Number | Name | Date | Kind |
---|---|---|---|
4479941 | Veber et al. | Oct 1984 | |
4855303 | Hoover et al. | Aug 1989 | |
4857507 | Rosenberg et al. | Aug 1989 | |
4882420 | Thaisrivongs | Nov 1989 | |
4985407 | Foxton et al. | Jan 1991 |
Number | Date | Country |
---|---|---|
0222523 | May 1987 | EPX |
2171103 | Feb 1986 | GBX |
2196958 | Aug 1987 | GBX |
2203740 | Apr 1988 | GBX |
Entry |
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Plattner et al., J. Med. Chem. 1988, 31(12):2277-2288. |
Michael H. Gelb et al., "Fluoro Ketone Inhibitors of Hydrolytic Enzymes", Biochemistry, v. 24, No. 8, Apr. 9, 1985, pp. 1813 through 1817-M12. |
U.S. Ser. No. 07/384,236 filed Jul. 24, 1989, which is a CIP of 07/206,023 filed Jun. 17, 1988, now abandoned, which is a CIP of 07/113,772 filed Oct. 26, 1987, now abandoned. |