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last 30 patents
Information
Patent Grant
Pyrrolo[2,1-f][1,2,4]triazine derivatives serving as selective HER2...
Patent number
12,030,897
Issue date
Jul 9, 2024
Medshine Discovery Inc.
Kevin X Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Crystal form a of (5-amino-8-(2-methyl-6-(trifluoromethyl)pyridin-4...
Patent number
11,649,239
Issue date
May 16, 2023
Medshine Discovery Inc.
Kevin X. Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
LSD1 inhibitor and preparation method and application thereof
Patent number
11,433,053
Issue date
Sep 6, 2022
Medshine Discovery Inc.
Lingyun Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyridopyrimidine compounds acting as mTORC 1/2 dual inhibitors
Patent number
11,377,444
Issue date
Jul 5, 2022
Medshine Discovery Inc.
Kevin X Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Sulfonyl-substituted isoquinolines as inhibitors of RHO kinase and...
Patent number
11,155,559
Issue date
Oct 26, 2021
CHINA RESOURCES PHARMACEUTICAL HOLDINGS COMPANY LIMITED
Yuanshan Yao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
[1,2,4]triazolo[1,5-c]pyrimidine derivative as A2A receptor inhibitor
Patent number
11,117,899
Issue date
Sep 14, 2021
Medshine Discovery Inc.
Kevin X Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
[1,2,4]triazolo[1,5-c]pyrimidine derivative as A2A receptor inhibitor
Patent number
11,066,411
Issue date
Jul 20, 2021
Medshine Discovery Inc.
Kevin X Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dimethylphosphine oxide compound
Patent number
11,046,720
Issue date
Jun 29, 2021
GUIZHOU INOCHINI TECHNOLOGY CO., LTD
Lingyun Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Isoquinolinesulfonyl derivative as RHO kinase inhibitor
Patent number
9,856,264
Issue date
Jan 2, 2018
Medshine Discovery Inc.
Lingyun Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
SALT FORM AND CRYSTAL FORM OF HETEROCYCLIC SUBSTITUTED PURINONE DER...
Publication number
20240254145
Publication date
Aug 1, 2024
ZAI LAB (SHANGHAI) CO., LTD.
Kevin X. Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FUSED POLYCYCLIC SUBSTITUTED 5-CARBOXYLIC ACID THIENOPYRIMIDINE DIO...
Publication number
20240158413
Publication date
May 16, 2024
SOTER BIOPHARMA PTE. LTD.
Kevin X. Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
TETRAHYDROISOQUINOLINE DERIVATIVE AND USE THEREOF
Publication number
20230365558
Publication date
Nov 16, 2023
MEDSHINE DISCOVERY INC.
Kevin X CHEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRIMIDOPYRROLE SPIRO COMPOUNDS AND DERIVATIVES THEREOF AS DNA-PK I...
Publication number
20230055321
Publication date
Feb 23, 2023
Kevin X CHEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRIMIDOIMIDAZOLE COMPOUNDS USED AS DNA-PK INHIBITORS
Publication number
20230026616
Publication date
Jan 26, 2023
MEDSHINE DISCOVERY INC.
Kevin X CHEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SALT AND CRYSTAL FORM OF MTORC1/2 DUAL KINASE ACTIVITY INHIBITOR AN...
Publication number
20220306622
Publication date
Sep 29, 2022
MEDSHINE DISCOVERY INC.
Kevin X CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINAZOLINE AND CINNOLINE DERIVATIVES AS DNA-PK INHIBITOR
Publication number
20220267310
Publication date
Aug 25, 2022
MEDSHINE DISCOVERY INC.
Kevin X Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SALT FORM AND CRYSTAL FORM OF A2A RECEPTOR ANTAGONIST AND PREPARATI...
Publication number
20220185825
Publication date
Jun 16, 2022
CSTONE PHARMACEUTICAL (SUZHOU) CO., LTD.
Kevin X CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLO[2,1-F][1,2,4]TRIAZINE DERIVATIVES SERVING AS SELECTIVE HER2...
Publication number
20210323979
Publication date
Oct 21, 2021
MEDSHINE DISCOVERY INC.
Kevin X CHEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
DIMETHYLPHOSPHINE OXIDE COMPOUND
Publication number
20210147453
Publication date
May 20, 2021
GUIZHOU INOCHINI TECHNOLOGY CO., LTD
Lingyun WU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CRYSTAL FORM AND SALT TYPE OF TRIAZOLOPYRIMIDINE COMPOUND AND PREPA...
Publication number
20210094957
Publication date
Apr 1, 2021
MEDSHINE DISCOVERY INC.
Kevin X. Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINAZOLINE DERIVATIVE AND USE THEREOF
Publication number
20210078958
Publication date
Mar 18, 2021
MEDSHINE DISCOVERY INC.
Kevin X. CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
LSD1 INHIBITOR AND PREPARATION METHOD AND APPLICATION THEREOF
Publication number
20200345700
Publication date
Nov 5, 2020
MEDSHINE DISCOVERY INC.
Lingyun WU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRIDOPYRIMIDINE COMPOUNDS ACTING AS MTORC 1/2 DOUBLE-KINASE INHIBI...
Publication number
20200339568
Publication date
Oct 29, 2020
MEDSHINE DISCOVERY INC.
Kevin X CHEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ISOQUINOLINYLSULFONYL DERIVATIVE AND USE THEREOF
Publication number
20200207772
Publication date
Jul 2, 2020
CHINA RESOURCES PHARMACEUTICAL HOLDINGS COMPANY LIMITED
Yuanshan YAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
[1,2,4]TRIAZOLO[1,5-C]PYRIMIDINE DERIVATIVE AS A2A RECEPTOR INHIBITOR
Publication number
20200131184
Publication date
Apr 30, 2020
MEDSHINE DISCOVERY INC.
KEVIN X CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ISOQUINOLINESULFONYL DERIVATIVE AS RHO KINASE INHIBITOR
Publication number
20170037050
Publication date
Feb 9, 2017
MEDSHINE DISCOVERY INC.
Lingyun WU
C07 - ORGANIC CHEMISTRY