Robert Mazzola

Person

Clinton, NJ, US

People

Patents Grantslast 30 patents

Information Patent Grant
3-(1H-pyrazol-4-yl)pyridine allosteric modulators of the M4 muscari...
- Patent number 11,970,479
- Issue date Apr 30, 2024
- Merck Sharp & Dohme LLC
- John J. Acton
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
3-(1H-pyrazol-4-yl)pyridine allosteric modulators of the M4 muscari...
- Patent number 11,339,156
- Issue date May 24, 2022
- Merck Sharp & Dohme Corp.
- John J. Acton
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Heteroaryl piperidine ether allosteric modulators of the M4 muscari...
- Patent number 11,319,298
- Issue date May 3, 2022
- Merck Sharp & Dohme Corp.
- Jianming Bao
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
6,5-fused heteroaryl piperidine ether allosteric modulators of the...
- Patent number 11,230,556
- Issue date Jan 25, 2022
- Merck Sharp & Dohme Corp.
- Xiaolei Gao
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
3-(1H-pyrazol-4-yl)pyridine allosteric modulators of the M4 muscari...
- Patent number 11,149,036
- Issue date Oct 19, 2021
- MSD R&D (CHINA) CO., LTD
- John J. Acton
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
5-(pyridin-3-yl)oxazole allosteric modulators of the M4 muscarinic...
- Patent number 10,981,902
- Issue date Apr 20, 2021
- Merck Sharp & Dohme Corp.
- Jianming Bao
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Azabicyclo[4.1.0]heptane allosteric modulators of the M4 muscarinic...
- Patent number 10,945,771
- Issue date Mar 16, 2021
- Merck Sharp & Dohme Corp.
- Dane James Clausen
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
3-(1H-pyrazol-4-yl)pyridine allosteric modulators of the M4 muscari...
- Patent number 10,933,056
- Issue date Mar 2, 2021
- Merck Sharp & Dohme Corp.
- John J. Acton
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
6,6-fused heteroaryl piperidine ether allosteric modulators of the...
- Patent number 10,836,775
- Issue date Nov 17, 2020
- Merck Sharp & Dohme Corp.
- Xiaolei Gao
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-5-one allosteric modulators of...
- Patent number 10,351,564
- Issue date Jul 16, 2019
- Merck Sharop & Dohme, Corp.
- Xiaolei Gao
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
6,7-dihydro-5H-pyrrolo[3,4-B]pyridin-5-one allosteric modulators of...
- Patent number 10,329,289
- Issue date Jun 25, 2019
- Merck Sharp & Dohme Corp.
- Jianming Bao
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Quinoxalines and AZA-quinoxalines as CRTH2 receptor modulators
- Patent number 9,469,615
- Issue date Oct 18, 2016
- Merck Sharp & Dohme Corp.
- Christopher W. Boyce
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Quinazolinone-type compounds as CRTH2 antagonists
- Patent number 8,927,559
- Issue date Jan 6, 2015
- Merck Sharp & Dohme Corp.
- Robert G. Aslanian
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Heterocyclic aspartyl protease inhibitors
- Patent number 8,829,036
- Issue date Sep 9, 2014
- Merck Sharp & Dohme Corp.
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Heterocyclic aspartyl protease inhibitors
- Patent number 8,778,980
- Issue date Jul 15, 2014
- Merck Sharp & Dohme Corp.
- Zhaoning Zhu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Substituted isoindolines as aspartyl protease inhibitors
- Patent number 8,722,708
- Issue date May 13, 2014
- Merck Sharp & Dohme Inc.
- Andrew Stamford
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Heterocyclic aspartyl protease inhibitors
- Patent number 8,691,833
- Issue date Apr 8, 2014
- Merck Sharp & Dohme Corp.
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Heterocyclic aspartyl protease inhibitors
- Patent number 8,691,831
- Issue date Apr 8, 2014
- Merck Sharp & Dohme Corp.
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Aspartyl protease inhibitors
- Patent number 8,629,155
- Issue date Jan 14, 2014
- Merck Sharp & Dohme, Corp.
- Yusheng Wu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Gamma secretase modulators
- Patent number 8,518,975
- Issue date Aug 27, 2013
- Merck Sharp + Dohme Corp.
- Robert G. Aslanian
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Gamma secretase modulators
- Patent number 8,357,682
- Issue date Jan 22, 2013
- Zhaoning Zhu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Aspartyl protease inhibitors
- Patent number 8,168,641
- Issue date May 1, 2012
- Schering Corporation
- Yusheng Wu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Heterocyclic aspartyl protease inhibitors
- Patent number 7,763,609
- Issue date Jul 27, 2010
- Schering Corporation
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Heterocyclic aspartyl protease inhibitors
- Patent number 7,700,603
- Issue date Apr 20, 2010
- Schering Corporation
- Zhaoning Zhu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Compounds for the treatment of inflammatory disorders
- Patent number 7,652,020
- Issue date Jan 26, 2010
- Schering Corporation
- Zhuyan Guo
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Compounds for the treatment of inflammatory disorders
- Patent number 7,598,242
- Issue date Oct 6, 2009
- Schering Corporation
- Zhaoning Zhu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Heterocyclic aspartyl protease inhibitors
- Patent number 7,592,348
- Issue date Sep 22, 2009
- Schering Corporation
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Grant
Selective D1/D5 receptor antagonists for the treatment of obesity a...
- Patent number 7,504,391
- Issue date Mar 17, 2009
- Schering Corporation
- Duane A. Burnett
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Compounds for the treatment of inflammatory disorders
- Patent number 7,034,057
- Issue date Apr 25, 2006
- Schering Corporation
- Zhaoning Zhu
- C07 - ORGANIC CHEMISTRY
Information Patent Grant
Compounds for the treatment of inflammatory disorders
- Patent number 6,838,466
- Issue date Jan 4, 2005
- Schering Corporation
- Zhaoning Zhu
- C07 - ORGANIC CHEMISTRY

Patents Applicationslast 30 patents

Information Patent Application
3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARI...
- Publication number 20210395224
- Publication date Dec 23, 2021
- MERCK SHARP & DOHME CORP.
- John J. Acton
- C07 - ORGANIC CHEMISTRY
Information Patent Application
3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARI...
- Publication number 20210380580
- Publication date Dec 9, 2021
- MERCK SHARP & DOHME CORP.
- John J. ACTON
- C07 - ORGANIC CHEMISTRY
Information Patent Application
3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARI...
- Publication number 20200207758
- Publication date Jul 2, 2020
- MERCK SHARP & DOHME CORP.
- John J. ACTON
- C07 - ORGANIC CHEMISTRY
Information Patent Application
5-(PYRIDIN-3-YL)OXAZOLE ALLOSTERIC MODULATORS OF THE M4 MUSCARINIC...
- Publication number 20200109137
- Publication date Apr 9, 2020
- MERCK SHARP & DOHME CORP.
- Jianming BAO
- C07 - ORGANIC CHEMISTRY
Information Patent Application
6,5-FUSED HETEROARYL PIPERIDINE ETHER ALLOSTERIC MODULATORS OF THE...
- Publication number 20200095261
- Publication date Mar 26, 2020
- MERCK SHARP & DOHME CORP.
- Xiaolei GAO
- C07 - ORGANIC CHEMISTRY
Information Patent Application
AZABICYCLO[4.1.0]HEPTANE ALLOSTERIC MODULATORS OF THE M4 MUSCARINI...
- Publication number 20200095262
- Publication date Mar 26, 2020
- MERCK SHARP & DOHME CORP.
- Dane James CLAUSEN
- C07 - ORGANIC CHEMISTRY
Information Patent Application
3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARI...
- Publication number 20200069671
- Publication date Mar 5, 2020
- MERCK SHARP & DOHME CORP.
- John J. Acton
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
HETEROARYL PIPERIDINE ETHER ALLOSTERIC MODULATORS OF THE M4 MUSCARI...
- Publication number 20190315708
- Publication date Oct 17, 2019
- MERCK SHARP & DOHME CORP.
- Jianming BAO
- C07 - ORGANIC CHEMISTRY
Information Patent Application
6,6-FUSED HETEROARYL PIPERIDINE ETHER ALLOSTERIC MODULATORS OF THE...
- Publication number 20190315762
- Publication date Oct 17, 2019
- MERCK SHARP & DOHME CORP.
- Xiaolei GAO
- C07 - ORGANIC CHEMISTRY
Information Patent Application
6,7-DIHYDRO-5H-PYRROLO[3,4-B]PYRIDIN-5-ONE ALLOSTERIC MODULATORS OF...
- Publication number 20190062331
- Publication date Feb 28, 2019
- MERCK SHARP & DOHME CORP.
- JIANMING BAO
- C07 - ORGANIC CHEMISTRY
Information Patent Application
3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARI...
- Publication number 20190000824
- Publication date Jan 3, 2019
- MERCK SHARP & DOHME CORP.
- John J. Acton
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
6,7-DIHYDRO-5H-PYRROLO[3,4-B]PYRIDIN-5-ONE ALLOSTERIC MODULATORS OF...
- Publication number 20170183342
- Publication date Jun 29, 2017
- JIANMING BAO
- C07 - ORGANIC CHEMISTRY
Information Patent Application
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
- Publication number 20150105354
- Publication date Apr 16, 2015
- MERCK SHARP & DOHME CORP.
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
SILYL-CONTAINING HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF...
- Publication number 20150057246
- Publication date Feb 26, 2015
- Michael P. Dwyer
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
SILYL-CONTAINING HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF...
- Publication number 20140378416
- Publication date Dec 25, 2014
- Michael P. Dwyer
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
PREPARATION AND USE OF COMPOUNDS AS PROTEASE INHIBITORS
- Publication number 20140206715
- Publication date Jul 24, 2014
- Pharmacopeia, LLC
- Andrew W. Stamford
- C07 - ORGANIC CHEMISTRY
Information Patent Application
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
- Publication number 20140057910
- Publication date Feb 27, 2014
- Schering Corporation
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
QUINOXALINES AND AZA-QUINOXALINES AS CRTH2 RECEPTOR MODULATORS
- Publication number 20130303517
- Publication date Nov 14, 2013
- Christopher W. Boyce
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
QUINAZOLINONE-TYPE COMPOUNDS AS CRTH2 ANTAGONISTS
- Publication number 20130210805
- Publication date Aug 15, 2013
- Robert G. Aslanian
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
- Publication number 20130018066
- Publication date Jan 17, 2013
- Schering Corporation & Pharmacopeia Drug Discovery Inc.
- Zhaoning Zhu
- C07 - ORGANIC CHEMISTRY
Information Patent Application
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
- Publication number 20120276118
- Publication date Nov 1, 2012
- Pharmacopeia Inc.
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
ASPARTYL PROTEASE INHIBITORS
- Publication number 20120232064
- Publication date Sep 13, 2012
- Schering Corporation
- Yusheng Wu
- C07 - ORGANIC CHEMISTRY
Information Patent Application
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
- Publication number 20110218194
- Publication date Sep 8, 2011
- Schering Corporation & Pharmacopeia Drug Discovery Inc.
- Zhaoning Zhu
- C07 - ORGANIC CHEMISTRY
Information Patent Application
GAMMA SECRETASE MODULATORS
- Publication number 20110082153
- Publication date Apr 7, 2011
- Schering Corporation
- Robert G. Aslanian
- C07 - ORGANIC CHEMISTRY
Information Patent Application
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
- Publication number 20100292203
- Publication date Nov 18, 2010
- Schering Corporation
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS
- Publication number 20100145048
- Publication date Jun 10, 2010
- Schering Corporation
- Zhuyan Guo
- C07 - ORGANIC CHEMISTRY
Information Patent Application
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
- Publication number 20090306047
- Publication date Dec 10, 2009
- Schering Corporation
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS
- Publication number 20090258868
- Publication date Oct 15, 2009
- Schering Corporation
- Zhaoning Zhu
- C07 - ORGANIC CHEMISTRY
Information Patent Application
Heterocyclic aspartyl protease inhibitors
- Publication number 20080200445
- Publication date Aug 21, 2008
- Schering Corporation and Pharmacopeia Drug Discovery, Inc.
- Zhaoning Zhu
- A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information Patent Application
Preparation and use of compounds as protease inhibitors
- Publication number 20080176868
- Publication date Jul 24, 2008
- Schering Corporation
- Andrew Stamford
- C07 - ORGANIC CHEMISTRY

Robert Mazzola

Person

Patents Grantslast 30 patents

3-(1H-pyrazol-4-yl)pyridine allosteric modulators of the M4 muscari...

3-(1H-pyrazol-4-yl)pyridine allosteric modulators of the M4 muscari...

Heteroaryl piperidine ether allosteric modulators of the M4 muscari...

6,5-fused heteroaryl piperidine ether allosteric modulators of the...

3-(1H-pyrazol-4-yl)pyridine allosteric modulators of the M4 muscari...

5-(pyridin-3-yl)oxazole allosteric modulators of the M4 muscarinic...

Azabicyclo[4.1.0]heptane allosteric modulators of the M4 muscarinic...

3-(1H-pyrazol-4-yl)pyridine allosteric modulators of the M4 muscari...

6,6-fused heteroaryl piperidine ether allosteric modulators of the...

6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-5-one allosteric modulators of...

6,7-dihydro-5H-pyrrolo[3,4-B]pyridin-5-one allosteric modulators of...

Quinoxalines and AZA-quinoxalines as CRTH2 receptor modulators

Quinazolinone-type compounds as CRTH2 antagonists

Heterocyclic aspartyl protease inhibitors

Heterocyclic aspartyl protease inhibitors

Substituted isoindolines as aspartyl protease inhibitors

Heterocyclic aspartyl protease inhibitors

Heterocyclic aspartyl protease inhibitors

Aspartyl protease inhibitors

Gamma secretase modulators

Gamma secretase modulators

Aspartyl protease inhibitors

Heterocyclic aspartyl protease inhibitors

Heterocyclic aspartyl protease inhibitors

Compounds for the treatment of inflammatory disorders

Compounds for the treatment of inflammatory disorders

Heterocyclic aspartyl protease inhibitors

Selective D1/D5 receptor antagonists for the treatment of obesity a...

Compounds for the treatment of inflammatory disorders

Compounds for the treatment of inflammatory disorders

Patents Applicationslast 30 patents

3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARI...

3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARI...

3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARI...

5-(PYRIDIN-3-YL)OXAZOLE ALLOSTERIC MODULATORS OF THE M4 MUSCARINIC...

6,5-FUSED HETEROARYL PIPERIDINE ETHER ALLOSTERIC MODULATORS OF THE...

AZABICYCLO[4.1.0]HEPTANE ALLOSTERIC MODULATORS OF THE M4 MUSCARINI...

3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARI...

HETEROARYL PIPERIDINE ETHER ALLOSTERIC MODULATORS OF THE M4 MUSCARI...

6,6-FUSED HETEROARYL PIPERIDINE ETHER ALLOSTERIC MODULATORS OF THE...

6,7-DIHYDRO-5H-PYRROLO[3,4-B]PYRIDIN-5-ONE ALLOSTERIC MODULATORS OF...

3-(1H-PYRAZOL-4-YL)PYRIDINE ALLOSTERIC MODULATORS OF THE M4 MUSCARI...

6,7-DIHYDRO-5H-PYRROLO[3,4-B]PYRIDIN-5-ONE ALLOSTERIC MODULATORS OF...

HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS

SILYL-CONTAINING HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF...

SILYL-CONTAINING HETEROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF...

PREPARATION AND USE OF COMPOUNDS AS PROTEASE INHIBITORS

HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS

QUINOXALINES AND AZA-QUINOXALINES AS CRTH2 RECEPTOR MODULATORS

QUINAZOLINONE-TYPE COMPOUNDS AS CRTH2 ANTAGONISTS

HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS

HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS

ASPARTYL PROTEASE INHIBITORS

HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS

GAMMA SECRETASE MODULATORS

HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS

COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS

HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS

HETEROCYCLIC ASPARTYL PROTEASE INHIBITORS

Heterocyclic aspartyl protease inhibitors

Preparation and use of compounds as protease inhibitors