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Wuppertal, DE
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last 30 patents
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Patent Grant
Macrocyclic fluorine substituted indole derivatives
Patent number
12,152,041
Issue date
Nov 26, 2024
The Broad Institute, Inc.
Steven James Ferrara
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted macrocyclic indole derivatives
Patent number
11,891,404
Issue date
Feb 6, 2024
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocyclic indole derivatives
Patent number
11,492,358
Issue date
Nov 8, 2022
The Broad Institute, Inc.
Sarah Anna Liesa Johannes
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Macrocyclic chlorine substituted indole derivatives
Patent number
11,478,451
Issue date
Oct 25, 2022
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocyclic chlorine substituted indole derivatives
Patent number
11,447,504
Issue date
Sep 20, 2022
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted macrocyclic indole derivatives
Patent number
11,440,923
Issue date
Sep 13, 2022
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocyclic indole derivatives
Patent number
11,401,278
Issue date
Aug 2, 2022
The Broad Institute, Inc.
Laura Furst
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Macrocyclic fluorine substituted indole derivatives
Patent number
11,286,263
Issue date
Mar 29, 2022
The Broad Institute, Inc.
Steven James Ferrara
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocyclic indole derivatives
Patent number
10,981,932
Issue date
Apr 20, 2021
Bayer Aktiengesellschaft
Sarah Anna Liesa Johannes
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted piperidinyl tetrahydroquinolines
Patent number
10,961,221
Issue date
Mar 30, 2021
Bayer Pharma Aktiengesellschaft
Eva Maria Becker-Pelster
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Amino-substituted imidazo[1,2-A] pyridinecarboxamides and their use
Patent number
10,662,185
Issue date
May 26, 2020
Bayer Pharma Aktiengesellschaft
Alexandros Vakalopoulos
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted piperidinyl tetrahydroquinolines
Patent number
10,323,020
Issue date
Jun 18, 2019
Bayer Pharma Aktiengesellschaft
Eva Maria Becker-Pelster
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use
Patent number
10,052,312
Issue date
Aug 21, 2018
Bayer Pharma Aktiengesellschaft
Alexandros Vakalopoulos
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted piperidinyl tetrahydroquinolines
Patent number
9,944,621
Issue date
Apr 17, 2018
Bayer Pharma Aktiengesellschaft
Eva Maria Becker-Pelster
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Amido-substituted azole compounds
Patent number
9,884,063
Issue date
Feb 6, 2018
Bayer Pharma Aktiengesellschaft
Knut Eis
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
3-aryl-substituted imidazo[1,2-A]pyridines and their use
Patent number
9,776,997
Issue date
Oct 3, 2017
Bayer Pharma Aktiengesellschaft
Alexandros Vakalopoulos
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Cyano-substituted imidazo[1,2-A]pyridinecarboxamides and their use
Patent number
9,771,360
Issue date
Sep 26, 2017
Bayer Pharma Aktiengesellschaft
Alexandros Vakalopoulos
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted piperidinyltetrahydroquinolines
Patent number
9,624,198
Issue date
Apr 18, 2017
Bayer Pharma Aktiengesellschaft
Eva Maria Becker-Pelster
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted bipiperidinyl derivatives
Patent number
9,624,199
Issue date
Apr 18, 2017
Bayer Pharma Aktiengesellschaft
Eva Maria Becker-Pelster
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use
Patent number
9,624,214
Issue date
Apr 18, 2017
Bayer Pharma Aktiengesellschaft
Alexandros Vakalopoulos
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrazolo[1,5-A]-pyridine-3-carboxamides and use thereof
Patent number
9,422,285
Issue date
Aug 23, 2016
Bayer Pharma Aktiengesellschaft
Alexandros Vakalopoulos
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use
Patent number
9,126,998
Issue date
Sep 8, 2015
Bayer Pharma AG
Alexandros Vakalopoulos
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Patents Applications
last 30 patents
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Patent Application
BICYCLIC TRIAZINE DERIVATIVES FOR THE TREATMENT OF CANCER
Publication number
20250066370
Publication date
Feb 27, 2025
DEUTSCHES KREBSFORSCHUNGSZENTRUM
Kai THEDE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRAZOLOPYRAZINES ACTING ON CANCERS VIA INHIBITION OF CDK12
Publication number
20230192700
Publication date
Jun 22, 2023
Bayer Aktiengesellschaft
Markus BERGER
C07 - ORGANIC CHEMISTRY
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Patent Application
PYRAZOLOTRIAZINES
Publication number
20230117034
Publication date
Apr 20, 2023
Bayer Aktiengesellschaft
Kai THEDE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
INHIBITORS OF ADRENORECEPTOR ADRAC2
Publication number
20230115270
Publication date
Apr 13, 2023
Bayer Aktiengesellschaft
Martina DELBECK
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED MACROCYCLIC INDOLE DERIVATIVES
Publication number
20230112244
Publication date
Apr 13, 2023
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMIDAZOTRIAZINES ACTING ON CANCER VIA INHIBITION OF CDK12
Publication number
20230106032
Publication date
Apr 6, 2023
Bayer Aktiengesellschaft
Kai THEDE
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYCLIC FLUORINE SUBSTITUTED INDOLE DERIVATIVES
Publication number
20220281891
Publication date
Sep 8, 2022
THE BROAD INSTITUTE, INC.
Steven J. Ferrara
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYCLIC INDOLE DERIVATIVES
Publication number
20210292341
Publication date
Sep 23, 2021
THE BROAD INSTITUTE, INC.
Laura Furst
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYCLIC CHLORINE SUBSTITUTED INDOLE DERIVATIVES
Publication number
20210277022
Publication date
Sep 9, 2021
Bayer Aktiengesellschaft
Kai Thede
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED MACROCYCLIC INDOLE DERIVATIVES
Publication number
20210269456
Publication date
Sep 2, 2021
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ARYL ANNULATED MACROCYCLIC INDOLE DERIVATIVES
Publication number
20210253598
Publication date
Aug 19, 2021
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC FLUORINE SUBSTITUTED INDOLE DERIVATIVES
Publication number
20210079018
Publication date
Mar 18, 2021
THE BROAD INSTITUTE, INC.
Steven J. Ferrara
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC INDOLE DERIVATIVES
Publication number
20200087322
Publication date
Mar 19, 2020
Sarah Anna Liesa Johannes
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMINO-SUBSTITUTED IMIDAZO[1,2-A] PYRIDINECARBOXAMIDES AND THEIR USE
Publication number
20190248783
Publication date
Aug 15, 2019
BAYER PHARMA AKTIENGESELLSCHAFT
Alexandros VAKALOPOULOS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMINO-SUBSTITUTED IMIDAZO[1,2-A] PYRIDINECARBOXAMIDES AND THEIR USE
Publication number
20180319794
Publication date
Nov 8, 2018
BAYER PHARMA AKTIENGESELLSCHAFT
Alexandros VAKALOPOULOS
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMIDO-SUBSTITUTED CYCLOHEXANE DERIVATIVES
Publication number
20180148418
Publication date
May 31, 2018
BAYER PHARMA AKTIENGESELLSCHAFT
Knut EIS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PIPERIDINYL TETRAHYDROQUINOLINES
Publication number
20180141930
Publication date
May 24, 2018
BAYER PHARMA AKTIENGESELLSCHAFT
Eva Maria BECKER-PELSTER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PIPERIDINYL TETRAHYDROQUINOLINES
Publication number
20180141931
Publication date
May 24, 2018
BAYER PHARMA AKTIENGESELLSCHAFT
Eva Maria BECKER-PELSTER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
CYANO-SUBSTITUTED IMIDAZO[1,2-A]PYRIDINECARBOXAMIDES AND THEIR USE
Publication number
20170217954
Publication date
Aug 3, 2017
BAYER PHARMA AKTIENGESELLSCHAFT
Alexandros VAKALOPOULOS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMINO-SUBSTITUTED IMIDAZO[1,2-A]PYRIDINECARBOXAMIDES AND THEIR USE
Publication number
20170182014
Publication date
Jun 29, 2017
BAYER PHARMA AKTIENGESELLSCHAFT
Alexandros VAKALOPOULOS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMIDO-SUBSTITUTED AZOLE COMPOUNDS
Publication number
20170020886
Publication date
Jan 26, 2017
BAYER PHARMA AKTIENGESELLSCHAFT
Knut EIS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PIPERIDINYL-TETRAHYDROQUINOLINES
Publication number
20160318901
Publication date
Nov 3, 2016
BAYER PHARMA AKTIENGESELLSCHAFT
Eva Maria BECKER-PELSTER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED BIPIPERIDINYL DERIVATIVES
Publication number
20160318866
Publication date
Nov 3, 2016
BAYER PHARMA AKTIENGESELLSCHAFT
Eva Maria BECKER-PELSTER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED BIPIPERIDINYL DERIVATIVES
Publication number
20160304492
Publication date
Oct 20, 2016
BAYER PHARMA AKTIENGESELLSCHAFT
Eva Maria BECKER-PELSTER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PIPERIDINYLTETRAHYDROQUINOLINES
Publication number
20160304491
Publication date
Oct 20, 2016
BAYER PHARMA AKTIENGESELLSCHAFT
Eva Maria BECKER-PELSTER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRAZOLO[1,5-A]-PYRIDINE-3-CARBOXAMIDES AND USE THEREOF
Publication number
20160185775
Publication date
Jun 30, 2016
Bayer Pharma Aktiengesellschaft
Alexandros VAKALOPOULOS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED IMIDAZO[1,2-A]PYRAZINECARBOXAMIDES AND USE THEREOF
Publication number
20160176880
Publication date
Jun 23, 2016
Bayer Pharma Aktiengesellschaft
Alexandros VAKALOPOULOS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3-ARYL-SUBSTITUTED IMIDAZO[1,2-A]PYRIDINES AND THEIR USE
Publication number
20160122341
Publication date
May 5, 2016
Bayer Pharma Aktiengesellschaft
Alexandros VAKALOPOULOS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
AMINO-SUBSTITUTED IMIDAZO[1,2-A]PYRIDINECARBOXAMIDES AND THEIR USE
Publication number
20150274719
Publication date
Oct 1, 2015
BAYER PHARMA AKTIENGESELLSCHAFT
Alexandros VAKALOPOULOS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Amino-substituted imidazo[1,2-a]pyridinecarboxamides and their use
Publication number
20140179672
Publication date
Jun 26, 2014
BAYER PHARMA AKTIENGESELLSCHAFT
Alexandros VAKALOPOULOS
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE