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Wyatt Paul
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Cambridgeshire, GB
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Patents Grants
last 30 patents
Information
Patent Grant
N-myristoyl transferase inhibitors
Patent number
9,828,346
Issue date
Nov 28, 2017
University of Dundee
Stephen Brand
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazole derivatives as protein kinase modulators
Patent number
9,283,226
Issue date
Mar 15, 2016
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
N-myristoyl transferase inhibitors
Patent number
9,156,811
Issue date
Oct 13, 2015
Univeristy of Dundee
Stephen Brand
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
9,051,278
Issue date
Jun 9, 2015
Astex Therapeutics, Ltd.
Valerio Berdini
C04 - CEMENTS CONCRETE ARTIFICIAL STONE CERAMICS REFRACTORIES
Information
Patent Grant
Ortho-condensed pyridine and pyrimidine derivatives (e.g., purines)...
Patent number
9,006,430
Issue date
Apr 14, 2015
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Ortho-condensed pyridine and pyrimidine derivatives (e.g., purines)...
Patent number
8,809,336
Issue date
Aug 19, 2014
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazole compounds that modulate the activity of CDK, GSK and auror...
Patent number
8,778,936
Issue date
Jul 15, 2014
Astex Therapeutics Limited
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
8,779,147
Issue date
Jul 15, 2014
Astex Therapeutics, Ltd.
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazole derivatives as protein kinase modulators
Patent number
8,691,806
Issue date
Apr 8, 2014
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Ortho-condensed pyridine and pyrimidine derivatives (e.g., purines)...
Patent number
8,546,407
Issue date
Oct 1, 2013
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted diketopiperazines as oxytocin antagonists
Patent number
8,541,579
Issue date
Sep 24, 2013
Glaxo Group Limited
Alan David Borthwick
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Combinations of pyrazole kinase inhibitors
Patent number
8,404,718
Issue date
Mar 26, 2013
Astex Therapeutics Limited
Jayne Elizabeth Curry
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted diketopiperazines as oxytocin antagonists
Patent number
8,367,673
Issue date
Feb 5, 2013
Glaxo Group Limited
Alan David Borthwick
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
4-(2,6-dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid piperid...
Patent number
8,293,767
Issue date
Oct 23, 2012
Astex Therapeutics Limited
Paul Graham Wyatt
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazole derivatives as protein kinase modulators
Patent number
8,247,576
Issue date
Aug 21, 2012
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazole compounds that modulate the activity of CDK, GSK and auror...
Patent number
8,110,573
Issue date
Feb 7, 2012
Astex Therapeutics Limited
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
8,080,666
Issue date
Dec 20, 2011
Astex Therapeutics, Ltd.
Valerio Berdini
C04 - CEMENTS CONCRETE ARTIFICIAL STONE CERAMICS REFRACTORIES
Information
Patent Grant
4-(2,6-dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid piperid...
Patent number
8,013,163
Issue date
Sep 6, 2011
Astex Therapeutics Limited
Paul Graham Wyatt
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzimidazole derivatives and their use as protein kinase inhibitors
Patent number
7,977,477
Issue date
Jul 12, 2011
Astex Therapeutics, Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
7,825,140
Issue date
Nov 2, 2010
Astex Therapeutics, Ltd.
Valerio Berdini
C04 - CEMENTS CONCRETE ARTIFICIAL STONE CERAMICS REFRACTORIES
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
7,745,638
Issue date
Jun 29, 2010
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted diketopiperazines as oxytocin antagonists
Patent number
7,514,437
Issue date
Apr 7, 2009
SmithKline Beecham Corp.
Alan David Borthwick
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
3,4-disubstituted 1H-pyrazole compounds and their use as cyclin dep...
Patent number
7,385,059
Issue date
Jun 10, 2008
Astex Therapeutics Limited
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Use of DNA sequences for male sterility in transgenic plants
Patent number
7,345,222
Issue date
Mar 18, 2008
Gene Shears. Pty. Limited
Roderick John Scott
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Grant
Synthesis and screening of ligands using X-ray crystallography
Patent number
7,149,280
Issue date
Dec 12, 2006
Astex Therapeutics Limited
Harren Jhoti
G01 - MEASURING TESTING
Information
Patent Grant
Inducible promoters
Patent number
6,841,720
Issue date
Jan 11, 2005
Biogemma UK LTD
John Draper
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Grant
Protein complementation in transgenic plants
Patent number
6,791,011
Issue date
Sep 14, 2004
Gene Shears Pty. Limited
Wyatt Paul
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Grant
Method for the production of modified plants
Patent number
6,291,741
Issue date
Sep 18, 2001
Gene Shears Pty. Limited
Wyatt Paul
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Grant
Callase-related DNAs and their use in artificial male sterility
Patent number
5,955,653
Issue date
Sep 21, 1999
Biogemma UK Limited
Roderick John Scott
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Grant
Tapetum-specific promoters from Brassicaceae spp
Patent number
5,723,754
Issue date
Mar 3, 1998
Roderick John Scott
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
PYRAZOLE DERIVATIVES AS PROTEIN KINASE MODULATORS
Publication number
20160250187
Publication date
Sep 1, 2016
Astex Therapeutics Ltd.
Valerio BERDINI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
N-MYRISTOYL TRANSFERASE INHIBITORS
Publication number
20160060224
Publication date
Mar 3, 2016
UNIVERSITY OF DUNDEE
Stephen Brand
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SPERM FUNCTION/ACTIVITY
Publication number
20150231149
Publication date
Aug 20, 2015
UNIVERSITY OF DUNDEE
Christopher Barratt
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3,4-DISUBSTITUTED 1H-PYRAZOLE COMPOUNDS AND THEIR USE AS CYCLIN DEP...
Publication number
20140371213
Publication date
Dec 18, 2014
ASTEX THERAPEUTICS, LTD.
Valerio BERDINI
C04 - CEMENTS CONCRETE ARTIFICIAL STONE CERAMICS REFRACTORIES
Information
Patent Application
ORTHO-CONDENSED PYRIDINE AND PYRIMIDINE DERIVATIVES (E.G., PURINES)...
Publication number
20140303177
Publication date
Oct 9, 2014
ASTEX THERAPEUTICS LIMITED
Valerio BERDINI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLE DERIVATIVES AS PROTEIN KINASE MODULATORS
Publication number
20140271662
Publication date
Sep 18, 2014
Astex Therapeutics Ltd.
Valerio BERDINI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Ortho-Condensed Pyridine and Pyrimidine Derivatives (e.g., Purines)...
Publication number
20140107137
Publication date
Apr 17, 2014
Valerio BERDINI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS
Publication number
20140010892
Publication date
Jan 9, 2014
ASTEX THERAPEUTICS LIMITED
Valerio BERDINI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED DIKETOPIPERAZINES AS OXYTOCIN ANTAGONISTS
Publication number
20130131338
Publication date
May 23, 2013
Glaxo Group Limited
Alan David Borthwick
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLE DERIVATIVES AS PROTEIN KINASE MODULATORS
Publication number
20130005702
Publication date
Jan 3, 2013
ASTEX THERAPEUTICS LIMITED
Valerio BERDINI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3,4-DISUBSTITUTED 1H-PYRAZOLE COMPOUNDS AND THEIR USE AS CYCLIN DEP...
Publication number
20120213791
Publication date
Aug 23, 2012
ASTEX THERAPEUTICS, LTD.
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLE COMPOUNDS THAT MODULATE THE ACTIVITY OF CDK, GSK AND AUROR...
Publication number
20120190673
Publication date
Jul 26, 2012
ASTEX THERAPEUTICS LIMITED
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Application
N-Myristoyl Transferase Inhibitors
Publication number
20110312921
Publication date
Dec 22, 2011
Stephen Brand
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
4-(2,6-DICHLORO-BENZOYLAMINO)-1H-PYRAZOLE-3-CARBOXYLIC ACID PIPERID...
Publication number
20110274616
Publication date
Nov 10, 2011
ASTEX THERAPEUTICS LIMITED
Paul Graham Wyatt
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS PROTEIN KINASE INHIBITORS
Publication number
20110224203
Publication date
Sep 15, 2011
ASTEX THERAPEUTICS LIMITED
Valerio BERDINI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLE DERIVATIVES AS PROTEIN KINASE MODULATORS
Publication number
20110144080
Publication date
Jun 16, 2011
ASTEX THERAPEUTICS LIMITED
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3,4-DISUBSTITUTED 1H-PYRAZOLE COMPOUNDS AND THEIR USE AS CYCLIN DEP...
Publication number
20110003799
Publication date
Jan 6, 2011
ASTEX THERAPEUTICS, LTD.
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Combinations of Pyrazole Kinase Inhibitors
Publication number
20110002879
Publication date
Jan 6, 2011
ASTEX THERAPEUTICS LIMITED
Jayne Elizabeth CURRY
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLE DERIVATIVES AS THAT MODULATE THE ACTIVITY OF CDK, GSK AND...
Publication number
20100160324
Publication date
Jun 24, 2010
ASTEX THERAPEUTICS LIMITED
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Application
4-(2, 6-Dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid (1-met...
Publication number
20090318500
Publication date
Dec 24, 2009
ASTEX THERAPEUTICS LIMITED
Gary Trewartha
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Ortho-Condensed Pyridine and Pyrimidine Derivatives (e.g., Purines)...
Publication number
20090247538
Publication date
Oct 1, 2009
ASTEX THERAPEUTICS LIMITED
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Substituted Diketopiperazines As Oxytocin Antagonists
Publication number
20090186867
Publication date
Jul 23, 2009
Glaxo Group Limited
Alan David Borthwick
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Ortho-Condensed Pyridine and Pyrimidine Derivatives (e.g., Purines)...
Publication number
20090099213
Publication date
Apr 16, 2009
ASTEX THERAPEUTICS LIMITED
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pharmaceutical Compounds
Publication number
20090036435
Publication date
Feb 5, 2009
ASTEX THERAPEUTICS LIMITED
Jayne Elizabeth Curry
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
4-(2,6-dichloro-benzoylamino)-1H-pyrazole-3-carboxylic acid piperid...
Publication number
20090012124
Publication date
Jan 8, 2009
ASTEX THERAPEUTICS LIMITED
Paul Graham Wyatt
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Thiazole And Isothiazole Derivatives That Modulate The Activity Of...
Publication number
20080312223
Publication date
Dec 18, 2008
ASTEX THERAPEUTICS LIMITED
Valerio Berdini
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrazole Derivatives for the Inhibition of CDK'S and GSK'S
Publication number
20080306069
Publication date
Dec 11, 2008
ASTEX THERAPEUTICS LIMITED
Paul Graham Wyatt
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Compounds for Treating Protein-Kinase Mediated Disorders
Publication number
20080275029
Publication date
Nov 6, 2008
ASTEX THERAPEUTICS LIMITED
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3,4-DISUBSTITUTED 1H-PYRAZOLE COMPOUNDS AND THEIR USE AS CYCLIN DEP...
Publication number
20080269207
Publication date
Oct 30, 2008
ASTEX THERAPEUTICS, LTD.
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3,4-DISUBSTITUTED 1H-PYRAZOLE COMPOUNDS AND THEIR USE AS CYCLIN DEP...
Publication number
20080200509
Publication date
Aug 21, 2008
ASTEX THERAPEUTICS, LTD.
Valerio Berdini
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE