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Gaston S. M. Diels
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Patents Grants
last 30 patents
Information
Patent Grant
Pyrazole derivatives as MALT1 inhibitors
Patent number
12,077,521
Issue date
Sep 3, 2024
JANSSEN PHARMACEUTICA NV
Tianbao Lu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Monocyclic and bicyclic ring system substituted carbanucleoside ana...
Patent number
11,993,614
Issue date
May 28, 2024
JANSSEN PHARMACEUTICA NV
Tongfei Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-6 bicyclic aromatic ring substituted nucleoside analogues for use...
Patent number
11,883,367
Issue date
Jan 30, 2024
JANSSEN PHARMACEUTICA NV
Tongfei Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
6-6 bicyclic aromatic ring substituted nucleoside analogues for use...
Patent number
11,318,157
Issue date
May 3, 2022
JANSSEN PHARMACEUTICA NV
Tongfei Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Monocyclic and bicyclic ring system substituted carbanucleoside ana...
Patent number
11,098,062
Issue date
Aug 24, 2021
JANSSEN PHARMACEUTICA NV
Tongfei Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazole derivatives as MALT1 inhibitors
Patent number
11,040,031
Issue date
Jun 22, 2021
JANSSEN PHARMACEUTICA NV
Tianbao Lu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazole derivatives as MALT1 inhibitors
Patent number
10,954,214
Issue date
Mar 23, 2021
JANSSEN PHARMACEUTICA NV
Tianbao Lu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted nucleoside analogues for use as PRMT5 inhibitors
Patent number
10,898,504
Issue date
Jan 26, 2021
JANSSEN PHARMACEUTICA NV
Didier Jean-Claude Berthelot
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazole derivatives as MALT1 inhibitors
Patent number
10,888,550
Issue date
Jan 12, 2021
JANSSEN PHARMACEUTICA NV
Tianbao Lu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-6 bicyclic aromatic ring substituted nucleoside analogues for use...
Patent number
10,653,711
Issue date
May 19, 2020
JANSSEN PHARMACEUTICA NV
Tongfei Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Macrocylic pyrimidine derivatives
Patent number
10,017,509
Issue date
Jul 10, 2018
JANSSEN PHARMACEUTICA NV
Gaston Stanislas Marcella Diels
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinazoline derivatives
Patent number
9,273,013
Issue date
Mar 1, 2016
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinazoline derivatives
Patent number
8,394,786
Issue date
Mar 12, 2013
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-azauracil derivatives as IL-5 inhibitors
Patent number
6,743,792
Issue date
Jun 1, 2004
Janssen Pharmaceutica N.V.
Eddy Jean Edgard Freyne
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
PDE IV inhibiting pyridine derivatives
Patent number
6,656,959
Issue date
Dec 2, 2003
JANSSEN PHARMACEUTICA NV
Eddy Jean Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,3-dihydro-1-(phenylalkyl)-2H-imidazol-2-one derivatves
Patent number
6,403,805
Issue date
Jun 11, 2002
JANSSEN PHARMACEUTICA NV
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,3-dihydro-1-(phenylalkyl)-2H-imidazol-2-one compounds and their u...
Patent number
5,994,376
Issue date
Nov 30, 1999
Janssen Pharmaceutica, N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,3-dihydro-1-(phenylalkenyl)-2H-imidazol-2-one derivatives having...
Patent number
5,952,510
Issue date
Sep 14, 1999
Janssen Pharmaceutica, N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,3-dihydro-2H-imidazol-2-one compounds
Patent number
5,869,515
Issue date
Feb 9, 1999
Janssen Pharmaceutica N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo [1,2-A] (pyrrolo, thieno or furano) [2,3-D] azepine derivat...
Patent number
5,629,308
Issue date
May 13, 1997
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo[2,1-b]benzazepine derivatives, compositions and method of use
Patent number
5,468,743
Issue date
Nov 21, 1995
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Imidazo[1,2-a](pyrrolo, thieno or furano) [3,2a-d]azepine derivativ...
Patent number
5,461,050
Issue date
Oct 24, 1995
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted thiazolyl and substituted pyridinyl derivatives
Patent number
5,360,807
Issue date
Nov 1, 1994
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Hydroxyalkylfuranyl derivatives
Patent number
5,272,150
Issue date
Dec 21, 1993
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
(4-piperidinylmethyl and -hetero)purines
Patent number
5,258,380
Issue date
Nov 2, 1993
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pharmacologically active (Bicyclic heterocyclyl)methyl and -hetero)...
Patent number
5,151,424
Issue date
Sep 29, 1992
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2-(heterocyclylalkyl)imidazopyridines
Patent number
5,086,056
Issue date
Feb 4, 1992
Janssen Pharmaceutica N.V.
Frans E. Janssens
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Anti-hystaminic [(bicyclic heterocyclyl) methyl and --hetero] subst...
Patent number
5,071,846
Issue date
Dec 10, 1991
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
(4-piperidinylmethyl and -hetero) purines
Patent number
5,041,448
Issue date
Aug 20, 1991
Janssen Pharmaceutica N.V.
Frans E. Janssens
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2-(heterocyclylalkyl)imidazopyridines for treating allergic diseases
Patent number
5,011,842
Issue date
Apr 30, 1991
Janssen Pharmaceutica N.V.
