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Methvin Isaac
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Ontario, CA
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Patents Grants
last 30 patents
Information
Patent Grant
Substituted heteroaryls as inhibitors of the BCL6 BTB domain protei...
Patent number
11,518,764
Issue date
Dec 6, 2022
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Rima Al-awar
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Deuterated compounds as inhibitors of the BCL6 BTB domain protein-p...
Patent number
11,505,539
Issue date
Nov 22, 2022
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Methvin Isaac
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted carboxamides as inhibitors of WDR5 protein-protein binding
Patent number
11,319,299
Issue date
May 3, 2022
Propellon Therapeutics Inc.
Rima Al-Awar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Tricyclic inhibitors of the BCL6 BTB domain protein-protein interac...
Patent number
11,242,351
Issue date
Feb 8, 2022
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Rima Al-awar
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Quinolone compounds as inhibitors of the BCL6 BTB domain protein-pr...
Patent number
11,192,880
Issue date
Dec 7, 2021
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Methvin Isaac
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted carboxamides as inhibitors of WDR5 protein-protein binding
Patent number
11,174,250
Issue date
Nov 16, 2021
Propellon Therapeutics Inc.
Rima Al-Awar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Use of D-serine derivatives for the treatment of anxiety disorders
Patent number
8,450,336
Issue date
May 28, 2013
NPS Pharmaceuticals, Inc.
Guy Higgins
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Oxadiazole derivatives and their use as metabotropic glutamate rece...
Patent number
8,377,940
Issue date
Feb 19, 2013
Astrazeneca AB
Joshua Clayton
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Oxadiazole derivatives and their use as metabotropic glutamate rece...
Patent number
8,377,939
Issue date
Feb 19, 2013
Astrazeneca AB
Joshua Clayton
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Metabotropic glutamate-receptor-potentiating isoindolones
Patent number
8,153,638
Issue date
Apr 10, 2012
Astrazeneca AB
Bradford Van Wagenen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Isoindolone compounds and their use as metabotropic glutamate recep...
Patent number
7,968,570
Issue date
Jun 28, 2011
Astrazeneca AB
Joshua Clayton
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pharmaceutically active compounds containing tetrazolyl and triazol...
Patent number
7,960,422
Issue date
Jun 14, 2011
Astrazeneca AB
Erwan Arzel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Piperazines and piperidines as Mglur5 potentiators
Patent number
7,935,703
Issue date
May 3, 2011
Astrazeneca AB
Abdelmalik Slassi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted isoindolones and their use as metabotropic glutamate re...
Patent number
7,868,008
Issue date
Jan 11, 2011
Astrazeneca AB
Bradford Van Wagenen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Oxazolidinone compounds and their use as metabotropic glutamate rec...
Patent number
7,816,354
Issue date
Oct 19, 2010
Astrazeneca AB
Abdelmalik Slassi
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Metabotropic glutamate-receptor-potentiating isoindolones
Patent number
7,807,706
Issue date
Oct 5, 2010
Astrazeneca AB
Bradford Van Wagenen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Metabotropic glutamate receptor oxadiazole ligands and their use as...
Patent number
7,799,792
Issue date
Sep 21, 2010
Astrazeneca AB
Joshua Clayton
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Spiro-oxazolidinone compounds and their use as metabotropic glutama...
Patent number
7,790,717
Issue date
Sep 7, 2010
Astrazeneca AB
Ian Egle
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
mGluR5 modulators
Patent number
7,772,235
Issue date
Aug 10, 2010
Astrazeneca AB
Methvin Isaac
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tetrazole compounds and their use as metabotropic glutamate recepto...
Patent number
7,691,892
Issue date
Apr 6, 2010
Astrazeneca AB
Martin Johansson
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
MGluR5 modulators I
Patent number
7,678,796
Issue date
Mar 16, 2010
Astrazeneca AB
Andreas Wallberg
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Additional heteropolycyclic compounds and their use as metabotropic...
Patent number
7,585,881
Issue date
Sep 8, 2009
Astrazeneca AB
Louise Edwards
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Fused heterocyclic compounds and their use as metabotropic glutamat...
Patent number
7,576,077
Issue date
Aug 18, 2009
Astrazeneca AB
David Wensbo
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Spiro-oxazolidinone compounds and their use as metabotropic glutama...
Patent number
7,485,722
Issue date
Feb 3, 2009
Astrazeneca AB
Ian Egle
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds for the treatment of neurological, psychiatric or pain di...
Patent number
7,476,684
Issue date
Jan 13, 2009
Astrazeneca AB
Alexander Minidis
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds
Patent number
7,456,200
Issue date
Nov 25, 2008
Astrazeneca AB
Jalaj Arora
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heteropolycyclic compounds and their use as metabotropic glutamate...
Patent number
7,112,595
Issue date
Sep 26, 2006
NPS Pharmaceuticals, Inc.
Bradford Van Wagenen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds
Patent number
7,074,809
Issue date
Jul 11, 2006
AstraZeneca AB
Jalaj Arora
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Compounds having 5-HT6 receptor antagonist activity
Patent number
6,897,215
Issue date
May 24, 2005
NPS Allelix Corp.
Tao Xin
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heterocyclic compounds for the treatment of migraine
Patent number
6,716,837
Issue date
Apr 6, 2004
NPS Allelix Biopharmaceuticals, Inc.
Louise Edwards
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
HALO-SUBSTITUTED AMINO AZA-HETEROARYL COMPOUNDS AS INHIBITORS OF TH...
Publication number
20240425479
Publication date
Dec 26, 2024
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Ahn Chau
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HALO-SUBSTITUTED AMINO PYRIDINE COMPOUNDS AS INHIBITORS OF THE HAEM...
Publication number
20240343704
Publication date
Oct 17, 2024
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Anh Chau
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED AMINO AZA-HETEROARYL COMPOUNDS AS INHIBITORS OF THE HAE...
Publication number
20240317723
Publication date
Sep 26, 2024
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Rima Al-Awar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ERGOLINE-DERIVED AGONISTS OF THE 5-HT2A RECEPTOR
Publication number
20240279226
Publication date
Aug 22, 2024
Diamond Therapeutics Inc.
Methvin ISAAC
C07 - ORGANIC CHEMISTRY
Information
Patent Application
5-HT2A AND/OR 5-HT2C RECEPTOR AGONISTS
Publication number
20240182480
Publication date
Jun 6, 2024
Diamond Therapeutics Inc.
Methvin ISAAC
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ISOINDOLINONE AMINOPYRIMIDINE COMPOUNDS AS INHIBITORS OF NUAK KINAS...
Publication number
20240092763
Publication date
Mar 21, 2024
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Rima Al-Awar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
THIENYL AND CYCLOALKYL AMINOPYRIMIDINE COMPOUNDS AS INHIBITORS OF N...
Publication number
20240025887
Publication date
Jan 25, 2024
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Rima Al-Awar
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED CARBOXAMIDES AS INHIBITORS OF WDR5 PROTEIN-PROTEIN BINDING
Publication number
20230219926
Publication date
Jul 13, 2023
Propellon Therapeutics Inc.
Rima AL-AWAR
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TRICYCLIC INHIBITORS OF THE BCL6 BTB DOMAIN PROTEIN-PROTEIN INTERAC...
Publication number
20210053978
Publication date
Feb 25, 2021
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Rima Al-awar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INHIBITORS OF WDR5 PROTEIN-PROTEIN BINDING
Publication number
20200385371
Publication date
Dec 10, 2020
PROPELLON THERAPEUTICS INC.
Rima Al-Awar
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INHIBITORS OF THE BCL6 BTB DOMAIN PROTEIN-PROTEIN INTERACTION AND U...
Publication number
20200331921
Publication date
Oct 22, 2020
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Rima Al-awar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL QUINOLONE COMPOUNDS AS INHIBITORS OF THE BCL6 BTB DOMAIN PROT...
Publication number
20200325119
Publication date
Oct 15, 2020
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Methvin Isaac
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL DEUTERATED COMPOUNDS AS INHIBITORS OF THE BCL6 BTB DOMAIN PRO...
Publication number
20200308147
Publication date
Oct 1, 2020
ONTARIO INSTITUTE FOR CANCER RESEARCH (OICR)
Methvin Isaac
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INHIBITORS OF WDR5 PROTEIN-PROTEIN BINDING
Publication number
20190119264
Publication date
Apr 25, 2019
PROPELLON THERAPEUTICS INC.
Rima Al-Awar
C07 - ORGANIC CHEMISTRY
Information
Patent Application
INHIBITORS OF WDR5 PROTEIN-PROTEIN BINDING
Publication number
20190112290
Publication date
Apr 18, 2019
PROPELLON THERAPEUTICS INC.
Rima Al-Awar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
USE OF D-SERINE DERIVATIVES FOR THE TREATMENT OF ANXIETY DISORDERS
Publication number
20140018549
Publication date
Jan 16, 2014
NPS Pharmaceuticals, Inc.
Guy Higgins
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Substituted Isoindolones and Their Use as Metabotropic Glutamate Re...
Publication number
20110166155
Publication date
Jul 7, 2011
Bradford Van Wagenen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AZA-Isoindolones and Their Use as Metabotropic Glutamate Receptor P...
Publication number
20110053953
Publication date
Mar 3, 2011
Abdelmalik Slassi
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Metabotropic Glutamate-Receptor-Potentiating Isoindolones
Publication number
20100317674
Publication date
Dec 16, 2010
Bradford Van Wagenen
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Metabotropic Glutamate Receptor Oxadiazole Ligands and Their Use as...
Publication number
20100280082
Publication date
Nov 4, 2010
AstraZeneca AB
Joshua Clayton
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Oxadiazole Derivatives and Their Use as Metabotropic Glutamate Rece...
Publication number
20100267740
Publication date
Oct 21, 2010
AstraZeneca AB
Joshua Clayton
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Piperazine and Piperidine MGLUR5 Potentiators
Publication number
20100144710
Publication date
Jun 10, 2010
AstraZeneca AB
Jalaj Arora
C07 - ORGANIC CHEMISTRY
Information
Patent Application
USE OF D-SERINE DERIVATIVES FOR THE TREATMENT OF ANXIETY DISORDERS
Publication number
20100016403
Publication date
Jan 21, 2010
Guy Higgins
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TETRAHYDRO-5H-PYRIDO[2,3-D]AZEPINES AS 5-HT2C LIGANDS
Publication number
20090312306
Publication date
Dec 17, 2009
Guangri Sun
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Isoindolone compounds and their use as metabotropic glutamate recep...
Publication number
20090275578
Publication date
Nov 5, 2009
AstraZeneca AB
Joshua Clayton
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Bicyclic Benzimidazole Compounds and Their Use as Metabotropic Glut...
Publication number
20090192169
Publication date
Jul 30, 2009
Ian Egle
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Metabotropic Glutamate Receptor-Potentiating Isoindolones
Publication number
20090149505
Publication date
Jun 11, 2009
AstraZeneca AB
James R. Empfield
C07 - ORGANIC CHEMISTRY
Information
Patent Application
New compounds 067
Publication number
20090131454
Publication date
May 21, 2009
AstraZeneca AB
Erwan Arzel
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SPIRO-OXAZOLIDINONE COMPOUNDS AND THEIR USE AS METABOTROPIC GLUTAMA...
Publication number
20090124578
Publication date
May 14, 2009
AstraZeneca AB
Ian EGLE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMINO 1,2,4-TRIAZOLE DERIVATIVES AS MODULATORS OF MGLUR5
Publication number
20090111821
Publication date
Apr 30, 2009
AstraZeneca AB
Methvin ISAAC
C07 - ORGANIC CHEMISTRY