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C07D239/86
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HETEROCYCLIC COMPOUNDS
C07D239/00
Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
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C07D239/86
with hetero atoms directly attached in position 4
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last 30 patents
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Patent Grant
4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for...
Patent number
12,049,461
Issue date
Jul 30, 2024
Gilead Sciences, Inc.
Ling-Jie Gao
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
11,702,424
Issue date
Jul 18, 2023
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Anti-Wolbachia pyrido[2,3-d]pyrimidine compounds
Patent number
11,518,760
Issue date
Dec 6, 2022
Liverpool School of Tropical Medicine
Stephen A. Ward
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Activators of autophagic flux and phospholipase d and clearance of...
Patent number
11,261,199
Issue date
Mar 1, 2022
The Trustees of Columbia University In the City of New York
Kirsten Alison Rinderspacher
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Activators of autophagic flux and phospholipase D and clearance of...
Patent number
11,230,558
Issue date
Jan 25, 2022
The Trustees of Columbia University In the City of New York
Kirsten Alison Rinderspacher
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Activators of autophagic flux and phospholipase D and clearance of...
Patent number
11,008,341
Issue date
May 18, 2021
The Trustees of Columbia University In the City of New York
Kirsten Alison Rinderspacher
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for...
Patent number
10,882,851
Issue date
Jan 5, 2021
Gilead Sciences, Inc.
Ling-Jie Gao
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Activators of autophagic flux and phospholipase D and clearance of...
Patent number
10,865,214
Issue date
Dec 15, 2020
The Trustees of Columbia University in they City of New York
Kirsten Alison Rinderspacher
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
10,793,579
Issue date
Oct 6, 2020
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Activators of autophagic flux and phospholipase D and clearance of...
Patent number
10,626,124
Issue date
Apr 21, 2020
The Trustees of Columbia University In the City of New York
Kirsten Alison Rinderspacher
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Quinazoline derivatives substituted by aniline, preparation method...
Patent number
10,507,209
Issue date
Dec 17, 2019
XUANZHU PHARMA CO, LTD.
Yanyan Dong
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Activators of autophagic flux and phospholipase D and clearance of...
Patent number
10,487,091
Issue date
Nov 26, 2019
The Trustees of Columbia University In the City of New York
Kirsten Alison Rinderspacher
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
10,329,302
Issue date
Jun 25, 2019
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Methods for preparation of quinazoline derivatives
Patent number
9,988,357
Issue date
Jun 5, 2018
Araxes Pharma LLC
Neelakandha S. Mani
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
9,879,022
Issue date
Jan 30, 2018
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Quinazoline derivatives substituted by aniline, preparation method...
Patent number
9,730,934
Issue date
Aug 15, 2017
Xuanzhu Pharma Co., Ltd.
Zhenhua Huang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Method for preparing 1-(4-(4-(3,4-dichloro-2-fluorophenylamino)-7-m...
Patent number
9,518,043
Issue date
Dec 13, 2016
Hanmi Pharm. Co., Ltd.
Keuk Chan Bang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
9,458,168
Issue date
Oct 4, 2016
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds and methods for enzyme-mediated tumor imaging and therapy
Patent number
9,320,815
Issue date
Apr 26, 2016
President and Fellows of Harvard College
Amin I. Kassis
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Fused heterocyclic compound
Patent number
9,260,436
Issue date
Feb 16, 2016
Sumitomo Chemical Company, Limited
Masaki Takahashi
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Morpholinylquinazolines
Patent number
9,126,952
Issue date
Sep 8, 2015
Merck Patent GmbH
Werner Mederski
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...
Patent number
8,648,197
Issue date
Feb 11, 2014
Millennium Pharmaceuticals, Inc.
Kenneth G. Carson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Compounds and methods for enzyme-mediated tumor imaging and therapy
Patent number
8,394,953
Issue date
Mar 12, 2013
President and Fellows of Harvard College
Amin I. Kassis
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...
Patent number
8,168,788
Issue date
May 1, 2012
Millennium Pharmaceuticals, Inc.
Kenneth G. Carson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Combination therapy of her expressing tumors
Patent number
8,163,287
Issue date
Apr 24, 2012
Genentech, Inc.
Mark X. Sliwkowski
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
4-(tetrazol-5-yl)-quinazoline derivatives as anti-cancer agent
Patent number
8,080,558
Issue date
Dec 20, 2011
Natco Pharma Limited
Durga Prasad Konakanchi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Sulphoximine-substituted quinoline and quinazoline derivatives as k...
Patent number
8,003,787
Issue date
Aug 23, 2011
Bayer Schering Pharma AG
Knut Eis
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...
Patent number
7,880,002
Issue date
Feb 1, 2011
Millennium Pharmaceuticals, Inc.
Kenneth G. Carson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Process for preparing quinazoline Rho-kinase inhibitors and interme...
Patent number
7,645,878
Issue date
Jan 12, 2010
Bayer HealthCare LLC
Donald Bankston
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dipeptidyl peptidase inhibitors for the treatment of diabetes
Patent number
7,253,172
Issue date
Aug 7, 2007
Merck & Co., Inc.
Linda Brockunier
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
ANTI-WOLBACHIA PYRIDO[2,3-d]PYRIMIDINECOMPOUNDS
Publication number
20230348460
Publication date
Nov 2, 2023
LIVERPOOL SCHOOL OF TROPICAL MEDICINE
Stephen A. Ward
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
Publication number
20230339960
Publication date
Oct 26, 2023
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TYROSINE KINASE INHIBITORS AND PHARMACEUTICAL APPLICATION THEREOF
Publication number
20230043449
Publication date
Feb 9, 2023
JIANGSU CONCORD BIOTECHNOLOGY CO., LTD
Huabiao CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR...
Publication number
20210276988
Publication date
Sep 9, 2021
GILEAD SCIENCES, INC.
Ling-Jie GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
Publication number
20200377511
Publication date
Dec 3, 2020
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...
Publication number
20200216469
Publication date
Jul 9, 2020
THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
Kirsten Alison Rinderspacher
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS
Publication number
20190345157
Publication date
Nov 14, 2019
LIVERPOOL SCHOOL OF TROPICAL MEDICINE
Stephen A. Ward
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
Publication number
20190270751
Publication date
Sep 5, 2019
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...
Publication number
20180319818
Publication date
Nov 8, 2018
NY STATE PSYCHIATRIC INSTITUTE
Kirsten Alison Rinderspacher
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...
Publication number
20180312526
Publication date
Nov 1, 2018
THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
Kirsten Alison Rinderspacher
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...
Publication number
20180312527
Publication date
Nov 1, 2018
THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
Kirsten Alison Rinderspacher
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
Publication number
20180127432
Publication date
May 10, 2018
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
QUINAZOLINE DERIVATIVES SUBSTITUTED BY ANILINE, PREPARATION METHOD...
Publication number
20170304305
Publication date
Oct 26, 2017
XUANZHU PHARMA CO., LTD.
Yanyan DONG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...
Publication number
20170210759
Publication date
Jul 27, 2017
THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
Kirsten Alison Rinderspacher
C07 - ORGANIC CHEMISTRY
Information
Patent Application
METHODS FOR PREPARATION OF QUINAZOLINE DERIVATIVES
Publication number
20170190672
Publication date
Jul 6, 2017
Araxes Pharma LLC
Neelakandha S. Mani
C07 - ORGANIC CHEMISTRY
Information
Patent Application
4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR...
Publication number
20160257673
Publication date
Sep 8, 2016
GILEAD SCIENCES, INC.
Ling-Jie GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Method For Preparing 1-(4-(4-(3,4-Dichloro-2-Fluorophenylamino)-7-M...
Publication number
20150344458
Publication date
Dec 3, 2015
HANMI PHARM CO., LTD.
Keuk Chan BANG
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMBINATION THERAPY OF HER EXPRESSING TUMORS
Publication number
20150086545
Publication date
Mar 26, 2015
Genentech, Inc.
Mark X. Sliwkowski
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PIPERAZINYL-PYRROLIDINE COMPOUNDS USEFUL AS CHEMOKINE R...
Publication number
20140364420
Publication date
Dec 11, 2014
Millennium Pharmaceuticals, Inc.
Kenneth G. Carson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS AND METHODS FOR ENZYME-MEDIATED TUMOR IMAGING AND THERAPY
Publication number
20130336887
Publication date
Dec 19, 2013
President and Fellows of Harvard College
Amin I. Kassis
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
QUINAZOLINE DERIVATIVES SUBSTITUTED BY ANILINE, PREPARATION METHOD...
Publication number
20130184297
Publication date
Jul 18, 2013
XUANZHU PHARMA CO., LTD
Zhenhua Huang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PIPERAZINYL-PYRROLIDINE COMPOUNDS USEFUL AS CHEMOKINE R...
Publication number
20130123270
Publication date
May 16, 2013
Millennium Pharmaceuticals, Inc.
Kenneth G. Carson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Morpholinylquinazolines
Publication number
20130012489
Publication date
Jan 10, 2013
Merck Patent GmbH
Werner Mederski
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMBINATION THERAPY OF HER EXPRESSING TUMORS
Publication number
20120251530
Publication date
Oct 4, 2012
Mark X Sliwkowski
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...
Publication number
20110237601
Publication date
Sep 29, 2011
Millennium Pharmaceuticals, Inc.
Kenneth G. Carson
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
COMPOUNDS AS THE ESTROGEN RELATED RECEPTORS MODULATORS AND THE USES...
Publication number
20110071148
Publication date
Mar 24, 2011
Guangzhou Institute of Biomedicine and Health, Chinese Academy of Sciences
Ke Ding
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL 4-(TETRAZOL-5-YL)-QUINAZOLINE DERIVATIVES AS ANTI CANCER AGENT
Publication number
20100261740
Publication date
Oct 14, 2010
Natco Pharma Limited
Durga Prasad Konkanchi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PROCESS FOR PREPARING QUINAZOLINE RHO-KINASE INHIBITORS AND INTERME...
Publication number
20100125139
Publication date
May 20, 2010
Donald Bankston
C07 - ORGANIC CHEMISTRY
Information
Patent Application
COMPOUNDS AND METHODS FOR ENZYME-MEDIATED TUMOR IMAGING AND THERAPY
Publication number
20090324495
Publication date
Dec 31, 2009
President and Fellows of Harvard College
Amin I. Kassis
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Use of Oxindole Derivatives in the Treatment of Dementia Related Di...
Publication number
20090312322
Publication date
Dec 17, 2009
AstraZeneca AB
Stefan Berg
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE