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Patents Grants
last 30 patents
Information
Patent Grant
6-fused heteroaryldihydropyrimidines for the treatment and prophyla...
Patent number
12,351,575
Issue date
Jul 8, 2025
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Tricyclic compounds for the treatment of cancer
Patent number
12,247,036
Issue date
Mar 11, 2025
HOFFMANN-LA ROCHE INC.
Jianguo Chen
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Aminocarbamoyl compounds for the treatment of viral infections
Patent number
12,060,333
Issue date
Aug 13, 2024
HOFFMANN-LA ROCHE INC.
Chungen Liang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Heteroaryl heterocyclyl compounds for the treatment of autoimmune d...
Patent number
11,713,327
Issue date
Aug 1, 2023
HOFFMANN-LA ROCHE INC.
Fabian Dey
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dihydropyrimidinyl benzazepine carboxamide compounds
Patent number
11,046,671
Issue date
Jun 29, 2021
HOFFMANN-LA ROCHE INC.
Fabian Dey
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dihydropyrimidinyl benzazepine carboxamide compounds
Patent number
10,590,112
Issue date
Mar 17, 2020
HOFFMANN-LA ROCHE INC.
Fabian Dey
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzazepine dicarboxamide compounds with secondary amide function
Patent number
10,544,102
Issue date
Jan 28, 2020
HOFFMANN-LA ROCHE INC.
Lisha Wang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Sulfinylphenyl or sulfonimidoylphenyl benzazepines
Patent number
10,428,027
Issue date
Oct 1, 2019
HOFFMANN-LA ROCHE INC.
Sabine Hoves
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-fused heteroaryldihydropyrimidines for the treatment and prophyla...
Patent number
10,428,069
Issue date
Oct 1, 2019
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzazepine dicarboxamide compounds with tertiary amide function
Patent number
10,370,338
Issue date
Aug 6, 2019
HOFFMANN-LA ROCHE INC.
Lisha Wang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Aza-oxo-indoles for the treatment and prophylaxis of respiratory sy...
Patent number
10,189,838
Issue date
Jan 29, 2019
Hoffman-La Roche Inc.
Lisha Wang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-fused heteroaryldihydropyrimidines for the treatment and prophyla...
Patent number
10,081,627
Issue date
Sep 25, 2018
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzazepine sulfonamide compounds
Patent number
9,890,124
Issue date
Feb 13, 2018
HOFFMANN-LA ROCHE INC.
Sabine Hoves
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aza-oxo-indoles for the treatment and prophylaxis of respiratory sy...
Patent number
9,890,155
Issue date
Feb 13, 2018
HOFFMANN-LA ROCHE INC.
Lisha Wang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
4-methyl-dihydropyrimidines for the treatment and prophylaxis of He...
Patent number
9,856,247
Issue date
Jan 2, 2018
HOFFMANN-LA ROCHE INC.
Lei Guo
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzazepine dicarboxamide compounds
Patent number
9,822,065
Issue date
Nov 21, 2017
HOFFMANN-LA ROCHE INC.
Sabine Hoves
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Aza-oxo-indoles for the treatment and prophylaxis of respiratory sy...
Patent number
9,670,211
Issue date
Jun 6, 2017
Hoffmann-La Roche Inc.
Lu Gao
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Benzazepine dicarboxamide compounds
Patent number
9,597,333
Issue date
Mar 21, 2017
HOFFMANN-LA ROCHE INC.
Sabine Hoves
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Benzazepine dicarboxamide compounds
Patent number
9,475,775
Issue date
Oct 25, 2016
HOFFMANN-LA ROCHE INC.
Sabine Hoves
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6-amino acid heteroaryldihydropyrimidines for the treatment and pro...
Patent number
9,447,086
Issue date
Sep 20, 2016
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
6-fused heteroaryldihydropyrimidines for the treatment and prophyla...
Patent number
9,233,978
Issue date
Jan 12, 2016
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
N-hydroxy-benzamids for the treatment of cancer
Patent number
8,716,285
Issue date
May 6, 2014
Hoffmann-La Roche Inc.
Lei Guo
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
HALOINDOLE MACROCYCLIC COMPOUNDS FOR THE TREATMENT OF CANCER
Publication number
20250206761
Publication date
Jun 26, 2025
HOFFMANN-LA ROCHE INC.
Jianguo CHEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
MACROCYCLIC COMPOUNDS FOR THE TREATMENT OF CANCER
Publication number
20250163072
Publication date
May 22, 2025
HOFFMANN-LA ROCHE INC.
Jianguo CHEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TRICYCLIC COMPOUNDS FOR THE TREATMENT OF CANCER
Publication number
20240417410
Publication date
Dec 19, 2024
HOFFMANN-LA ROCHE INC.
Jianguo CHEN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
IMIDAZO[1,2-A]PYRIDINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DI...
Publication number
20230279001
Publication date
Sep 7, 2023
HOFFMANN-LA ROCHE INC.
Dongdong CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HYDROPYRIDO[1,2-a]PYRAZINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUN...
Publication number
20230022297
Publication date
Jan 26, 2023
HOFFMANN-LA ROCHE INC.
Jianguo CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SPIRO(ISOBENZOFURANAZETIDINE) COMPOUNDS FOR THE TREATMENT OF AUTOIM...
Publication number
20230002415
Publication date
Jan 5, 2023
HOFFMANN-LA ROCHE INC.
Jianguo CHEN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
QUINOLINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE
Publication number
20220363665
Publication date
Nov 17, 2022
HOFFMANN-LA ROCHE INC.
Fabian DEY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
AMINOCARBAMOYL COMPOUNDS FOR THE TREATMENT OF VIRAL INFECTIONS
Publication number
20220064128
Publication date
Mar 3, 2022
HOFFMANN-LA ROCHE INC.
Chungen Liang
C07 - ORGANIC CHEMISTRY
Information
Patent Application
HETEROCYCLYL COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE
Publication number
20210395239
Publication date
Dec 23, 2021
HOFFMANN-LA ROCHE INC.
Fabian DEY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLIDINYL AMIDE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE
Publication number
20210323977
Publication date
Oct 21, 2021
HOFFMANN-LA ROCHE INC.
Haixia Liu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
ARYL COMPOUNDS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL INFEC...
Publication number
20210309658
Publication date
Oct 7, 2021
HOFFMANN-LA ROCHE INC.
Fabian DEY
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
TRICYCLIC COMPOUNDS FOR THE TREATMENT AND PROPHYLAXIS OF BACTERIAL...
Publication number
20210309657
Publication date
Oct 7, 2021
HOFFMANN-LA ROCHE INC.
Fabian DEY
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL HETEROARYL HETEROCYCLYL COMPOUNDS FOR THE TREATMENT OF AUTOIM...
Publication number
20210300947
Publication date
Sep 30, 2021
HOFFMANN-LA ROCHE INC.
FABIAN DEY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLIDINE AMINE COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE
Publication number
20210253575
Publication date
Aug 19, 2021
HOFFMANN-LA ROCHE INC.
Fabian Dey
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DIHYDROPYRIMIDINYL BENZAZEPINE CARBOXAMIDE COMPOUNDS
Publication number
20200172513
Publication date
Jun 4, 2020
HOFFMANN-LA ROCHE INC.
Fabian Dey
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
6-fused heteroaryldihydropyrimidines for the treatment and prophyla...
Publication number
20200062753
Publication date
Feb 27, 2020
HOFFMANN-LA ROCHE INC.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
DIHYDROPYRIMIDINYL BENZAZEPINE CARBOXAMIDE COMPOUNDS
Publication number
20190135788
Publication date
May 9, 2019
HOFFMANN-LA ROCHE INC.
Fabian Dey
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZAZEPINE DICARBOXAMIDE COMPOUNDS WITH TERTIARY AMIDE FUNCTION
Publication number
20190077763
Publication date
Mar 14, 2019
HOFFMANN-LA ROCHE INC.
Lisha Wang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
BENZAZEPINE DICARBOXAMIDE COMPOUNDS WITH SECONDARY AMIDE FUNCTION
Publication number
20190077764
Publication date
Mar 14, 2019
HOFFMANN-LA ROCHE INC.
Lisha Wang
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Novel 6-fused heteroaryldihydropyrimidines for the treatment and pr...
Publication number
20180370969
Publication date
Dec 27, 2018
HOFFMANN-LA ROCHE INC.
Lei Guo
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Sulfinylphenyl or Sulfonimidoylphenyl Benzazepines
Publication number
20180194735
Publication date
Jul 12, 2018
HOFFMANN-LA ROCHE INC.
Sabine Hoves
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL AZA-OXO-INDOLES FOR THE TREATMENT AND PROPHYLAXIS OF RESPIRAT...
Publication number
20180072726
Publication date
Mar 15, 2018
HOFFMANN-LA ROCHE INC.
Lisha WANG
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL AZA-OXO-INDOLES FOR THE TREATMENT AND PROPHYLAXIS OF RESPIRAT...
Publication number
20180072725
Publication date
Mar 15, 2018
HOFFMANN-LA ROCHE INC.
Lisha Wang
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL 4-METHYL-DIHYDROPYRIMIDINES FOR THE TREATMENT AND PROPHYLAXIS...
Publication number
20170334898
Publication date
Nov 23, 2017
HOFFMANN-LA ROCHE INC.
Lei Guo
C07 - ORGANIC CHEMISTRY
Information
Patent Application
BENZAZEPINE SULFONAMIDE COMPOUNDS
Publication number
20170275253
Publication date
Sep 28, 2017
HOFFMANN-LA ROCHE INC.
Sabine Hoves
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Benzazepine Dicarboxamide Compounds
Publication number
20170014423
Publication date
Jan 19, 2017
HOFFMANN-LA ROCHE INC.
Sabine Hoves
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
Benzazepine Dicarboxamide Compounds
Publication number
20160257653
Publication date
Sep 8, 2016
HOFFMANN-LA ROCHE INC.
Sabine Hoves
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL 6-AMINO ACID HETEROARYLDIHYDROPYRIMIDINES FOR THE TREATMENT A...
Publication number
20160237078
Publication date
Aug 18, 2016
Hoffmann-La Roche Inc.
Lei Guo
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL AZA-OXO-INDOLES FOR THE TREATMENT AND PROPHYLAXIS OF RESPIRAT...
Publication number
20160229853
Publication date
Aug 11, 2016
HOFFMANN-LA ROCHE INC.
Lu GAO
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL AZA-OXO-INDOLES FOR THE TREATMENT AND PROPHYLAXIS OF RESPIRAT...
Publication number
20160159794
Publication date
Jun 9, 2016
HOFFMANN-LA ROCHE INC.
Lisha Wang
C07 - ORGANIC CHEMISTRY