Frans E. Janssens
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
Information
Patent Application
MACROCYCLIC 2-ALLYLTETRAHYDROFURANS AS INHIBITORS OF MCL-1
Publication number
20240239812
Publication date
Jul 18, 2024
Janssen Pharmaceutica N.V.
Frederik Jan Rita ROMBOUTS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Monocyclic And Bicyclic Ring System Substituted Carbanucleoside Ana...
Publication number
20240124493
Publication date
Apr 18, 2024
Janssen Pharmaceutica N.V.
Tongfei Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC SPIROCYCLE DERIVATIVES AS MCL-1 INHIBITORS
Publication number
20240067660
Publication date
Feb 29, 2024
Janssen Pharmaceutica N.V.
Frederik Jan Rita ROMBOUTS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-6 BICYCLIC AROMATIC RING SUBSTITUTED NUCLEOSIDE ANALOGUES FOR USE...
Publication number
20230330127
Publication date
Oct 19, 2023
Janssen Pharmaceutica N.V.
Tongfei Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC-2-AMINO-3-FLUORO-BUT-3-ENAMIDES AS INHIBITORS OF MCL-1
Publication number
20230219906
Publication date
Jul 13, 2023
Janssen Pharmaceutica N.V.
Soufyan JERHAOUI
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL 6-6 BICYCLIC AROMATIC RING SUBSTITUTED NUCLEOSIDE ANALOGUES F...
Publication number
20230071711
Publication date
Mar 9, 2023
Janssen Pharmaceutica N.V.
Tongfei Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLE DERIVATIVES AS MALT1 INHIBITORS
Publication number
20220315557
Publication date
Oct 6, 2022
Janssen Pharmaceutica N.V.
Tianbao LU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRIDINE RINGS CONTAINING DERIVATIVES AS MALT1 INHIBITORS
Publication number
20220162187
Publication date
May 26, 2022
Johannes Wilhelmus J. THURING
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel Monocyclic And Bicyclic Ring System Substituted Carbanucleosi...
Publication number
20210371433
Publication date
Dec 2, 2021
Janssen Pharmaceutica N.V.
Tongfei Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL 6-6 BICYCLIC AROMATIC RING SUBSTITUTED NUCLEOSIDE ANALOGUES F...
Publication number
20200360416
Publication date
Nov 19, 2020
Janssen Pharmaceutica N.V.
Tongfei Wu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL SUBSTITUTED NUCLEOSIDE ANALOGUES FOR USE AS PRMT5 INHIBITORS
Publication number
20200289539
Publication date
Sep 17, 2020
Janssen Pharmaceutica N.V.
Didier Jean-Claude BERTHELOT
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLE DERIVATIVES AS MALT1 INHIBITORS
Publication number
20190381012
Publication date
Dec 19, 2019
Janssen Pharmaceutica N.V.
Tianbao LU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLE DERIVATIVES AS MALT1 INHIBITORS
Publication number
20190381019
Publication date
Dec 19, 2019
Janssen Pharmaceutica N.V.
Tianbao Lu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL MONOCYCLIC AND BICYCLIC RING SYSTEM SUBSTITUTED CARBANUCLEOSI...
Publication number
20190263833
Publication date
Aug 29, 2019
Janssen Pharmaceutica N.V.
Tongfei WU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL 6-6 BICYCLIC AROMATIC RING SUBSTITUTED NUCLEOSIDE ANALOGUES F...
Publication number
20180243328
Publication date
Aug 30, 2018
Janssen Pharmaceutica N.V.
Tongfei Wu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLE DERIVATIVES AS MALT1 INHIBITORS
Publication number
20180170909
Publication date
Jun 21, 2018
JANSSEN BIOTECH, INC.
Tianbao Lu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYLIC PYRIMIDINE DERIVATIVES
Publication number
20170022202
Publication date
Jan 26, 2017
Janssen Pharmaceutica N.V.
Gaston Stanislas Marcella DIELS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYLIC PYRIDINE DERIVATIVES
Publication number
20170022201
Publication date
Jan 26, 2017
Janssen Pharmaceutica N.V.
Gaston Stanislas Marcella Diels
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINAZOLINE DERIVATIVES
Publication number
20160207938
Publication date
Jul 21, 2016
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINAZOLINE DERIVATIVES
Publication number
20130178624
Publication date
Jul 11, 2013
Janssen Pharmaceutica N.V.
Eddy Jean Edgard FREYNE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Dimeric Compounds Of Piperidine, Piperazine Or Morpholine Or Their...
Publication number
20070299109
Publication date
Dec 27, 2007
Miroslav Cik
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Pyrrolopyrimidine Derivatives
Publication number
20070270588
Publication date
Nov 22, 2007
TAISHO PHARMACEUTICAL CO., LTD.
Francois P. Bischoff
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Macrocyclic quinazoline derivatives as antiproliferative agents
Publication number
20060247237
Publication date
Nov 2, 2006
Janssen Pharmaceutica N.V.
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Heteroaryl amines as glycogen synthase kinase 3beta inhibitors (gsk...
Publication number
20050004125
Publication date
Jan 6, 2005
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6-Azauracil derivatives as IL-5 inhibitors
Publication number
20030220331
Publication date
Nov 27, 2003
Eddy Jean Edgard Freyne
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
6-azauracil derivatives as IL-5 inhibitors
Publication number
20020042416
Publication date
Apr 11, 2002
Eddy Jean Edgard Freyne
C07 - ORGANIC CHEMISTRY