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Christoph Wolfgang Zapf
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Marlborough, MA, US
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Patents Grants
last 30 patents
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
12,202,836
Issue date
Jan 21, 2025
Pfizer Inc.
John David Trzupek
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Cyano cyclobutyl compounds for Cbl-b inhibition and uses thereof
Patent number
12,049,471
Issue date
Jul 30, 2024
NURIX THERAPEUTICS, INC.
Arthur T. Sands
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3-substituted piperidine compounds for Cbl-b inhibition, and use th...
Patent number
11,951,133
Issue date
Apr 9, 2024
NURIX THERAPEUTICS, INC.
Arthur T. Sands
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
11,702,424
Issue date
Jul 18, 2023
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Cyano cyclobutyl compounds for CBL-B inhibition and uses thereof
Patent number
11,530,229
Issue date
Dec 20, 2022
NURIX THERAPEUTICS, INC.
Arthur T. Sands
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3-substituted piperidine compounds for Cbl-b inhibition, and use th...
Patent number
11,464,802
Issue date
Oct 11, 2022
NURIX THERAPEUTICS, INC.
Arthur T. Sands
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Grant
Substituted benzyl-triazole compounds for Cbl-b inhibition, and fur...
Patent number
11,401,267
Issue date
Aug 2, 2022
NURIX THERAPEUTICS, INC.
Arthur T. Sands
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bruton's tyrosine kinase inhibitors
Patent number
10,815,213
Issue date
Oct 27, 2020
Pfizer Inc.
John Robert Springer
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
10,793,579
Issue date
Oct 6, 2020
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bicyclic heteroaryl derivatives as CFTR potentiators
Patent number
10,766,904
Issue date
Sep 8, 2020
CYSTIC FIBROSIS FOUNDATION
Joseph Walter Strohbach
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrrolopyrimidines as CFTR potentiators
Patent number
10,494,374
Issue date
Dec 3, 2019
CYSTIC FIBROSIS FOUNDATION
Joseph Walter Strohbach
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic heteroaryl derivatives as CFTR potentiators
Patent number
10,377,762
Issue date
Aug 13, 2019
CYSTIC FIBROSIS FOUNDATION
Joseph Walter Strohbach
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
10,329,302
Issue date
Jun 25, 2019
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds as IRAK4 modulators
Patent number
10,316,018
Issue date
Jun 11, 2019
Pfizer Inc.
Katherine Lin Lee
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrrolopyrimidines as CFTR potentiators
Patent number
10,301,315
Issue date
May 28, 2019
Cystic Fibrosis Foundation Therapeutics, Inc.
Joseph Walter Strohbach
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bruton's tyrosine kinase inhibitors
Patent number
10,266,513
Issue date
Apr 23, 2019
Pfizer Inc.
John Robert Springer
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic heteroaryl derivatives as CFTR potentiators
Patent number
10,208,053
Issue date
Feb 19, 2019
Cystic Fibrosis Foundation Therapeutics, Inc.
Joseph Walter Strohbach
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds as IRAK4 modulators
Patent number
10,174,000
Issue date
Jan 8, 2019
Pfizer Inc.
Katherine Lin Lee
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic heteroaryl derivatives as CFTR potentiators
Patent number
10,131,670
Issue date
Nov 20, 2018
Cystic Fibrosis Foundation Therapeutics, Inc.
Joseph Walter Strohbach
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
9,879,022
Issue date
Jan 30, 2018
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bicyclic-fused heteroaryl or aryl compounds
Patent number
9,458,168
Issue date
Oct 4, 2016
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
CYANO CYCLOBUTYL COMPOUNDS FOR CBL-B INHIBITION AND USES THEREOF
Publication number
20240409555
Publication date
Dec 12, 2024
Nurix Therapeutics, Inc.
Arthur T. SANDS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
3-SUBSTITUTED PIPERIDINE COMPOUNDS FOR CBL-B INHIBITION, AND USE TH...
Publication number
20240293458
Publication date
Sep 5, 2024
Nurix Therapeutics, Inc.
Arthur T. SANDS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
Publication number
20230339960
Publication date
Oct 26, 2023
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Pyrrolopyrimidines as CFTR Potentiators
Publication number
20230250100
Publication date
Aug 10, 2023
CYSTIC FIBROSIS FOUNDATION
Joseph Walter Strohbach
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CYANO CYCLOBUTYL COMPOUNDS FOR CBL-B INHIBITION AND USES THEREOF
Publication number
20230212186
Publication date
Jul 6, 2023
Nurix Therapeutics, Inc.
Arthur T. SANDS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FUR...
Publication number
20230150991
Publication date
May 18, 2023
Nurix Therapeutics, Inc.
Arthur T. SANDS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
UREA, AMIDE, AND SUBSTITUTED HETEROARYL COMPOUNDS FOR CBL-B INHIBITION
Publication number
20220387395
Publication date
Dec 8, 2022
Nurix Therapeutics, Inc.
Arthur T. SANDS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3-SUBSTITUTED PIPERIDINE COMPOUNDS FOR CBL-B INHIBITION, AND USE TH...
Publication number
20220378839
Publication date
Dec 1, 2022
Nurix Therapeutics, Inc.
Arthur T. SANDS
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Application
INHIBITORS OF CBL-B AND METHODS OF USE THEREOF
Publication number
20220324835
Publication date
Oct 13, 2022
Nurix Therapeutics, Inc.
Paul A. BARSANTI
C12 - BIOCHEMISTRY BEER SPIRITS WINE VINEGAR MICROBIOLOGY ENZYMOLOGY MUTATION...
Information
Patent Application
Pyrrolopyrimidines as CFTR Potentiators
Publication number
20210171534
Publication date
Jun 10, 2021
CYSTIC FIBROSIS FOUNDATION
Joseph Walter Strohbach
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BENZYL-TRIAZOLE COMPOUNDS FOR CBL-B INHIBITION, AND FUR...
Publication number
20210053961
Publication date
Feb 25, 2021
Nurix Therapeutics, Inc.
Arthur T. SANDS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
CYANO CYCLOBUTYL COMPOUNDS FOR CBL-B INHIBITION AND USES THEREOF
Publication number
20210053986
Publication date
Feb 25, 2021
Nurix Therapeutics, Inc.
Arthur T. SANDS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bruton's Tyrosine Kinase Inhibitors
Publication number
20210002251
Publication date
Jan 7, 2021
Pfizer Inc.
John Robert Springer
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
Publication number
20200377511
Publication date
Dec 3, 2020
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3-SUBSTITUTED PIPERIDINE COMPOUNDS FOR CBL-B INHIBITION, AND USE OF...
Publication number
20200323904
Publication date
Oct 15, 2020
Nurix Therapeutics, Inc.
Arthur T. Sands
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
RORC2 INHIBITORS AND METHODS OF USE THEREOF
Publication number
20200039960
Publication date
Feb 6, 2020
Pfizer Inc.
Mark Edward Schnute
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRROLOPYRIMIDINES AS CFTR POTENTIATORS
Publication number
20200017512
Publication date
Jan 16, 2020
CYSTIC FIBROSIS FOUNDATION
Joseph Walter Strohbach
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC HETEROARYL DERIVATIVES AS CFTR POTENTIATORS
Publication number
20190330219
Publication date
Oct 31, 2019
CYSTIC FIBROSIS FOUNDATION
Joseph Walter Strohbach
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
Publication number
20190270751
Publication date
Sep 5, 2019
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRROLOPYRIMIDINES AS CFTR POTENTIATORS
Publication number
20190225621
Publication date
Jul 25, 2019
CYSTIC FIBROSIS FOUNDATION THERAPEUTICS INC.
Joseph Walter Strohbach
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bruton's Tyrosine Kinase Inhibitors
Publication number
20190202798
Publication date
Jul 4, 2019
Pfizer Inc.
John Robert Springer
C07 - ORGANIC CHEMISTRY
Information
Patent Application
RORC2 INHIBITORS AND METHODS OF USE THEREOF
Publication number
20190144429
Publication date
May 16, 2019
Pfizer Inc.
Mark Edward Schnute
Y02 - TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMA...
Information
Patent Application
BICYCLIC-FUSED HETEROARYL OR ARYL COMPOUNDS AS IRAK4 MODULATORS
Publication number
20190092750
Publication date
Mar 28, 2019
Pfizer Inc.
KATHERINE LIN LEE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC HETEROARYL DERIVATIVES AS CFTR POTENTIATORS
Publication number
20190016727
Publication date
Jan 17, 2019
Cystic Fibrosis Foundation Therapeutics, Inc.
Joseph Walter Strohbach
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC HETEROARYL DERIVATIVES AS CFTR POTENTIATORS
Publication number
20190016728
Publication date
Jan 17, 2019
Cystic Fibrosis Foundation Therapeutics, Inc.
Joseph Walter Strohbach
C07 - ORGANIC CHEMISTRY
Information
Patent Application
RORC2 INHIBITORS AND METHODS OF USE THEREOF
Publication number
20180282304
Publication date
Oct 4, 2018
Pfizer Inc.
Mark Edward Schnute
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC-FUSED HETEROARYL OR ARYL COMPOUNDS AS IRAK4 MODULATORS
Publication number
20180244646
Publication date
Aug 30, 2018
Pfizer Inc.
KATHERINE LIN LEE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC HETEROARYL DERIVATIVES AS CFTR POTENTIATORS
Publication number
20180170938
Publication date
Jun 21, 2018
Cystic Fibrosis Foundation Therapeutics, Inc.
Joseph Walter Strohbach
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRROLOPYRIMIDINES AS CFTR POTENTIATORS
Publication number
20180141954
Publication date
May 24, 2018
Cystic Fibrosis Foundation Therapeutics, Inc.
Joseph Walter Strohbach
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Bicyclic-Fused Heteroaryl or Aryl Compounds
Publication number
20180127432
Publication date
May 10, 2018
Pfizer Inc.
John David Trzupek
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE