Sundram et al. J. Am. Chem. Soc., vol. 118, No. 51, pp. 13107-13108, Dec. 1996.* |
Wang et al. Book of Abstracts, 213th ACS National Meeting, San Francisco, Apr. 13-17 (1997), CARB-064. American Chemical Society: Washington, D.C., Nov. 1997.* |
Brickner et al. J. Med. Chem. vol. 39, No. 3, pp. 673-679, Oct. 1997.* |
Rao et al. J. Am. Chem. Soc., vol. 119, No. 43, pp. 10286-10290, Oct. 1997.* |
Brickner, S. J., et al. “Synthesis and Antibacterial Activity of U-100592 and u-100766, Two Oxazolidinone Antibacterial Agents for the Potential Treatment of Multidrug-Resistant Gram-Positive Bacterial Infections.” J. Med. Chem. 39:673-679 (1986). |
Holmes, et al. “Novel Dimeric Penicillin Derived Inhibitors of HIV-1 Proteinase: Interaction with the Catalytic Aspartases.” Bioorg. Med. Chem. Lett. 3(4): 503-508 (1993). |
Portoghese, P.S. The Role of Concepts in Structure-Activity Relationship Studies of Opioid Ligands. J. med. Chem. 35(11): 1927-1937 (1992). |
Rao, et al. “Tight Binding of a Dimeric Dervative of Vancomycin with Dimeris L-Lys-D-Ala-D-Ala.” J. Am. Chem. Soc. 119(43): 10286-10290 (1997). |
Salvi, et al. “Formation of Bis (Fmoc-amino ethyl)-N-glycine derivatives by reductive amination of Fmoc-amino aldehydes with NaBH3CN.” Tetrahedron Letters. 35: 1181-1184 (1994). |
Shuker, et al. “Discovering High-Affinity Ligands for Proteins: SAR by NMR.” Science. 274: 1531-1534 (1996). |
Sundram, U.N., et al. “Novel Vancomycin Dimers with Activity againt Vancomycin-Resistant Enterococci.” J. Am. Chem. Soc. 118: 13107-13108 (1996). |
Tucker, J. A., et al. “Piperazinyl Oxazolidinone Antibacterial Agents Containing a pyridine, Diazene, or Triazene Heteroaromatic Ring.” J. Med Chem. 41:3727-3735 (1988). |
Zeng, et al. Automated Analytical/Preparative High-performance Liquid Chromatography-Mass Spectrometry System for the Rapid Characterization and Purification of Compound Libraries. J. Chrom. A. 794:3-13 (1998). |
Ahonkhai, V. I. et al. “In Vitro Activity of U-57930E, a New Clindamycin Analog, Against Aerobic Gram-Positive Bacteria.” Antimicrobial Agents and Chemotherapy. 21(6):902-905 (1982). |
Ballesta, J. P., et al. “Peptidyltransferase inhibitors: Structure-Activity Relationship Analysis by Chemical Modification.” The Ribosome. Ch. 44, pp 502-510, Hill, et al, eds. (1982). |
Barden, T. C., et al. “Glycylcyclines. 3. 9-Aminodoxycyclinecarboxamides.” J. Med. Chem. 37(20):3205-3211 (1994). |
Blackwood, R. K., et al. “Some Transformations of Tetracycline at the 4-Position.” Can. J. Chem. 43:1382-1388 (1965). |
Brenner, et al. “Encoded combinatorial chemistry.” Proc. Natl. Acad. Sci., USA. 89:5381-5383 (1992). |
CAS 1771-31-9, 53864—51-0. |
Cooperman, B.S. et al. “Antiobiotic Probes of Escherichia coli Ribosomal Peptidyltransferase.” The Ribosome. Ch. 42, pp 491-502, Hill, et al. eds. (1990). |
Cooperman. “Affintiy labelling of Ribosomes.” Methods Enzymol. 164: 341-361 (1988). |
Cundliffe, E. “Recognition Sites for Antibiotics within rRNA.” The Ribosome. Chapter 41, pp 479-510, Hill, et al. eds. (1990). |
Delaware, D. L., et al. “Aminoglycoside Antibiotics (Dihydrostreptomycin Analogues).” J. Antibiotics, XXXIX(2):251-258 91986). |
Herrinton, P. M., et al. “Oxidation and Alkylation of Spectinomycin Derivatives; Synthesis of Trospectomycin from Spectinomycin.” J. Org. Chem. 678-682 (1993). |
Jaynes, et al. “Photoinduced Affinity Labeling of the Escherichia coli Ribosome Puromycin Site.” Biochemistry. 17: 561-569 (1978). |
Kirst, Ph.D., H. A. “2 Semi-synthetic derivatives of Erythromycin.” Prog. Med. Chem., 30(2):57-88 (1993) (Ellis and Luscombe, eds.). |
Lemieux, R. U., et al. “The Chemistry of Streptomycin.” Advances in Carbohydrate Chemistry. 52:337-384 (1948). |
Mossa, J. S., et al. “Streptomycin.” Analytical Profiles of Drug Substances. 16:507, 531-535,587 (1987) (Flored, ed.). |
Rosenbrook, Jr., W., et al. “Spectinomycin Modification.” ACS Symposium, Series 125, 133-144 (1980). |
Spahn, C. M. T., et al. “Throwing a spanner in the works: antibiotics and the translation apparatus.” J. Mol. Med. 74:423-439 (1996). |
Thomas, R. C., et al. “Synthesis of Spectinomycin Analogs.” ACS Symposium, Series 125, 121-131 (1980). |
Tohma, S., et al. “Ashimycins A and B, new streptomycin Analogues.” J. Antibiotics. XLII(8):1205-1212 (1989). |
White, D. R., et al. “The Synthesis of Trospectomycin (6′-n-Propylspectinomycin, U-63,366F) From Spectinomycin.” Tetrahedron Letters. 30(12): 1469-1472 (1989). |