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Ulrich Klar
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Berlin, DE
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last 30 patents
Information
Patent Grant
Substituted macrocyclic indole derivatives
Patent number
11,891,404
Issue date
Feb 6, 2024
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocyclic indole derivatives
Patent number
11,492,358
Issue date
Nov 8, 2022
The Broad Institute, Inc.
Sarah Anna Liesa Johannes
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Macrocyclic chlorine substituted indole derivatives
Patent number
11,478,451
Issue date
Oct 25, 2022
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocyclic chlorine substituted indole derivatives
Patent number
11,447,504
Issue date
Sep 20, 2022
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted macrocyclic indole derivatives
Patent number
11,440,923
Issue date
Sep 13, 2022
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocyclic indole derivatives
Patent number
11,401,278
Issue date
Aug 2, 2022
The Broad Institute, Inc.
Laura Furst
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4H-pyrrolo[3,2-c]pyridin-4-one derivatives
Patent number
11,339,157
Issue date
May 24, 2022
Bayer Aktiengesellschaft
Stephan Siegel
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted dihydroimidazopyridinediones as MKNK1 and MKNK2 inhibitors
Patent number
11,311,520
Issue date
Apr 26, 2022
Bayer Pharma Aktiengesellschaft
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocyclic fluorine substituted indole derivatives
Patent number
11,286,263
Issue date
Mar 29, 2022
The Broad Institute, Inc.
Steven James Ferrara
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Macrocyclic indole derivatives
Patent number
10,981,932
Issue date
Apr 20, 2021
Bayer Aktiengesellschaft
Sarah Anna Liesa Johannes
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazolopyridinamines as MKNK1 and MKNK2 inhibitors
Patent number
10,487,092
Issue date
Nov 26, 2019
Bayer Pharma Aktiengesellschaft
Anja Giese
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
4H-pyrrolo[3,2-C]pyridin-4-one derivatives
Patent number
10,428,063
Issue date
Oct 1, 2019
Bayer Pharma Aktiengesellschaft
Keith Graham
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
3-amino-1,5,6,7-tetrahydro-4H-indol-4-ones
Patent number
10,428,044
Issue date
Oct 1, 2019
Bayer Pharma Aktiengesellschaft
Keith Graham
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
1H-pyrrol-3-amines
Patent number
10,308,629
Issue date
Jun 4, 2019
Bayer Pharma Aktiengesellschaft
Keith Graham
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
3-amino-1,5,6,7-tetrahydro-4H-indol-4-ones
Patent number
10,227,299
Issue date
Mar 12, 2019
Bayer Pharma Aktiengesellschaft
Keith Graham
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
17-hydroxy-17-pentafluoroethyl-estra-4,9(10)-dien-11-aryl derivativ...
Patent number
10,155,004
Issue date
Dec 18, 2018
Bayer Intellectual Property GmbH
Wolfgang Schwede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
17-hydroxy-17-pentafluoroethyl-estra-4,9(10)-dien-11-aryl derivativ...
Patent number
9,717,739
Issue date
Aug 1, 2017
Bayer Intellectual Property GmbH
Wolfgang Schwede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted thiazolopyrimidines
Patent number
9,675,612
Issue date
Jun 13, 2017
Bayer Pharma Aktiengesellschaft
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrazolopyrimidinylamino-indazoles
Patent number
9,556,181
Issue date
Jan 31, 2017
Bayer Pharma Aktiengesellschaft
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Thienopyrimidines
Patent number
9,540,392
Issue date
Jan 10, 2017
Bayer Pharma Aktiengesellschaft
Georg Kettschau
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted imidazopyridazines
Patent number
9,512,130
Issue date
Dec 6, 2016
Bayer Pharma Aktiengesellschaft
Marcus Koppitz
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted imidazopyridazines
Patent number
9,512,126
Issue date
Dec 6, 2016
Bayer Intellectual Property GmbH
Marcus Koppitz
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Imidazopyrazines
Patent number
9,468,642
Issue date
Oct 18, 2016
Bayer Intellectual Property GmbH
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted benzimidazoles
Patent number
9,388,140
Issue date
Jul 12, 2016
Bayer Intellectual Property GmbH
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted pyrrolopyrimidinylamino-benzothiazolones as MKNK kinase...
