Balasaubramanian et al., J. Med. Chem., vol. 36, pp. 300-303 "Active Site-Directed Synthetic Thrombin Inhibitors: Synthesis, in Vitro . . . " (1993). |
Shuman et al., J. Med. Chem., vol. 36, pp. 314-319 "Highly Selective Tripeptide Thrombin Inhibitors" (1993). |
Kettner et al., The Journal of Biological Chemistry, vol. 265, pp. 18289-18297, "The Selective Inhibition of Thrombin by Peptides of Boroarginine" (1990). |
Okumura et al., The Journal of Biological Chemistry, vol. 263, pp. 3435-3443, "Platelet Glycocalicin--Interaction with Thrombin and Role as Thrombin Receptor . . . " (1978). |
Tollefsen et al., The Journal of Biological Chemistry, vol. 249, pp. 2646-2651, "The Binding of Thrombin to the Surface of Human Platelets" (1974). |
Vu et al., Cell, vol. 64, pp. 1057-1068, "Molecular Cloning of a Functional Thrombin Receptor Reveals a Novel Proteolytic . . . " (1991). |
Gronke et al., The Journal of Biological Chemistry, vol. 262, pp. 3030-3036, "Thrombin Interaction with Platelets" (1987). |
Workman, Jr. et al., vol. 252, p. 7118-7123, "Structure-Function Relationships Interaction of a-Thrombin with Blood Platelets" (1977). |
Hui et al., Biochemical and Biophysical Research Communications, vol. 184, pp. 790-796, "Minimal Sequence Requirement of Thrombin Receptor Agonist Peptide" (1992). |
Vassallo, Jr. et al., The Journal of Biological Chemistry, vol. 267, pp. 6081-6085, "Structure-Function Relationships in the Activation of Platelet . . . " (1992). |
Scarborough et al., The Journal of Biological Chemistry, vol. 267, pp. 13146-13149, "Tethered Ligand Agonist Peptides--Structure Requirements . . . " (1992). |
Iwanowicz et al., Organic & Medicinal Chemistry Letters, vol. 2, pp. 1607-1612, "a-Hydroxy- and a-ketoester Functionalized Thrombin Inhibitors" (1992). |
Edwards et al., J. Am. Chem. Soc., vol. 114, pp. 1854-1863, "Design, Synthesis, and Kinetic Evaluation of a Unique Class of Elastase Inhibitors . . . " (1992). |
Phillips, David R., Thrombos, Diathes. haemorrh. (Stuttg.), vol. 32, p. 207, "Thrombin Interation with Human Platelets Potentiation of Thrombin-induced . . . " (1974). |
Berndt, Michael C. and David R. Phillips, Platelets in Biology and Pathology, Chapter 3, pp. 43-75, "Platelet membrane proteins: composition and receptor function" (1981). |
Martin et al., Biochemistry, vol. 14, pp. 1308-1314, "Platelet Stimulation by Thrombin and Other Proteases" (1975). |
Greco et al., Blood, vol. 75, pp. 1983-1990, "PPACK-Thrombin Inhibits Thrombin-Induced Platelet" (1990). |
Bode et al., The EMBO Journal, vol. 8, pp. 3467-3475, "The refined 1.9 A crystal structure of human a-thrombin . . . " (1989). |
Tapparelli et al., TIPS, vol. 14, pp. 366-376, "Synthetic low-molecular weight thrombin inhibitors: molecular design and pharmaceological profile . . . " (1993). |
Hussain et al., Peptides, vol. 12, pp. 1153-1154, "Brief Communication--Anticoagulant Activity of a Peptide Boronic Acid Thrombin . . . " (1991). |