilly and Company
Thomas Albert Engler
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMINO PYRAZOLE COMPOUND
Publication number
20100286139
Publication date
Nov 11, 2010
Eli Lilly and Company
Timothy Paul Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMINO PYRAZOLE COMPOUND
Publication number
20100152181
Publication date
Jun 17, 2010
Eli Lilly and Company
Timothy Paul Burkholder
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMIDAZO[1,2-A]PYRIDINE COMPOUNDS AS VEGF-R2 INHIBITORS
Publication number
20090227622
Publication date
Sep 10, 2009
David Anthony Barda
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PURINE DERIVATIVES AS KINASE INHIBITORS
Publication number
20090105229
Publication date
Apr 23, 2009
Thomas Albert Engler
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel compounds as pharmaceutical agents
Publication number
20060058295
Publication date
Mar 16, 2006
Eli Lilly and Company
Douglas Wade Beight
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Kinase inhibitors
Publication number
20050288321
Publication date
Dec 29, 2005
Pamela Ann Albaugh
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Purine derivatives as kinase inhibitors
Publication number
20050090483
Publication date
Apr 28, 2005
Eli Lilly and Company
Thomas Albert Engler
C07 - ORGANIC CHEMISTRY