Patent number
9,382,255
Issue date
Jul 5, 2016
Bayer Pharma Aktiengesellschaft
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted benzothienopyrimidines
Patent number
9,296,757
Issue date
Mar 29, 2016
Bayer Pharma Aktiengesellschaft
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Substituted imidazo[1,2-a]pyrazines as MPS-1 inhibitors
Patent number
9,284,317
Issue date
Mar 15, 2016
Bayer Intellectual Property GmbH
Marcus Koppitz
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Substituted imidazopyridazines
Patent number
9,255,100
Issue date
Feb 9, 2016
Bayer Intellectual Property GmbH
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
6-thio-substituted imidazo[1,2-a]pyrazines as Mps-1 inhibitors
Patent number
9,212,184
Issue date
Dec 15, 2015
Bayer Intellectual Property GmbH
Marcus Koppitz
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
17-hydroxy-17-pentafluorethyl-estra-4,9(10)-dien-11-aryl derivative...
Patent number
9,206,219
Issue date
Dec 8, 2015
Bayer Intellectual Property GmbH
Ulrich Klar
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
N-[2-({4-[3-(ANILINO)-4-OXO-4,5,6,7-TETRAHYDRO-1H-PYRROLO[3,2-C]PYR...
Publication number
20230416249
Publication date
Dec 28, 2023
Bayer Aktiengesellschaft
Stephan SIEGEL
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED MACROCYCLIC INDOLE DERIVATIVES
Publication number
20230112244
Publication date
Apr 13, 2023
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC FLUORINE SUBSTITUTED INDOLE DERIVATIVES
Publication number
20220281891
Publication date
Sep 8, 2022
THE BROAD INSTITUTE, INC.
Steven J. Ferrara
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYCLIC INDOLE DERIVATIVES
Publication number
20210292341
Publication date
Sep 23, 2021
THE BROAD INSTITUTE, INC.
Laura Furst
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYCLIC CHLORINE SUBSTITUTED INDOLE DERIVATIVES
Publication number
20210277022
Publication date
Sep 9, 2021
Bayer Aktiengesellschaft
Kai Thede
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED MACROCYCLIC INDOLE DERIVATIVES
Publication number
20210269456
Publication date
Sep 2, 2021
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
ARYL ANNULATED MACROCYCLIC INDOLE DERIVATIVES
Publication number
20210253598
Publication date
Aug 19, 2021
Bayer Aktiengesellschaft
Kai Thede
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED DIHYDROIMIDAZOPYRIDINEDIONES AS MKNK1 AND MKNK2 INHIBITORS
Publication number
20210085656
Publication date
Mar 25, 2021
BAYER PHARMA AKTIENGESELLSCHAFT
Ulrich KLAR
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYCLIC FLUORINE SUBSTITUTED INDOLE DERIVATIVES
Publication number
20210079018
Publication date
Mar 18, 2021
THE BROAD INSTITUTE, INC.
Steven J. Ferrara
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETERO-1,5,6,7-TETRAHYDRO-4H-INDOL-4-ONES
Publication number
20200216439
Publication date
Jul 9, 2020
BAYER PHARMA AKTIENGESELLSCHAFT
Keith GRAHAM
C07 - ORGANIC CHEMISTRY
Information
Patent Application
MACROCYCLIC INDOLE DERIVATIVES
Publication number
20200087322
Publication date
Mar 19, 2020
Sarah Anna Liesa Johannes
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED IMIDAZOPYRIDINPYRIMIDINES
Publication number
20190388425
Publication date
Dec 26, 2019
BAYER PHARMA AKTIENGESELLSCHAFT
Ulrich KLAR
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED DIHYDROIMIDAZOPYRIDINEDIONES AS MKNK1 AND MKNK2 INHIBITORS
Publication number
20190350910
Publication date
Nov 21, 2019
BAYER PHARMA AKTIENGESELLSCHAFT
Ulrich KLAR
C07 - ORGANIC CHEMISTRY
Information
Patent Application
1H-PYRROL-3-AMINES
Publication number
20180222881
Publication date
Aug 9, 2018
BAYER PHARMA AKTIENGESELLSCHAFT
Keith GRAHAM
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PYRAZOLOPYRIDINAMINES AS MKNK1 AND MKNK2 INHIBITORS
Publication number
20180162877
Publication date
Jun 14, 2018
BAYER PHARMA AKTIENGESELLSCHAFT
Anja GIESE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3-AMINO-1,5,6,7-TETRAHYDRO-4H-INDOL-4-ONES
Publication number
20180155285
Publication date
Jun 7, 2018
BAYER PHARMA AKTIENGESELLSCHAFT
Keith GRAHAM
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
4H-PYRROLO[3,2-C]PYRIDIN-4-ONE DERIVATIVES
Publication number
20180016272
Publication date
Jan 18, 2018
BAYER PHARMA AKTIENGESELLSCHAFT
Keith GRAHAM
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
17-HYDROXY-17-PENTAFLUOROETHYL-ESTRA-4,9(10)-DIEN-11-ARYL DERIVATIV...
Publication number
20170202857
Publication date
Jul 20, 2017
Bayer Intellectual Property GmbH
Wolfgang SCHWEDE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZOTHIADIAZOLAMINES
Publication number
20170197979
Publication date
Jul 13, 2017
BAYER PHARMA AKTIENGESELLSCHAFT
Anja GIESE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED TETRAHYDROPYRIDOTHIENOPYRIMIDINES
Publication number
20170107229
Publication date
Apr 20, 2017
Bayer Pharma Aktiengesellschaft
Ulrich KLAR
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
3-AMINO-1,5,6,7-TETRAHYDRO-4H-INDOL-4-ONES
Publication number
20170101391
Publication date
Apr 13, 2017
BAYER PHARMA AKTIENGESELLSCHAFT
Keith GRAHAM
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
THIENOPYRIMIDINES AS MKNK1 AND MKNK2 INHIBITORS
Publication number
20160297833
Publication date
Oct 13, 2016
BAYER PHARMA AKTIENGESELLSCHAFT
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED THIENOPYRIMIDINES AND PHARMACEUTICAL USE THEREOF
Publication number
20160159816
Publication date
Jun 9, 2016
BAYER PHARMA AKTIENGESELLSCHAFT
Georg KETTSCHAU
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRAZOLOPYRIDINES
Publication number
20160159789
Publication date
Jun 9, 2016
BAYER PHARMA AKTIENGESELLSCHAFT
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED IMIDAZOPYRIDAZINES
Publication number
20160016959
Publication date
Jan 21, 2016
BAYER PHARMA AKTIENGESELLSCHAFT
Marcus Koppitz
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED THIAZOLOPYRIMIDINES
Publication number
20160009734
Publication date
Jan 14, 2016
BAYER PHARMA AKTIENGESELLSCHAFT
Ulrich KLAR
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRAZOLOPYRIMIDINYLAMINO-INDAZOLES
Publication number
20160002245
Publication date
Jan 7, 2016
BAYER PHARMA AKTIENGESELLSCHAFT
Ulrich KLAR
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
17-HYDROXY-17-PENTAFLUOROETHYL-ESTRA-4,9(10)-DIEN-11-ARYL DERIVATIV...
Publication number
20150342962
Publication date
Dec 3, 2015
Bayer Intellectual Property GmbH
Wolfgang SCHWEDE
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED INDAZOL-PYRROLOPYRIMIDINES USEFUL IN THE TREATMENT OF H...
Publication number
20150252047
Publication date
Sep 10, 2015
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
SUBSTITUTED PYRROLOPYRIMIDINYLAMINO-BENZOTHIAZOLONES AS MKNK KINASE...
Publication number
20150239891
Publication date
Aug 27, 2015
BAYER PHARMA AKTIENGESELLSCHAFT
Ulrich Klar
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE