Membership
Tour
Register
Log in
Gregor James MacDonald
Follow
Person
Ranst, BE
People
Overview
Industries
Organizations
People
Information
Impact
Patents Grants
last 30 patents
Information
Patent Grant
1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′]bipyri...
Patent number
11,071,729
Issue date
Jul 27, 2021
Addex Pharmaceuticals SA
Jose Maria Cid-Nunez
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 6,7-dihydropyrazolo[1,5-a]pyrazines as negative alloste...
Patent number
10,584,129
Issue date
Mar 10, 2020
Janssen Pharmaceuticals NV
Sergio-Alvar Alonso-de Diego
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted 6,7-dihydropyrazolo[1,5-a]pyrazines as negative alloste...
Patent number
10,106,542
Issue date
Oct 23, 2018
JANSSEN PHARMACEUTICA NV
Sergio-Alvar Alonso-de Diego
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
5,6-dihydro-2H-[1,4]oxazin-3-yl-amine derivatives useful as inhibit...
Patent number
9,828,350
Issue date
Nov 28, 2017
JANSSEN PHARMACEUTICA NV
Andrés Avelino Trabanco-Suárez
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperidin-4YL-pyridazin-3-ylamine derivatives as fast dissociating...
Patent number
9,751,860
Issue date
Sep 5, 2017
Janssen Pharmaceutica NV
Marcel Frans Leopold De Bruyn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1,2,4-triazolo [4,3-A] pyridine derivatives and their use for the t...
Patent number
9,737,533
Issue date
Aug 22, 2017
Janssen Pharmaceuticals. Inc.
Jose Maria Cid-Nunez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Piperidin-4-yl-pyridazin-3-ylamine derivatives as fast dissociating...
Patent number
9,468,640
Issue date
Oct 18, 2016
Janssen Pharmaceutica N.V.
Marcel Frans Leopold De Bruyn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Fast-dissociating dopamine 2 receptor antagonists
Patent number
9,422,296
Issue date
Aug 23, 2016
JANSSEN PHARMACEUTICA NV
Gregor James Macdonald
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
2-aniline-4-aryl substituted thiazole derivatives
Patent number
9,388,175
Issue date
Jul 12, 2016
JANSSEN PHARMACEUTICA NV
Johannes Wilhelmus John F. Thuring
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive...
Patent number
9,271,967
Issue date
Mar 1, 2016
Janssen Pharmaceuticals, Inc.
José Maria Cid-Núñez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1, 4-disubstituted 3-cyano-pyridone derivatives and their use as po...
Patent number
9,266,834
Issue date
Feb 23, 2016
Janssen Pharmaceuticals, Inc.
Hassan Julien Imogai
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted pyrazolo[1,5-a]pyrazines as mGluR5 receptor modulators
Patent number
9,255,103
Issue date
Feb 9, 2016
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,2,4-triazolo [4,3-a] pyridine derivatives and their use for the t...
Patent number
9,226,930
Issue date
Jan 5, 2016
Janssen Pharmaceuticals, Inc.
Jose Maria Cid-Nunez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrido[1,2-a]pyrazines and substituted pyrido[1,2-a][1,...
Patent number
9,181,245
Issue date
Nov 10, 2015
Janssen Pharmaceuticals, Inc.
Frederik Jan Rita Rombouts
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Bicyclic thiazoles as allosteric modulators of mGluR5 receptors
Patent number
9,174,953
Issue date
Nov 3, 2015
JANSSEN PHARMACEUTICA NV
Gregor James MacDonald
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′]bipyri...
Patent number
9,132,122
Issue date
Sep 15, 2015
Janssen Pharmaceuticals, Inc.
Jose Maria Cid-Nunez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1′,3′-disubstituted-4-phenyl-3,4,5,6-tetrahydro-2H,1′H-[1,4′] bipyr...
Patent number
9,114,138
Issue date
Aug 25, 2015
Janssen Pharmaceuticals, Inc.
Jose Maria Cid-Nunez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bicyclic oxazole and thiazole compounds and their use as allosteric...
Patent number
9,090,632
Issue date
Jul 28, 2015
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
7-aryl-1,2,4-triazolo[4,3-A]pyridine derivatives and their use as p...
Patent number
9,085,577
Issue date
Jul 21, 2015
Janssen Pharmaceuticals, Inc.
Jose Maria Cid-Nunez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1,4-disubstituted 3-cyano-pyridone derivatives and their use as pos...
Patent number
9,067,891
Issue date
Jun 30, 2015
Janssen Pharmaceuticals, Inc.
Jose Maria Cid-Nunez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Bicyclic thiazoles as allosteric modulators of mGluR5 receptors
Patent number
9,040,707
Issue date
May 26, 2015
JANSSEN PHARMACEUTICA NV
Gregor James MacDonald
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted bicyclic alkoxy pyrazole analogs as allosteric modulato...
Patent number
9,029,366
Issue date
May 12, 2015
Vanderbilt University
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive...
Patent number
9,012,448
Issue date
Apr 21, 2015
Janssen Pharmaceuticals, Inc.
José Maria Cid-Núñez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1,2,4-triazolo[4,3-a] pyridine derivatives and their use as positiv...
Patent number
8,993,591
Issue date
Mar 31, 2015
Janssen Pharmaceuticals, Inc.
José Maria Cid-Núñez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1,2,4-triazolo[4,3-a]pyridine derivatives and their use as positive...
Patent number
8,946,205
Issue date
Feb 3, 2015
Janssen Pharmaceuticals, Inc.
Jose Maria Cid-Nunez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted bicyclic heterocyclic compounds as gamma secretase modu...
Patent number
8,946,426
Issue date
Feb 3, 2015
Janssen Pharmaceuticals, Inc.
Henricus Jacobus Maria Gijsen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperidin-4-yl-pyridazin-3-ylamine derivatives as fast dissociating...
Patent number
8,940,743
Issue date
Jan 27, 2015
JANSSEN PHARMACEUTICA NV
Marcel Frans Leopold De Bruyn
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
1,2,4-triazolo [4,3-A] pyridine derivatives and their use for the t...
Patent number
8,937,060
Issue date
Jan 20, 2015
Janssen Pharmaceuticals, Inc.
Jose Maria Cid-Nunez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Thia(dia)zoles as fast dissociating dopamine 2 receptor antagonists
Patent number
8,933,101
Issue date
Jan 13, 2015
JANSSEN PHARMACEUTICA NV
Gregor James MacDonald
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4-alkoxypyridazine derivatives as fast dissociating dopamine 2 rece...
Patent number
8,906,921
Issue date
Dec 9, 2014
JANSSEN PHARMACEUTICA NV
Gregor James MacDonald
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
1',3'-Disubstituted-4-Phenyl-3,4,5,6-Tetrahydro-2H,1'H-[1,4']Bipyri...
Publication number
20220000856
Publication date
Jan 6, 2022
JANSSEN PHARMACEUTICALS, INC
Jose Maria Cid-Nunez
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1',3'-Disubstituted-4-Phenyl-3,4,5,6-Tetrahydro-2H,1'H-[1,4']Bipyri...
Publication number
20200038391
Publication date
Feb 6, 2020
JANSSEN PHARMACEUTICALS, INC
Jose Maria Cid-Nunez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZINES AS NEGATIVE ALLOSTE...
Publication number
20190055257
Publication date
Feb 21, 2019
Janssen Pharmaceutica N.V.
Sergio-Alvar Alonso-de Diego
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FAST DISSOCIATING DOPAMINE 2 RECEPTOR ANTAGONISTS
Publication number
20170022181
Publication date
Jan 26, 2017
Marcel Frans Leopold De Bruyn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
5,6-DIHYDRO-2H-[1,4]OXAZIN-3-YL-AMINE DERIVATIVES USEFUL AS INHIBIT...
Publication number
20160152581
Publication date
Jun 2, 2016
Janssen Pharmaceutica NV
Andrés Avelino Trabanco-Suárez
C07 - ORGANIC CHEMISTRY
Information
Patent Application
6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE...
Publication number
20160115169
Publication date
Apr 28, 2016
Janssen Pharmaceutica N.V.
Sergio-Alvar Alonso-de Diego
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1,2,4-Triazolo [4,3-A] Pyridine Derivatives and Their Use For The T...
Publication number
20160067245
Publication date
Mar 10, 2016
JANSSEN PHARMACEUTICALS, INC
JOSE MARIA CID-NUNEZ
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1',3'-Disubstituted-4-Phenyl-3,4,5,6-Tetrahydro-2H,1'H-[1,4']Bipyri...
Publication number
20150336930
Publication date
Nov 26, 2015
JANSSEN PHARMACEUTICALS, INC
JOSE MARIA CID-NUNEZ
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BICYCLIC ALKOXY PYRAZOLE ANALOGS AS ALLOSTERIC MODULATO...
Publication number
20150216863
Publication date
Aug 6, 2015
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1,2,4-Triazolo [4,3-A] Pyridine Derivatives and Their Use For The T...
Publication number
20150141403
Publication date
May 21, 2015
Jose Maria CID-NUNEZ
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PIPERIDIN-4-YL-PYRIDAZIN-3-YLAMINE DERIVATIVES AS FAST DISSOCIATING...
Publication number
20150141432
Publication date
May 21, 2015
Janssen Pharmaceutica N.V.
Marcel Frans, Leopold De Bruyn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED 3,4-DIHYDRO-2H-PYRIDO[1,2-A]PYRAZINE-1,6-DIONE DERIVATI...
Publication number
20150141411
Publication date
May 21, 2015
JANSSEN PHARMACEUTICALS, INC
Frederik Jan Rita Rombouts
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL SUBSTITUTED BICYCLIC HETEROCYCLIC COMPOUNDS AS GAMMA SECRETAS...
Publication number
20150094311
Publication date
Apr 2, 2015
CELLZOME LIMITED
HENRICUS JACOBUS MARIA GIJSEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
FAST-DISSOCIATING DOPAMINE 2 RECEPTOR ANTAGONISTS
Publication number
20140336381
Publication date
Nov 13, 2014
Gregor James Macdonald
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED IMIDAZOPYRIMIDIN-5(6H)-ONES AS ALLOSTERIC MODULATORS OF...
Publication number
20140329838
Publication date
Nov 6, 2014
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1, 4-Disubstituted 3-Cyano-Pyridone Derivatives and Their Use As Po...
Publication number
20140315903
Publication date
Oct 23, 2014
HASSAN JULIEN IMOGAI
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC PYRAZOLE COMPOUNDS AS ALLOSTERIC MODULATORS OF MGLUR5 RECE...
Publication number
20140213593
Publication date
Jul 31, 2014
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
7-ARYL-1,2,4-TRIAZOLO[4,3-A]PYRIDINE DERIVATIVES AND THEIR USE AS P...
Publication number
20140200208
Publication date
Jul 17, 2014
ADDEX PHARMA, S.A.
JOSE MARIA CID-NUNEZ
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE...
Publication number
20140155393
Publication date
Jun 5, 2014
JANSSEN PHARMACEUTICALS, INC
José Maria Cid-Núñez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BICYCLIC TRIAZOLE AND PYRAZOLE LACTAMS AS ALLOSTERIC MODULATORS OF...
Publication number
20140057870
Publication date
Feb 27, 2014
Vanderbilt University
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED BICYCLIC CYCLOALKYL PYRAZOLE LACTAM ANALOGS AS ALLOSTER...
Publication number
20130345204
Publication date
Dec 26, 2013
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BICYCLIC ALKOXY PYRAZOLE ANALOGS AS ALLOSTERIC MODULATO...
Publication number
20130345206
Publication date
Dec 26, 2013
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BICYCLIC ARALKYL PYRAZOLE LACTAM ANALOGS AS ALLOSTERIC...
Publication number
20130345205
Publication date
Dec 26, 2013
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED BICYCLIC ALKOXY PYRAZOLE ANALOGS AS ALLOSTERIC MODULATO...
Publication number
20130345203
Publication date
Dec 26, 2013
P. Jeffrey Conn
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE...
Publication number
20130338185
Publication date
Dec 19, 2013
JANSSEN PHARMACEUTICALS, INC
José Maria Cid-Núñez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BRIDGED ARYL PIPERAZINES DERIVATIVES USEFUL FOR THE TREATMENT OF CN...
Publication number
20130331395
Publication date
Dec 12, 2013
Janssen Pharmaceutica N.V.
Christopher Creighton
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BICYCLIC OXAZOLE LACTAMS AS ALLOSTERIC MODULATORS OF MGLUR5 RECEPTORS
Publication number
20130252943
Publication date
Sep 26, 2013
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1,2,4-TRIAZOLO[4,3-a]PYRIDINE DERIVATIVES AND THEIR USE AS POSITIVE...
Publication number
20130252952
Publication date
Sep 26, 2013
JANSSEN PHARMACEUTICALS, INC
José Maria Cid-Núñez
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED IMIDAZOPYRIMIDIN-5(6H)-ONES AS ALLOSTERIC MODULATORS OF...
Publication number
20130245043
Publication date
Sep 19, 2013
P. Jeffrey Conn
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1',3'-DISUBSTITUTED-4-PHENY-3,4,5,6-TETRAHYDRO-2H,1'H-[1,4']BIPYRID...
Publication number
20130196992
Publication date
Aug 1, 2013
Addex Pharmaceuticals SA
Jose Maria CID-NUNEZ
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE