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Patents Grants
last 30 patents
Information
Patent Grant
6-fused heteroaryldihydropyrimidines for the treatment and prophyla...
Patent number
12,351,575
Issue date
Jul 8, 2025
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Heteroaryl heterocyclyl compounds for the treatment of autoimmune d...
Patent number
11,713,327
Issue date
Aug 1, 2023
HOFFMANN-LA ROCHE INC.
Fabian Dey
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of synthesizing pyrazine compounds
Patent number
11,168,086
Issue date
Nov 9, 2021
HOFFMANN-LA ROCHE INC.
Taishan Hu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolopyrazine and triazolopyrazine compounds for the treatment o...
Patent number
10,683,299
Issue date
Jun 16, 2020
HOFFMANN-LA ROCHE INC.
Xingchun Han
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Carboxy tetrahydropyrazolopyrazine compounds for the treatment of i...
Patent number
10,562,905
Issue date
Feb 18, 2020
HOFFMANN-LA ROCHE INC.
Taishan Hu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
6-fused heteroaryldihydropyrimidines for the treatment and prophyla...
Patent number
10,428,069
Issue date
Oct 1, 2019
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
6-fused heteroaryldihydropyrimidines for the treatment and prophyla...
Patent number
10,081,627
Issue date
Sep 25, 2018
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazine compounds for the treatment of infectious diseases
Patent number
9,890,167
Issue date
Feb 13, 2018
HOFFMANN-LA ROCHE INC.
Taishan Hu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-bridged heteroaryldihydropyrimidines for the treatment and prophy...
Patent number
9,758,530
Issue date
Sep 12, 2017
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
6-bridged heteroaryldihydropyrimidines for the treatment and prophy...
Patent number
9,266,904
Issue date
Feb 23, 2016
Hoffmann-La Roche Inc.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
6-fused heteroaryldihydropyrimidines for the treatment and prophyla...
Patent number
9,233,978
Issue date
Jan 12, 2016
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
PYRAZOLO[3,4-B]PYRIDINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE D...
Publication number
20240360126
Publication date
Oct 31, 2024
HOFFMANN-LA ROCHE INC.
Dongdong Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HYDROISOQUINOLINE OR HYDRONAPHTHYRIDINE COMPOUNDS FOR THE TREATMENT...
Publication number
20240317735
Publication date
Sep 26, 2024
Hoffmann-La Roche Inc.
Fabian DEY
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1,8-NAPHTHYRIDIN-2-ONE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DI...
Publication number
20230041743
Publication date
Feb 9, 2023
HOFFMANN-LA ROCHE INC.
Hong SHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HYDROPYRAZINO[1,2-D][1,4]DIAZEPINE COMPOUNDS FOR THE TREATMENT OF A...
Publication number
20230034723
Publication date
Feb 2, 2023
HOFFMANN-LA ROCHE INC.
Hongtao XU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SPIRO(ISOBENZOFURANAZETIDINE) COMPOUNDS FOR THE TREATMENT OF AUTOIM...
Publication number
20230002415
Publication date
Jan 5, 2023
HOFFMANN-LA ROCHE INC.
Jianguo CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HEXAHYDRO-1H-PYRAZINO[1,2-A]PYRAZINE COMPOUNDS FOR THE TREATMENT OF...
Publication number
20220340597
Publication date
Oct 27, 2022
HOFFMANN-LA ROCHE INC.
Wei ZHU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL HETEROARYL HETEROCYCLYL COMPOUNDS FOR THE TREATMENT OF AUTOIM...
Publication number
20210300947
Publication date
Sep 30, 2021
HOFFMANN-LA ROCHE INC.
FABIAN DEY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDINYL HETEROCYCLYL COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DI...
Publication number
20210269451
Publication date
Sep 2, 2021
HOFFMANN-LA ROCHE INC.
HAIXIA LIU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CARBOXY TETRAHYDROPYRAZOLOPYRAZINE COMPOUNDS FOR THE TREATMENT OF I...
Publication number
20200181156
Publication date
Jun 11, 2020
HOFFMANN-LA ROCHE INC.
Taishan Hu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-fused heteroaryldihydropyrimidines for the treatment and prophyla...
Publication number
20200062753
Publication date
Feb 27, 2020
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL CARBOXY TETRAHYDROPYRAZOLOPYRAZINE COMPOUNDS FOR THE TREATMEN...
Publication number
20190322670
Publication date
Oct 24, 2019
HOFFMANN-LA ROCHE INC.
Taishan Hu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL PYRAZOLOPYRAZINE AND TRIAZOLOPYRAZINE COMPOUNDS FOR THE TREAT...
Publication number
20190248792
Publication date
Aug 15, 2019
HOFFMANN-LA ROCHE INC.
Xingchun Han
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Novel 6-fused heteroaryldihydropyrimidines for the treatment and pr...
Publication number
20180370969
Publication date
Dec 27, 2018
HOFFMANN-LA ROCHE INC.
Lei Guo
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL PYRAZINE COMPOUNDS FOR THE TREATMENT OF INFECTIOUS DISEASES
Publication number
20180334461
Publication date
Nov 22, 2018
HOFFMANN-LA ROCHE INC.
Taishan Hu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL 6-BRIDGED HETEROARYLDIHYDROPYRIMIDINES FOR THE TREATMENT AND...
Publication number
20160122363
Publication date
May 5, 2016
HOFFMANN-LA ROCHE INC.
Lei Guo
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel 6-fused heteroaryldihydropyrimidines for the treatment and pr...
Publication number
20160083383
Publication date
Mar 24, 2016
HOFFMANN-LA ROCHE INC.
Lei Guo
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel 6-fused heteroaryldihydropyrimidines for the treatment and pr...
Publication number
20150252057
Publication date
Sep 10, 2015
HOFFMANN-LA ROCHE INC.
Lei Guo
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL 6-BRIDGED HETEROARYLDIHYDROPYRIMIDINES FOR THE TREATMENT AND...
Publication number
20140343032
Publication date
Nov 20, 2014
Hoffmann-La Roche Inc.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE