with hetero atoms directly attached in position 4

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CPC
C07D239/86

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CCHEMISTRY METALLURGY C07Organic chemistry C07DHETEROCYCLIC COMPOUNDS C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings

Current Industry

C07D239/86with hetero atoms directly attached in position 4

Industries

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Patents Grantslast 30 patents

Information Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
- Patent number 12,202,836
- Issue date Jan 21, 2025
- Pfizer Inc.
- John David Trzupek
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for...
- Patent number 12,049,461
- Issue date Jul 30, 2024
- Gilead Sciences, Inc.
- Ling-Jie Gao
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
- Patent number 11,702,424
- Issue date Jul 18, 2023
- Pfizer Inc.
- John David Trzupek
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Anti-Wolbachia pyrido[2,3-d]pyrimidine compounds
- Patent number 11,518,760
- Issue date Dec 6, 2022
- Liverpool School of Tropical Medicine
- Stephen A. Ward
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Activators of autophagic flux and phospholipase d and clearance of...
- Patent number 11,261,199
- Issue date Mar 1, 2022
- The Trustees of Columbia University In the City of New York
- Kirsten Alison Rinderspacher
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Activators of autophagic flux and phospholipase D and clearance of...
- Patent number 11,230,558
- Issue date Jan 25, 2022
- The Trustees of Columbia University In the City of New York
- Kirsten Alison Rinderspacher
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Activators of autophagic flux and phospholipase D and clearance of...
- Patent number 11,008,341
- Issue date May 18, 2021
- The Trustees of Columbia University In the City of New York
- Kirsten Alison Rinderspacher
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for...
- Patent number 10,882,851
- Issue date Jan 5, 2021
- Gilead Sciences, Inc.
- Ling-Jie Gao
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Activators of autophagic flux and phospholipase D and clearance of...
- Patent number 10,865,214
- Issue date Dec 15, 2020
- The Trustees of Columbia University in they City of New York
- Kirsten Alison Rinderspacher
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
- Patent number 10,793,579
- Issue date Oct 6, 2020
- Pfizer Inc.
- John David Trzupek
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Activators of autophagic flux and phospholipase D and clearance of...
- Patent number 10,626,124
- Issue date Apr 21, 2020
- The Trustees of Columbia University In the City of New York
- Kirsten Alison Rinderspacher
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Quinazoline derivatives substituted by aniline, preparation method...
- Patent number 10,507,209
- Issue date Dec 17, 2019
- XUANZHU PHARMA CO, LTD.
- Yanyan Dong
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Activators of autophagic flux and phospholipase D and clearance of...
- Patent number 10,487,091
- Issue date Nov 26, 2019
- The Trustees of Columbia University In the City of New York
- Kirsten Alison Rinderspacher
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
- Patent number 10,329,302
- Issue date Jun 25, 2019
- Pfizer Inc.
- John David Trzupek
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Methods for preparation of quinazoline derivatives
- Patent number 9,988,357
- Issue date Jun 5, 2018
- Araxes Pharma LLC
- Neelakandha S. Mani
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
- Patent number 9,879,022
- Issue date Jan 30, 2018
- Pfizer Inc.
- John David Trzupek
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Quinazoline derivatives substituted by aniline, preparation method...
- Patent number 9,730,934
- Issue date Aug 15, 2017
- Xuanzhu Pharma Co., Ltd.
- Zhenhua Huang
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Method for preparing 1-(4-(4-(3,4-dichloro-2-fluorophenylamino)-7-m...
- Patent number 9,518,043
- Issue date Dec 13, 2016
- Hanmi Pharm. Co., Ltd.
- Keuk Chan Bang
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
- Patent number 9,458,168
- Issue date Oct 4, 2016
- Pfizer Inc.
- John David Trzupek
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Compounds and methods for enzyme-mediated tumor imaging and therapy
- Patent number 9,320,815
- Issue date Apr 26, 2016
- President and Fellows of Harvard College
- Amin I. Kassis
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Fused heterocyclic compound
- Patent number 9,260,436
- Issue date Feb 16, 2016
- Sumitomo Chemical Company, Limited
- Masaki Takahashi
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Morpholinylquinazolines
- Patent number 9,126,952
- Issue date Sep 8, 2015
- Merck Patent GmbH
- Werner Mederski
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...
- Patent number 8,648,197
- Issue date Feb 11, 2014
- Millennium Pharmaceuticals, Inc.
- Kenneth G. Carson
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Compounds and methods for enzyme-mediated tumor imaging and therapy
- Patent number 8,394,953
- Issue date Mar 12, 2013
- President and Fellows of Harvard College
- Amin I. Kassis
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...
- Patent number 8,168,788
- Issue date May 1, 2012
- Millennium Pharmaceuticals, Inc.
- Kenneth G. Carson
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Combination therapy of her expressing tumors
- Patent number 8,163,287
- Issue date Apr 24, 2012
- Genentech, Inc.
- Mark X. Sliwkowski
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
4-(tetrazol-5-yl)-quinazoline derivatives as anti-cancer agent
- Patent number 8,080,558
- Issue date Dec 20, 2011
- Natco Pharma Limited
- Durga Prasad Konakanchi
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Sulphoximine-substituted quinoline and quinazoline derivatives as k...
- Patent number 8,003,787
- Issue date Aug 23, 2011
- Bayer Schering Pharma AG
- Knut Eis
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...
- Patent number 7,880,002
- Issue date Feb 1, 2011
- Millennium Pharmaceuticals, Inc.
- Kenneth G. Carson
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Process for preparing quinazoline Rho-kinase inhibitors and interme...
- Patent number 7,645,878
- Issue date Jan 12, 2010
- Bayer HealthCare LLC
- Donald Bankston
- C07 - ORGANIC CHEMISTRY

Patents Applicationslast 30 patents

Information Patent Application
ANTI-WOLBACHIA PYRIDO[2,3-d]PYRIMIDINECOMPOUNDS
- Publication number 20230348460
- Publication date Nov 2, 2023
- LIVERPOOL SCHOOL OF TROPICAL MEDICINE
- Stephen A. Ward
- C07 - ORGANIC CHEMISTRY
Information Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
- Publication number 20230339960
- Publication date Oct 26, 2023
- Pfizer Inc.
- John David Trzupek
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
TYROSINE KINASE INHIBITORS AND PHARMACEUTICAL APPLICATION THEREOF
- Publication number 20230043449
- Publication date Feb 9, 2023
- JIANGSU CONCORD BIOTECHNOLOGY CO., LTD
- Huabiao CHEN
- C07 - ORGANIC CHEMISTRY
Information Patent Application
4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR...
- Publication number 20210276988
- Publication date Sep 9, 2021
- GILEAD SCIENCES, INC.
- Ling-Jie GAO
- C07 - ORGANIC CHEMISTRY
Information Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
- Publication number 20200377511
- Publication date Dec 3, 2020
- Pfizer Inc.
- John David Trzupek
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...
- Publication number 20200216469
- Publication date Jul 9, 2020
- THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
- Kirsten Alison Rinderspacher
- C07 - ORGANIC CHEMISTRY
Information Patent Application
COMPOUNDS
- Publication number 20190345157
- Publication date Nov 14, 2019
- LIVERPOOL SCHOOL OF TROPICAL MEDICINE
- Stephen A. Ward
- C07 - ORGANIC CHEMISTRY
Information Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
- Publication number 20190270751
- Publication date Sep 5, 2019
- Pfizer Inc.
- John David Trzupek
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...
- Publication number 20180319818
- Publication date Nov 8, 2018
- NY STATE PSYCHIATRIC INSTITUTE
- Kirsten Alison Rinderspacher
- C07 - ORGANIC CHEMISTRY
Information Patent Application
ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...
- Publication number 20180312526
- Publication date Nov 1, 2018
- THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
- Kirsten Alison Rinderspacher
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...
- Publication number 20180312527
- Publication date Nov 1, 2018
- THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
- Kirsten Alison Rinderspacher
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
- Publication number 20180127432
- Publication date May 10, 2018
- Pfizer Inc.
- John David Trzupek
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
QUINAZOLINE DERIVATIVES SUBSTITUTED BY ANILINE, PREPARATION METHOD...
- Publication number 20170304305
- Publication date Oct 26, 2017
- XUANZHU PHARMA CO., LTD.
- Yanyan DONG
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...
- Publication number 20170210759
- Publication date Jul 27, 2017
- THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK
- Kirsten Alison Rinderspacher
- C07 - ORGANIC CHEMISTRY
Information Patent Application
METHODS FOR PREPARATION OF QUINAZOLINE DERIVATIVES
- Publication number 20170190672
- Publication date Jul 6, 2017
- Araxes Pharma LLC
- Neelakandha S. Mani
- C07 - ORGANIC CHEMISTRY
Information Patent Application
4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR...
- Publication number 20160257673
- Publication date Sep 8, 2016
- GILEAD SCIENCES, INC.
- Ling-Jie GAO
- C07 - ORGANIC CHEMISTRY
Information Patent Application
Method For Preparing 1-(4-(4-(3,4-Dichloro-2-Fluorophenylamino)-7-M...
- Publication number 20150344458
- Publication date Dec 3, 2015
- HANMI PHARM CO., LTD.
- Keuk Chan BANG
- C07 - ORGANIC CHEMISTRY
Information Patent Application
COMBINATION THERAPY OF HER EXPRESSING TUMORS
- Publication number 20150086545
- Publication date Mar 26, 2015
- Genentech, Inc.
- Mark X. Sliwkowski
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
SUBSTITUTED PIPERAZINYL-PYRROLIDINE COMPOUNDS USEFUL AS CHEMOKINE R...
- Publication number 20140364420
- Publication date Dec 11, 2014
- Millennium Pharmaceuticals, Inc.
- Kenneth G. Carson
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
COMPOUNDS AND METHODS FOR ENZYME-MEDIATED TUMOR IMAGING AND THERAPY
- Publication number 20130336887
- Publication date Dec 19, 2013
- President and Fellows of Harvard College
- Amin I. Kassis
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
QUINAZOLINE DERIVATIVES SUBSTITUTED BY ANILINE, PREPARATION METHOD...
- Publication number 20130184297
- Publication date Jul 18, 2013
- XUANZHU PHARMA CO., LTD
- Zhenhua Huang
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
SUBSTITUTED PIPERAZINYL-PYRROLIDINE COMPOUNDS USEFUL AS CHEMOKINE R...
- Publication number 20130123270
- Publication date May 16, 2013
- Millennium Pharmaceuticals, Inc.
- Kenneth G. Carson
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
Morpholinylquinazolines
- Publication number 20130012489
- Publication date Jan 10, 2013
- Merck Patent GmbH
- Werner Mederski
- C07 - ORGANIC CHEMISTRY
Information Patent Application
COMBINATION THERAPY OF HER EXPRESSING TUMORS
- Publication number 20120251530
- Publication date Oct 4, 2012
- Mark X Sliwkowski
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...
- Publication number 20110237601
- Publication date Sep 29, 2011
- Millennium Pharmaceuticals, Inc.
- Kenneth G. Carson
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
COMPOUNDS AS THE ESTROGEN RELATED RECEPTORS MODULATORS AND THE USES...
- Publication number 20110071148
- Publication date Mar 24, 2011
- Guangzhou Institute of Biomedicine and Health, Chinese Academy of Sciences
- Ke Ding
- C07 - ORGANIC CHEMISTRY
Information Patent Application
NOVEL 4-(TETRAZOL-5-YL)-QUINAZOLINE DERIVATIVES AS ANTI CANCER AGENT
- Publication number 20100261740
- Publication date Oct 14, 2010
- Natco Pharma Limited
- Durga Prasad Konkanchi
- C07 - ORGANIC CHEMISTRY
Information Patent Application
PROCESS FOR PREPARING QUINAZOLINE RHO-KINASE INHIBITORS AND INTERME...
- Publication number 20100125139
- Publication date May 20, 2010
- Donald Bankston
- C07 - ORGANIC CHEMISTRY
Information Patent Application
COMPOUNDS AND METHODS FOR ENZYME-MEDIATED TUMOR IMAGING AND THERAPY
- Publication number 20090324495
- Publication date Dec 31, 2009
- President and Fellows of Harvard College
- Amin I. Kassis
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
Use of Oxindole Derivatives in the Treatment of Dementia Related Di...
- Publication number 20090312322
- Publication date Dec 17, 2009
- AstraZeneca AB
- Stefan Berg
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE

with hetero atoms directly attached in position 4

Industry

Parent Industries

Current Industry

Patents Grantslast 30 patents

Bicyclic-fused heteroaryl or aryl compounds

4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for...

Bicyclic-fused heteroaryl or aryl compounds

Anti-Wolbachia pyrido[2,3-d]pyrimidine compounds

Activators of autophagic flux and phospholipase d and clearance of...

Activators of autophagic flux and phospholipase D and clearance of...

Activators of autophagic flux and phospholipase D and clearance of...

4,6-di- and 2,4,6-trisubstituted quinazoline derivatives useful for...

Activators of autophagic flux and phospholipase D and clearance of...

Bicyclic-fused heteroaryl or aryl compounds

Activators of autophagic flux and phospholipase D and clearance of...

Quinazoline derivatives substituted by aniline, preparation method...

Activators of autophagic flux and phospholipase D and clearance of...

Bicyclic-fused heteroaryl or aryl compounds

Methods for preparation of quinazoline derivatives

Bicyclic-fused heteroaryl or aryl compounds

Quinazoline derivatives substituted by aniline, preparation method...

Method for preparing 1-(4-(4-(3,4-dichloro-2-fluorophenylamino)-7-m...

Bicyclic-fused heteroaryl or aryl compounds

Compounds and methods for enzyme-mediated tumor imaging and therapy

Fused heterocyclic compound

Morpholinylquinazolines

Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...

Compounds and methods for enzyme-mediated tumor imaging and therapy

Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...

Combination therapy of her expressing tumors

4-(tetrazol-5-yl)-quinazoline derivatives as anti-cancer agent

Sulphoximine-substituted quinoline and quinazoline derivatives as k...

Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...

Process for preparing quinazoline Rho-kinase inhibitors and interme...

Patents Applicationslast 30 patents

ANTI-WOLBACHIA PYRIDO[2,3-d]PYRIMIDINECOMPOUNDS

Bicyclic-Fused Heteroaryl or Aryl Compounds

TYROSINE KINASE INHIBITORS AND PHARMACEUTICAL APPLICATION THEREOF

4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR...

Bicyclic-Fused Heteroaryl or Aryl Compounds

ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...

COMPOUNDS

Bicyclic-Fused Heteroaryl or Aryl Compounds

ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...

ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...

ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...

Bicyclic-Fused Heteroaryl or Aryl Compounds

QUINAZOLINE DERIVATIVES SUBSTITUTED BY ANILINE, PREPARATION METHOD...

ACTIVATORS OF AUTOPHAGIC FLUX AND PHOSPHOLIPASE D AND CLEARANCE OF...

METHODS FOR PREPARATION OF QUINAZOLINE DERIVATIVES

4,6-DI- AND 2,4,6-TRISUBSTITUTED QUINAZOLINE DERIVATIVES USEFUL FOR...

Method For Preparing 1-(4-(4-(3,4-Dichloro-2-Fluorophenylamino)-7-M...

COMBINATION THERAPY OF HER EXPRESSING TUMORS

SUBSTITUTED PIPERAZINYL-PYRROLIDINE COMPOUNDS USEFUL AS CHEMOKINE R...

COMPOUNDS AND METHODS FOR ENZYME-MEDIATED TUMOR IMAGING AND THERAPY

QUINAZOLINE DERIVATIVES SUBSTITUTED BY ANILINE, PREPARATION METHOD...

SUBSTITUTED PIPERAZINYL-PYRROLIDINE COMPOUNDS USEFUL AS CHEMOKINE R...

Morpholinylquinazolines

COMBINATION THERAPY OF HER EXPRESSING TUMORS

Substituted piperazinyl-pyrrolidine compounds useful as chemokine r...

COMPOUNDS AS THE ESTROGEN RELATED RECEPTORS MODULATORS AND THE USES...

NOVEL 4-(TETRAZOL-5-YL)-QUINAZOLINE DERIVATIVES AS ANTI CANCER AGENT

PROCESS FOR PREPARING QUINAZOLINE RHO-KINASE INHIBITORS AND INTERME...

COMPOUNDS AND METHODS FOR ENZYME-MEDIATED TUMOR IMAGING AND THERAPY

Use of Oxindole Derivatives in the Treatment of Dementia Related Di...