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Yan Lou
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Pleasanton, CA, US
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Patents Grants
last 30 patents
Information
Patent Grant
Sulfonamido derivatives as cyclin-dependent kinase 2 inhibitors
Patent number
12,331,026
Issue date
Jun 17, 2025
Nikang Therapeutics, Inc.
Yan Lou
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Immunoproteasome inhibitors
Patent number
12,312,370
Issue date
May 27, 2025
Principia Biopharma Inc.
Yan Lou
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Fused tricyclic ring derivatives as SRC homology-2 phosphate inhibi...
Patent number
12,264,167
Issue date
Apr 1, 2025
Nikang Therapeutics, Inc.
Jiping Fu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
2,3-dihydrobenzo[b]thiophene derivatives as hypoxia inducible facto...
Patent number
12,171,741
Issue date
Dec 24, 2024
Nikang Therapeutics, Inc.
Jiping Fu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Indane derivatives as hypoxia inducible factor-2(α) inhibitors
Patent number
12,077,506
Issue date
Sep 3, 2024
Nikang Therapeutics, Inc.
Jiping Fu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Immunoproteasome inhibitors
Patent number
12,024,531
Issue date
Jul 2, 2024
Principia Biopharma Inc.
Yan Lou
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
BCL-2 inhibitors
Patent number
11,993,610
Issue date
May 28, 2024
Newave Pharmaceutical Inc.
Yi Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Immunoproteasome inhibitors
Patent number
11,827,656
Issue date
Nov 28, 2023
Principia Biopharma Inc.
Yan Lou
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tetrahydro-1H-cyclopenta[cd]indene derivatives as hypoxia inducible...
Patent number
11,753,366
Issue date
Sep 12, 2023
Nikang Therapeutics, Inc.
Jiping Fu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Condensed heterocyclic derivates as BCL-2 inhibitors for the treatm...
Patent number
11,680,072
Issue date
Jun 20, 2023
Newave Pharmaceutical Inc.
Yi Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Process of preparing 3-fluoro-5(((1R,2aR)-3,3,4,4-tetrafluoro-1,2a-...
Patent number
11,634,382
Issue date
Apr 25, 2023
Nikang Therapeutics, Inc.
Jiping Fu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Fused tricyclic ring derivatives as Src homology-2 phosphate inhibi...
Patent number
11,518,772
Issue date
Dec 6, 2022
Nikang Therapeutics, Inc.
Jiping Fu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tri-substituted heteroaryl derivatives as Src homology-2 phosphatas...
Patent number
11,459,340
Issue date
Oct 4, 2022
Nikang Therapeutics, Inc.
Jiping Fu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Hypoxia inducible factor-2(alpha) inhibitors and their use in the t...
Patent number
11,420,936
Issue date
Aug 23, 2022
Nikang Therapeutics, Inc.
Jiping Fu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
BCL-2 inhibitors
Patent number
11,365,206
Issue date
Jun 21, 2022
Newave Pharmaceutical Inc.
Yi Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Condensed heterocyclic derivates as BCL-2 inhibitors for the treatm...
Patent number
11,279,711
Issue date
Mar 22, 2022
Newave Pharmaceutical Inc.
Yi Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tetrahydro-1H-cyclopenta[cd]indene derivatives as hypoxia inducible...
Patent number
11,267,782
Issue date
Mar 8, 2022
Nikang Therapeutics, Inc.
Jiping Fu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Immunoproteasome inhibitors
Patent number
11,225,493
Issue date
Jan 18, 2022
Principia Biopharma Inc.
Yan Lou
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Immunoproteasome inhibitors
Patent number
11,154,563
Issue date
Oct 26, 2021
Principia Biopharma Inc.
Yan Lou
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Fused tricyclic ring derivatives as Src homology-2 phosphate inhibi...
Patent number
11,034,705
Issue date
Jun 15, 2021
Nikang Therapeutics, Inc.
Jiping Fu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Fused tricyclic ring derivatives as SRC homology-2 phosphatase inhi...
Patent number
10,894,797
Issue date
Jan 19, 2021
Nikang Therapeutics, Inc.
Jiping Fu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Biaryl amide compounds as kinase inhibitors
Patent number
10,709,712
Issue date
Jul 14, 2020
Novartis AG
Robert John Aversa
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Therapeutic agents for the treatment of HBV infection
Patent number
10,501,456
Issue date
Dec 10, 2019
Newave Pharmaceutical Inc.
Yi Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Covalent inhibitors of CDK-7
Patent number
10,456,397
Issue date
Oct 29, 2019
Newave Pharmaceutical Inc.
Yi Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds and compositions as kinase inhibitors
Patent number
10,392,404
Issue date
Aug 27, 2019
Novartis AG
Paul Andrew Barsanti
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
BCL-2 inhibitors
Patent number
10,377,755
Issue date
Aug 13, 2019
Newave Pharmaceutical Inc.
Yi Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Dual-warhead covalent inhibitors of FGFR-4
Patent number
10,253,029
Issue date
Apr 9, 2019
Newave Pharmaceutical Inc.
Yi Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Biaryl amide compounds as kinase inhibitors
Patent number
10,245,267
Issue date
Apr 2, 2019
Novartis AG
Robert John Aversa
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Therapeutic agents for the treatment of HBV infection
Patent number
10,239,872
Issue date
Mar 26, 2019
Newave Pharmaceutical Inc.
Yi Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Covalent inhibitors of CDK-7
Patent number
10,195,200
Issue date
Feb 5, 2019
Newave Pharmaceutical Inc.
Yi Chen
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
CONDENSED HETEROCYCLIC DERIVATIVES AS BCL-2 INHIBITORS FOR THE TREA...
Publication number
20250179090
Publication date
Jun 5, 2025
Newave Pharmaceutical Inc.
Yi Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BCL-2 INHIBITORS
Publication number
20250051329
Publication date
Feb 13, 2025
Newave Pharmaceutical Inc.
Yi Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS FOR DEGRADING CYCLIN-DEPENDENT KINASE 2 VIA UBIQUITIN PRO...
Publication number
20250018049
Publication date
Jan 16, 2025
NiKang Therapeutics, Inc.
Jiping FU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BCL-2 INHIBITORS
Publication number
20240425520
Publication date
Dec 26, 2024
Newave Pharmaceutical Inc.
Yi Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ALKYLIDENE DERIVATIVES AS KRAS INHIBITORS
Publication number
20240287100
Publication date
Aug 29, 2024
NiKang Therapeutics, Inc.
Jiping FU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Immunoproteasome Inhibitors
Publication number
20240199655
Publication date
Jun 20, 2024
Principia Biopharma Inc.
Yan Lou
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINAZOLINE AMINE DERIVATIVES AS KRAS INHIBITORS
Publication number
20240166669
Publication date
May 23, 2024
NiKang Therapeutics, Inc.
Jiping Fu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TETRAHYDRO-1H-CYCLOPENTA[CD]INDENE DERIVATIVES AS HYPOXIA INDUCIBLE...
Publication number
20230373909
Publication date
Nov 23, 2023
NiKang Therapeutics, Inc.
Jiping FU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SULFONAMIDO DERIVATIVES AS CYCLIN-DEPENDENT KINASE 2 INHIBITORS
Publication number
20230303509
Publication date
Sep 28, 2023
NiKang Therapeutics, Inc.
Yan LOU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CONDENSED HETEROCYCLIC DERIVATES AS BCL-2 INHIBITORS FOR THE TREATM...
Publication number
20230271979
Publication date
Aug 31, 2023
Newave Pharmaceutical Inc.
Yi Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PROCESS OF PREPARING 3-FLUORO-5(((1R,2AR)-3,3,4,4-TETRAFLUORO-1,2A-...
Publication number
20230202970
Publication date
Jun 29, 2023
NiKang Therapeutic, Inc.
Jiping FU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FUSED TRICYCLIC RING DERIVATIVES AS SRC HOMOLOGY-2 PHOSPHATE INHIBI...
Publication number
20230167134
Publication date
Jun 1, 2023
NiKang Therapeutics, Inc.
Jiping FU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
IMMUNOPROTEASOME INHIBITORS
Publication number
20230133165
Publication date
May 4, 2023
Principia Biopharma Inc.
Yan Lou
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESSES OF MAKING 3-FLUORO-5-(((1S,2aR)-1,3,3,4,4-PENTAFLUORO-2a-...
Publication number
20230115881
Publication date
Apr 13, 2023
NiKang Therapeutics, Inc.
Charles M. COOK
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BCL-2 INHIBITORS
Publication number
20220402941
Publication date
Dec 22, 2022
Newave Pharmaceutical Inc.
Yi Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HYPOXIA INDUCIBLE FACTOR-2(ALPHA) INHIBITORS AND THEIR USE IN THE T...
Publication number
20220380302
Publication date
Dec 1, 2022
NiKang Therapeutics, Inc.
Jiping FU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TRICYCLIC DERIVATIVES AS HYPOXIA INDUCIBLE FACTOR-2(ALPHA) INHIBITORS
Publication number
20220274914
Publication date
Sep 1, 2022
NiKang Therapeutics, Inc.
Jiping Fu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CONDENSED HETEROCYCLIC DERIVATES AS BCL-2 INHIBITORS FOR THE TREATM...
Publication number
20220220126
Publication date
Jul 14, 2022
Newave Pharmaceutical Inc.
Yi Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HYPOXIA INDUCIBLE FACTOR-2(ALPHA) INHIBITORS AND THEIR USE IN THE T...
Publication number
20220185771
Publication date
Jun 16, 2022
NiKang Therapeutics, Inc.
Jiping FU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
FUSED POLYCYCLIC PYRIDONE COMPOUNDS AS INFLUENZA VIRUS REPLICATION...
Publication number
20220177487
Publication date
Jun 9, 2022
NiKang Therapeutics, Inc.
Jiping FU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TETRAHYDRO-1H-CYCLOPENTA[CD]INDENE DERIVATIVES AS HYPOXIA INDUCIBLE...
Publication number
20220162158
Publication date
May 26, 2022
NiKang Therapeutics, Inc.
Jiping FU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PROCESS OF PREPARING 3-FLUORO-5(((1R,2AR)-3,3,4,4-TETRAFLUORO-1,2A-...
Publication number
20220119345
Publication date
Apr 21, 2022
NiKang Therapeutics, Inc.
Jiping FU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Immunoproteasome Inhibitors
Publication number
20220073538
Publication date
Mar 10, 2022
Principia Biopharma Inc.
Yan Lou
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2,3-DIHYDROBENZO[b]THIOPHENE DERIVATIVES AS HYPOXIA INDUCIBLE FACTO...
Publication number
20220054451
Publication date
Feb 24, 2022
NiKang Therapeutics, Inc.
Jiping FU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TRI-SUBSTITUTED HETEROARYL DERIVATIVES AS SRC HOMOLOGY-2 PHOSPHATE...
Publication number
20210380604
Publication date
Dec 9, 2021
NiKang Therapeutics, Inc.
Jiping FU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INDANE DERIVATIVES AS HYPOXIA INDUCIBLE FACTOR-2(ALPHA) INHIBITORS
Publication number
20210380536
Publication date
Dec 9, 2021
NiKang Therapeutics, Inc.
Jiping FU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ADENOSINE RECEPTOR BINDING COMPOUNDS
Publication number
20210355104
Publication date
Nov 18, 2021
NiKang Therapeutics, Inc.
Yan Lou
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TETRAHYDRO-1H-CYCLOPENTA[CD]INDENE DERIVATIVES AS HYPOXIA INDUCIBLE...
Publication number
20210347729
Publication date
Nov 11, 2021
NiKang Therapeutics, Inc.
Jiping FU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TETRAHYDRO-1H-CYCLOPENTA[CD]INDENE DERIVATIVES AS HYPOXIA INDUCIBLE...
Publication number
20210246102
Publication date
Aug 12, 2021
NiKang Therapeutics, Inc.
Jiping FU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FUSED TRICYCLIC RING DERIVATIVES AS SRC HOMOLOGY-2 PHOSPHATE INHIBI...
Publication number
20210188876
Publication date
Jun 24, 2021
Nikang Therapuetics, Inc.
Jiping FU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE