Claims
- 1. A compound selected from the group consisting of:
- AcSR.sup.2 SR.sup.1 Het and HalR.sup.2 SR.sup.1 Het wherein Ac is C.sub.1 -C.sub.12 acyl; Hal is halogen; R.sup.1 is a single bond or C.sub.1 -C.sub.4 alkylene; and R.sup.2 is a straight or branched C.sub.1 -C.sub.4 alkylene; Het is 1, 2, 3-triazol-4-yl, or a derivative which is optionally protected at a nitrogen atom by one or more protecting groups selected from C1-C8 alkyl, C7-C19 aralkyl; C1-C8 alkylthio; C6-C12 arylthio; C5-C8 cycloalkylidene; C2-C12 alkoxycarbonyl the alkyl of which is cyclic or acyclic, substituted or unsubstituted and is selected from the group consisting of methyl, ethyl, propyl, cyclopropylmethyl, cyclopropylethyl, isopropyl, butyl, isobutyl, pentyl, hexyl, trichloroethyl, pyridylmethyl, cyclopentyl or cyclohexyl; C8-C19 aralkoxycarbonyl the aralkyl of which is benzyl, benzhydryl or nitrobenzyl, C7-C15 aroyl; C3-C9 trialkylsilyl; C3-C9 alkoxydialkylsilyl; and an acid capable of forming acid addition salt.
- 2. The compound as claimed in claim 1 where R.sup.1 is a single bond.
- 3. The compound as claimed in claim 1 wherein R.sup.2 is methylene.
- 4. The compound as claimed in claim 1 wherein R.sup.2 is ethylidene.
- 5. The compound as claimed in claim 1 wherein Ac is acetyl.
- 6. The compound as claimed in claim 1 wherein Ac is benzoyl.
- 7. The compound as claimed in claim 1 wherein Hal is chloro.
Priority Claims (4)
Number |
Date |
Country |
Kind |
2-191899 |
Jul 1990 |
JPX |
|
2-289772 |
Oct 1990 |
JPX |
|
2-319578 |
Nov 1990 |
JPX |
|
3-147357 |
Jun 1991 |
JPX |
|
Parent Case Info
This is a divisional application of Ser. No. 07/729,413, filed Jul. 12, 1991 now U.S. Pat. No. 5,214,037.
US Referenced Citations (2)
Number |
Name |
Date |
Kind |
3481946 |
Schmidt et al. |
Dec 1969 |
|
4482565 |
Foglio et al. |
Nov 1984 |
|
Foreign Referenced Citations (3)
Number |
Date |
Country |
0210078 |
Jan 1987 |
EPX |
329457 |
Aug 1989 |
EPX |
2140807 |
Dec 1984 |
GBX |
Divisions (1)
|
Number |
Date |
Country |
Parent |
729413 |
Jul 1991 |
|