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William M. Leong
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Westfield, NJ, US
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Patents Grants
last 30 patents
Information
Patent Grant
Crystalline fumarate salts of n-ethyl-2-(5-fluoro-1H-indol-3-yl)-n-...
Patent number
12,180,158
Issue date
Dec 31, 2024
Gilgamesh Pharmaceuticals, Inc.
Andrew Carry Kruegel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Crystalline hydrochloride salts of N-ethyl-2-(5-fluoro-1H-indol-3-y...
Patent number
12,157,722
Issue date
Dec 3, 2024
Gilgamesh Pharmaceuticals, Inc.
Andrew Carry Kruegel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Crystalline salts of N-ethyl-(5-fluoro-1H-indol-3-yl)-N-methylethan...
Patent number
12,129,234
Issue date
Oct 29, 2024
Gilgamesh Pharmaceuticals, Inc.
Andrew Carry Kruegel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Isotopologues of 5-azacytidine
Patent number
10,646,503
Issue date
May 12, 2020
Celgene Corporation
John F. Traverse
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Isotopologues of 5-azacytidine
Patent number
10,463,683
Issue date
Nov 5, 2019
Celgene Corporation
John F. Traverse
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Isotopologues of 5-azacytidine
Patent number
10,220,050
Issue date
Mar 5, 2019
Celgene Corporation
John F. Traverse
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Processes for the preparation of (s)-3-(4-((4-(morpholinomethyl)ben...
Patent number
9,975,872
Issue date
May 22, 2018
Celgene Corporation
John F. Traverse
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Solid forms of 3-(5-amino-2-methyl-4-oxo-4H-quinazolin-3-yl)-piperi...
Patent number
9,969,713
Issue date
May 15, 2018
Celgene Corporation
George W. Muller
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pharmaceutical formulations, processes, solid forms and methods of...
Patent number
9,827,243
Issue date
Nov 28, 2017
Signal Pharmaceuticals, LLC
Matthew Michael Kreilein
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Solid forms of 3-(5-amino-2-methyl-4-oxo-4H-quinazolin-3-yl)-piperi...
Patent number
9,751,853
Issue date
Sep 5, 2017
Celgene Corporation
George W. Muller
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Isotopologues of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4H)-yl) pipe...
Patent number
9,682,952
Issue date
Jun 20, 2017
Celgene Corporation
Hon-Wah Man
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pharmaceutical compositions of 7-(6-(2-hydroxypropan-2-yl)pyridin-3...
Patent number
9,403,829
Issue date
Aug 2, 2016
Signal Pharmaceuticals, LLC
Terrence Joseph Connolly
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pharmaceutical formulations, processes, solid forms and methods of...
Patent number
9,359,364
Issue date
Jun 7, 2016
Signal Pharmaceuticals, LLC
Anil Menon
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Processes for the preparation of (S)-3-(4- (4-(morpholinomethyl)ben...
Patent number
9,309,220
Issue date
Apr 12, 2016
Celgene Corporation
John F. Traverse
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Synthesis of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4H)-yl)piperidin...
Patent number
9,303,014
Issue date
Apr 5, 2016
Celgene Corporation
Alexander L. Ruchelman
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Synthesis of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4H)-yl)piperidin...
Patent number
9,266,858
Issue date
Feb 23, 2016
Celgene Corporation
Alexander L. Ruchelman
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Solid forms of 3-(5-amino-2-methyl-4-oxo-4H-quinazolin-3-yl)-piperi...
Patent number
9,249,121
Issue date
Feb 2, 2016
Celgene Corporation
George W. Muller
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Asymmetric synthetic processes for the preparation of aminosulfone...
Patent number
9,126,906
Issue date
Sep 8, 2015
Celgene Corporation
Terrence J. Connolly
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of synthesis and purification of heteroaryl compounds
Patent number
9,079,900
Issue date
Jul 14, 2015
Signal Pharmaceuticals, LLC
Roy L. Harris
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Synthesis of 3-(5-amino-2-methyl-4-oxoquinazolin-3(4H)-yl)piperidin...
Patent number
9,067,912
Issue date
Jun 30, 2015
Celgene Corporation
Alexander L. Ruchelman
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Solid forms of 3-(5-amino-2-methyl-4-oxo-4H-quinazolin-3-yl)-piperi...
Patent number
8,802,685
Issue date
Aug 12, 2014
Celgene Corporation
George Muller
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of synthesis and purification of heteroaryl compounds
Patent number
8,686,135
Issue date
Apr 1, 2014
Signal Pharmaceuticals, LLC
Patrick Anthony Jokiel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Enantio- and stereo specific synthesis of β-amino-α-hydroxy amides
Patent number
8,680,294
Issue date
Mar 25, 2014
Merck Sharp & Dohme Corp.
John Traverse
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Process for preparing a 2-alkynyl substituted 5-amino-pyrazolo-[4,3...
Patent number
8,598,343
Issue date
Dec 3, 2013
Merck Sharp & Dohme Corp.
Shen-Chun Kuo
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of synthesis and purification of heteroaryl compounds
Patent number
8,569,494
Issue date
Oct 29, 2013
Signal Pharmaceuticals, LLC
Roy L. Harris
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Synthesis of CCR5 receptor antagonists
Patent number
7,728,135
Issue date
Jun 1, 2010
Schering Corporation
Xiongwei Shi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Preparation of pharmaceutical salts of piperazine compounds
Patent number
7,521,452
Issue date
Apr 21, 2009
Schering Corporation
Wenxue Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Synthesis of piperidine and piperazine compounds as CCR5 antagonists
Patent number
6,992,189
Issue date
Jan 31, 2006
Schering Corporation
William Leong
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Crystalline antifungal polymorph
Patent number
6,958,337
Issue date
Oct 25, 2005
Schering Corporation
David R. Andrews
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Preparation of rotamer mixtures of pharmaceutical salts
Patent number
6,936,718
Issue date
Aug 30, 2005
Schering Corporation
Minzhang Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
CRYSTALLINE HYDROCHLORIDE SALTS OF N-ETHYL-2-(5-FLUORO-1H-INDOL-3-Y...
Publication number
20240400509
Publication date
Dec 5, 2024
Gilgamesh Pharmaceuticals, Inc.
Andrew Carry Kruegel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESS FOR THE PRODUCTION OF SUBSTITUTED 2-[2-(PHENYL)ETHYLAMINO]A...
Publication number
20220185766
Publication date
Jun 16, 2022
Newron Pharmaceuticals S.p.A.
William Leong
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ISOTOPOLOGUES OF 5-AZACYTIDINE
Publication number
20200316099
Publication date
Oct 8, 2020
Celgene Corporation
John F. Traverse
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ISOTOPOLOGUES OF 5-AZACYTIDINE
Publication number
20200101095
Publication date
Apr 2, 2020
Celgene Corporation
John F. Traverse
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ISOTOPOLOGUES OF 5-AZACYTIDINE
Publication number
20190231803
Publication date
Aug 1, 2019
Celgene Corporation
John F. Traverse
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SOLID FORMS OF 3-(5-AMINO-2-METHYL-4-OXO-4H-QUINAZOLIN-3-YL)-PIPERI...
Publication number
20180305333
Publication date
Oct 25, 2018
Celgene Corporation
George W. Muller
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ISOTOPOLOGUES OF 5-AZACYTIDINE
Publication number
20180153916
Publication date
Jun 7, 2018
Celgene Corporation
John F. Traverse
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ISOTOPOLOGUES OF 3-(5-AMINO-2-METHYL-4-OXOQUINAZOLIN-3(4H)-YL)PIPER...
Publication number
20180093965
Publication date
Apr 5, 2018
Celgene Corporation
Hon-Wah Man
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHARMACEUTICAL FORMULATIONS, PROCESSES, SOLID FORMS AND METHODS OF...
Publication number
20180042924
Publication date
Feb 15, 2018
Signal Pharmaceuticals, LLC.
Anil Menon
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SOLID FORMS OF 3-(5-AMINO-2-METHYL-4-OXO-4H-QUINAZOLIN-3-YL)-PIPERI...
Publication number
20170342050
Publication date
Nov 30, 2017
Celgene Corporation
George W. MULLER
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR THE PREPARATION OF (S)-3-(4-((4-(MORPHOLINOMETHYL)BEN...
Publication number
20160251333
Publication date
Sep 1, 2016
Celgene Corporation
John F. Traverse
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHARMACEUTICAL FORMULATIONS, PROCESSES, SOLID FORMS AND METHODS OF...
Publication number
20160250210
Publication date
Sep 1, 2016
Signal Pharmaceuticals, LLC.
Anil Menon
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SOLID FORMS OF 3-(5-AMINO-2-METHYL-4-OXO-4H-QUINAZOLIN-3-YL)-PIPERI...
Publication number
20160214957
Publication date
Jul 28, 2016
Celgene Corporation
George W. MULLER
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SYNTHESIS OF 3-(5-AMINO-2-METHYL-4-OXOQUINAZOLIN-3(4H)-YL)PIPERIDIN...
Publication number
20160009685
Publication date
Jan 14, 2016
Celgene Corporation
Alexander L. RUCHELMAN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SYNTHESIS OF 3-(5-AMINO-2-METHYL-4-OXOQUINAZOLIN-3(4H)-YL)PIPERIDIN...
Publication number
20150274694
Publication date
Oct 1, 2015
Celgene Corporation
Alexander L. RUCHELMAN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ISOTOPOLOGUES OF 3-(5-AMINO-2-METHYL-4-OXOQUINAZOLIN-3(4H)-YL) PIPE...
Publication number
20150203469
Publication date
Jul 23, 2015
Celgene Corporation
Hon-Wah Man
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ISOTOPOLOGUES OF 5-AZACYTIDINE
Publication number
20150056280
Publication date
Feb 26, 2015
Celgene Corporation
John F. TRAVERSE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SOLID FORMS OF 3-(5-AMINO-2-METHYL-4-OXO-4H-QUINAZOLIN-3-YL)-PIPERI...
Publication number
20140378484
Publication date
Dec 25, 2014
George W. MULLER
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SYNTHESIS OF 3-(5-AMINO-2-METHYL-4-OXOQUINAZOLIN-3(4H)-YL)PIPERIDIN...
Publication number
20140330016
Publication date
Nov 6, 2014
Celgene Corporation
Alexander L. RUCHELMAN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHARMACEUTICAL FORMULATIONS, PROCESSES, SOLID FORMS AND METHODS OF...
Publication number
20140315908
Publication date
Oct 23, 2014
Signal Pharmaceuticals, LLC.
Anil Menon
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
METHODS OF SYNTHESIS AND PURIFICATION OF HETEROARYL COMPOUNDS
Publication number
20140155593
Publication date
Jun 5, 2014
Signal Pharmaceuticals, LLC.
Roy L. Harris
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES FOR THE PREPARATION OF (S)-3-(4-((4-(MORPHOLINOMETHYL)BEN...
Publication number
20140046058
Publication date
Feb 13, 2014
Celgene Corporation
John F. Traverse
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHODS OF SYNTHESIS AND PURIFICATION OF HETEROARYL COMPOUNDS
Publication number
20130245254
Publication date
Sep 19, 2013
Signal Pharmaceuticals, LLC.
Roy L. Harris
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ASYMMETRIC SYNTHETIC PROCESSES FOR THE PREPARATION OF AMINOSULFONE...
Publication number
20130217919
Publication date
Aug 22, 2013
Celgene Corporation
Terrence J. CONNOLLY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PHARMACEUTICAL COMPOSITIONS OF 7-(6-(2-HYDROXYPROPAN-2-YL)PYRIDIN-3...
Publication number
20130142873
Publication date
Jun 6, 2013
Signal Pharmaceuticals, LLC.
MAHMOUD S. ASSAF
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SOLID FORMS OF 3-(5-AMINO-2-METHYL-4-OXO-4H-QUINAZOLIN-3-YL)-PIPERI...
Publication number
20120232100
Publication date
Sep 13, 2012
George Muller
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESS FOR PREPARING A 2-ALKYNYL SUBSTITUTED 5-AMINO-PYRAZOLO-[4,3...
Publication number
20120220769
Publication date
Aug 30, 2012
Schering Corporation
Shen-Chun Kuo
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ENANTIO- AND STEREO-SPECIFIC SYNTHESES OF BETA-AMINO-ALPHA- HYDROXY...
Publication number
20120178942
Publication date
Jul 12, 2012
John Traverse
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESS FOR PREPARING CCR-5 RECEPTOR ANTAGONISTS UTILIZING 4-SUBSTI...
Publication number
20100063280
Publication date
Mar 11, 2010
Schering Corporation
John F. Traverse
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SYNTHESIS OF CCR5 RECEPTOR ANTAGONISTS
Publication number
20100036125
Publication date
Feb 11, 2010
Schering Corporation
Xiongwei Shi
C07 - ORGANIC CHEMISTRY