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Flemington, NJ, US
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Patents Grants
last 30 patents
Information
Patent Grant
Substituted N-heteroaryl spirolactam bipyrrolidines, preparation an...
Patent number
9,533,995
Issue date
Jan 3, 2017
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted phenyl cycloalkyl pyrrolidine (piperidine) spirolactams...
Patent number
9,453,023
Issue date
Sep 27, 2016
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-alkyl and N-acyl tetrahydro-isoquinoline derivatives,...
Patent number
8,871,788
Issue date
Oct 28, 2014
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-heteroaryl bipyrrolidine carboxamides, preparation an...
Patent number
8,859,588
Issue date
Oct 14, 2014
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-cycloamino-3-(pyrid-4-yl)imidazo[1,2-b]pyridazine derivatives, pr...
Patent number
8,846,676
Issue date
Sep 30, 2014
Sanofi
Antonio Almario Garcia
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-heteroaryl spirolactam bipyrrolidines, preparation an...
Patent number
8,796,278
Issue date
Aug 5, 2014
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-heterocycloalkyl bipyrrolidinylphenyl amide derivativ...
Patent number
8,754,095
Issue date
Jun 17, 2014
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted phenyl cycloalkyl pyrrolidine (piperidine) spirolactams...
Patent number
8,735,385
Issue date
May 27, 2014
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-heteroaryl tetrahydro-isoquinoline derivatives, prepa...
Patent number
8,623,877
Issue date
Jan 7, 2014
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-phenyl-bipyrrolidine carboxamides and therapeutic use...
Patent number
8,618,159
Issue date
Dec 31, 2013
Sanofi
Werngard Czechtizky
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted piperidine spiro pyrrolidinone and piperidinone, prepar...
Patent number
8,604,046
Issue date
Dec 10, 2013
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted tetrahydropyran spiro pyrrolidinone and piperidinone, p...
Patent number
8,383,814
Issue date
Feb 26, 2013
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-cycloamino-3-(pyrid-4-yl)imidazo[1,2-b]pyridazine derivatives, pr...
Patent number
8,354,405
Issue date
Jan 15, 2013
Sanofi
Antonio Almario Garcia
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-phenyl-bipyrrolidine carboxamides and therapeutic use...
Patent number
8,252,824
Issue date
Aug 28, 2012
Sanofi
Werngard Czechtizky
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted piperidine spiro pyrrolidinone and piperidinone, prepar...
Patent number
8,227,481
Issue date
Jul 24, 2012
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-phenyl-pyrrolidinylmethylpyrrolidine amides and thera...
Patent number
8,227,504
Issue date
Jul 24, 2012
Sanofi
Werngard Czechtizky
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-phenyl-bipyrrolidine ureas and therapeutic use thereof
Patent number
8,222,290
Issue date
Jul 17, 2012
Sanofi
Werngard Czechtizky
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted tetrahydropyran spiro pyrrolidinone and piperidinone, p...
Patent number
8,217,052
Issue date
Jul 10, 2012
Sanofi
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted N-phenyl-bipyrrolidine carboxamides and therapeutic use...
Patent number
8,088,808
Issue date
Jan 3, 2012
Sanofi
Werngard Czechtizky
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
[4-(5-aminomethyl-2-fluoro-phenyl)-piperidin-1-yl]-(4-bromo-3-methy...
Patent number
7,482,459
Issue date
Jan 27, 2009
Aventis Pharmaceuticals Inc.
Zhongli Gao
Patents Applications
last 30 patents
Information
Patent Application
MACROCYCLIC COMPOUNDS, COMPOSITIONS, AND METHODS OF USING THEREOF
Publication number
20250197420
Publication date
Jun 19, 2025
Sionna Therapeutics Inc.
Junkai Liao
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC COMPOUNDS, COMPOSITIONS, AND METHODS OF USING THEREOF
Publication number
20250197422
Publication date
Jun 19, 2025
Sionna Therapeutics Inc.
Junkai Liao
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INDOLE COMPOUNDS AND METHODS OF USE
Publication number
20240279220
Publication date
Aug 22, 2024
Genzyme Corporation
Junkai Liao
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INDOLE COMPOUNDS AND METHODS OF USE
Publication number
20240239784
Publication date
Jul 18, 2024
Genzyme Corporation
Junkai Liao
C07 - ORGANIC CHEMISTRY
Information
Patent Application
5-MEMBERED HETEROARYLAMINOSULFONAMIDES FOR TREATING CONDITIONS MEDI...
Publication number
20240002374
Publication date
Jan 4, 2024
Genzyme Corporation
Junkai Liao
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ARYLAMIDES AND METHODS OF USE THEREOF
Publication number
20230159439
Publication date
May 25, 2023
Genzyme Corporation
Junkai Liao
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ARYLAMIDES AND METHODS OF USE THEREOF
Publication number
20230159438
Publication date
May 25, 2023
Genzyme Corporation
Junkai Liao
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ARYLAMIDES AND METHODS OF USE THEREOF
Publication number
20230147360
Publication date
May 11, 2023
Genzyme Corporation
Junkai Liao
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
6-MEMBERED HETEROARYLAMINOSULFONAMIDES FOR TREATING DISEASES AND CO...
Publication number
20230137585
Publication date
May 4, 2023
Genzyme Corporation
Zhongli Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-HETEROARYL SPIROLACTAM BIPYRROLIDINES, PREPARATION AN...
Publication number
20140315923
Publication date
Oct 23, 2014
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PHENYL CYCLOALKYL PYRROLIDINE (PIPERIDINE) SPIROLACTAMS...
Publication number
20140275005
Publication date
Sep 18, 2014
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PHENYL CYCLOALKYL PYRROLIDINE (PIPERIDINE) SPIROLACTAMS...
Publication number
20130065877
Publication date
Mar 14, 2013
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-HETEROARYL BIPYRROLIDINE CARBOXAMIDES, PREPARATION AN...
Publication number
20130065923
Publication date
Mar 14, 2013
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-ALKYL AND N-ACYL TETRAHYDRO-ISOQUINOLINE DERIVATIVES,...
Publication number
20130065919
Publication date
Mar 14, 2013
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-HETEROCYCLOALKYL BIPYRROLIDINYLPHENYL AMIDE DERIVATIV...
Publication number
20130059891
Publication date
Mar 7, 2013
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-HETEROARYL SPIROLACTAM BIPYRROLIDINES, PREPARATION AN...
Publication number
20130059863
Publication date
Mar 7, 2013
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-PHENYL SPIROLACTAM BIPYRROLIDINES, PREPARATION AND TH...
Publication number
20130059874
Publication date
Mar 7, 2013
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-HETEROARYL TETRAHYDRO-ISOQUINOLINE DERIVATIVES, PREPA...
Publication number
20130059838
Publication date
Mar 7, 2013
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-CYCLOAMINO-3-(PYRID-4-YL)IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES, PR...
Publication number
20130012516
Publication date
Jan 10, 2013
SANOFI
Antonio ALMARIO GARCIA
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PIPERIDINE SPIRO PYRROLIDINONE AND PIPERIDINONE, PREPAR...
Publication number
20120258979
Publication date
Oct 11, 2012
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED TETRAHYDROPYRAN SPIRO PYRROLIDINONE AND PIPERIDINONE, P...
Publication number
20120238757
Publication date
Sep 20, 2012
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE...
Publication number
20120065234
Publication date
Mar 15, 2012
SANOFI
Werngard CZECHTIZKY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
2-ALKYL-6-CYCLOAMINO-3-(PYRIDIN-4-YL)IMIDAZO[1,2-B]-PYRIDAZINE DERI...
Publication number
20110312934
Publication date
Dec 22, 2011
Sanofi-Aventis
Antonio Almario Garcia
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PIPERIDINE SPIRO PYRROLIDINONE AND PIPERIDINONE, PREPAR...
Publication number
20110257213
Publication date
Oct 20, 2011
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED TETRAHYDROPYRAN SPIRO PYRROLIDINONE AND PIPERIDINONE, P...
Publication number
20110251225
Publication date
Oct 13, 2011
SANOFI
Zhongli GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-CYCLOAMINO-3-(PYRID-4-YL)IMIDAZO[1,2-b]PYRIDAZINE DERIVATIVES, PR...
Publication number
20100179154
Publication date
Jul 15, 2010
Sanofi-Aventis
Antonio ALMARIO GARCIA
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE...
Publication number
20100173949
Publication date
Jul 8, 2010
Sanofi-Aventis
Werngard CZECHTIZKY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-PHENYL-BIPYRROLIDINE UREAS AND THERAPEUTIC USE THEREOF
Publication number
20100173908
Publication date
Jul 8, 2010
Sanofi-Aventis
Werngard CZECHTIZKY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-PHENYL-BIPYRROLIDINE CARBOXAMIDES AND THERAPEUTIC USE...
Publication number
20100173897
Publication date
Jul 8, 2010
Sanofi-Aventis
Werngard CZECHTIZKY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED N-PHENYL-PYRROLIDINYLMETHYLPYRROLIDINE AMIDES AND THERA...
Publication number
20100173898
Publication date
Jul 8, 2010
Sanofi-Aventis
Werngard CZECHTIZKY
C07 - ORGANIC CHEMISTRY