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Patents Grants
last 30 patents
Information
Patent Grant
Heterocyclic compounds
Patent number
11,858,912
Issue date
Jan 2, 2024
HOFFMANN-LA ROCHE INC.
Mathis Braendlin
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Dihydropyrimidinylthiazole for the treatment and prophylaxis of hep...
Patent number
11,447,489
Issue date
Sep 20, 2022
HOFFMANN-LA ROCHE INC.
Xingchun Han
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Dihydropyrrolopyrimidines for the treatment and prophylaxis of hepa...
Patent number
11,225,482
Issue date
Jan 18, 2022
HOFFMANN-LA ROCHE INC.
Zhanling Cheng
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
PAPD5 and PAPD7 inhibitors for treating a hepatitis B infection
Patent number
11,191,775
Issue date
Dec 7, 2021
HOFFMANN-LA ROCHE INC.
Xingchun Han
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Methods of synthesizing pyrazine compounds
Patent number
11,168,086
Issue date
Nov 9, 2021
HOFFMANN-LA ROCHE INC.
Taishan Hu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tetrahydropyridopyrimidines for the treatment of HBV infection
Patent number
11,104,674
Issue date
Aug 31, 2021
HOFFMANN-LA ROCHE INC.
Zhanling Cheng
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Tetrahydropyridopyrimidines for the treatment and prophylaxis of he...
Patent number
10,968,218
Issue date
Apr 6, 2021
HOFFMANN-LA ROCHE INC.
Zhanling Cheng
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Tetrahydropyrazolopyridine compounds for the treatment of infectiou...
Patent number
10,781,206
Issue date
Sep 22, 2020
HOFFMANN-LA ROCHE INC.
Taishan Hu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Pyrazolopyrazine and triazolopyrazine compounds for the treatment o...
Patent number
10,683,299
Issue date
Jun 16, 2020
HOFFMANN-LA ROCHE INC.
Xingchun Han
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Tricyclic 4-pyridone-3-carboxylic acid derivatives for the treatmen...
Patent number
10,336,751
Issue date
Jul 2, 2019
HOFFMANN-LA ROCHE INC.
Zhanling Cheng
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6,7-dihydropyrido[2,1-A]phthalazin-2-ones for the treatment and pro...
Patent number
10,150,740
Issue date
Dec 11, 2018
HOFFMANN-LA ROCHE INC.
Zhanling Cheng
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
2-oxo-6,7-dihydrobenzo[a]quinolizine-3-carboxylic acid derivatives...
Patent number
10,093,671
Issue date
Oct 9, 2018
HOFFMANN-LA ROCHE INC.
Xingchun Han
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tetracyclic 4-oxo-pyridine-3-carboxylic acid derivatives for the tr...
Patent number
10,053,461
Issue date
Aug 21, 2018
HOFFMANN-LA ROCHE INC.
Xingchun Han
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Dihydroquinolizinones for the treatment and prophylaxis of hepatiti...
Patent number
9,949,966
Issue date
Apr 24, 2018
Hoffman-La Roche Inc.
Xingchun Han
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Grant
Dihydroquinolizinones for the treatment and prophylaxis of hepatiti...
Patent number
9,920,049
Issue date
Mar 20, 2018
Hoffman-La Roche Inc.
Song Yang
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Pyrazine compounds for the treatment of infectious diseases
Patent number
9,890,167
Issue date
Feb 13, 2018
HOFFMANN-LA ROCHE INC.
Taishan Hu
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Tetrahydropyridopyrimidines and tetrahydropyridopyridines for the t...
Patent number
9,845,322
Issue date
Dec 19, 2017
HOFFMANN-LA ROCHE INC.
Zhanling Cheng
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
6,7-dihydrobenzo[a]quinolizin-2-one derivatives for the treatment a...
Patent number
9,637,485
Issue date
May 2, 2017
HOFFMANN-LA ROCHE INC.
Xingchun Han
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Dihydroquinolizinones for the treatment and prophylaxis of hepatiti...
Patent number
9,458,153
Issue date
Oct 4, 2016
HOFFMANN-LA ROCHE INC.
Xingchun Han
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
3,3′-spiroindolinone derivatives
Patent number
8,076,482
Issue date
Dec 13, 2011
Hoffmann-La Roche Inc.
Li Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Spiroindolinone pyridine derivatives
Patent number
7,928,233
Issue date
Apr 19, 2011
Hoffmann-La Roche Inc.
Li Chen
C07 - ORGANIC CHEMISTRY
Information
Patent Grant
Spiroindolinone derivatives
Patent number
7,776,875
Issue date
Aug 17, 2010
Hoffman-La Roche Inc.
Li Chen
C07 - ORGANIC CHEMISTRY
Patents Applications
last 30 patents
Information
Patent Application
QUATERNARY AMMONIUM CATION SUBSTITUTED COMPOUNDS FOR THE TREATMENT...
Publication number
20240376073
Publication date
Nov 14, 2024
HOFFMANN-LA ROCHE INC.
Sandra Marie Joseph GRALL-ULSEMER
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
HETEROCYCLIC COMPOUNDS
Publication number
20240368117
Publication date
Nov 7, 2024
HOFFMANN-LA ROCHE INC.
Mathis BRAENDLIN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
OXOINDOLINE COMPOUND FOR THE TREATMENT OF INFLAMMATORY DISEASES OR...
Publication number
20240140933
Publication date
May 2, 2024
HOFFMANN-LA ROCHE INC.
Fabian DEY
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PYRROLO[2,3-B]PYRAZINE COMPOUNDS AS CCCDNA INHIBITORS FOR THE TREAT...
Publication number
20230248723
Publication date
Aug 10, 2023
HOFFMANN-LA ROCHE INC.
Jitao David ZHANG
G01 - MEASURING TESTING
Information
Patent Application
NOVEL IMIDAZOPYRAZINE DERIVATIVES
Publication number
20230141403
Publication date
May 11, 2023
HOFFMANN-LA ROCHE INC.
Zhanling CHENG
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL HETEROCYCLIC COMPOUNDS
Publication number
20230133845
Publication date
May 4, 2023
HOFFMANN-LA ROCHE INC.
Mathis BRAENDLIN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL IMIDAZOPYRAZINE DERIVATIVES
Publication number
20230012368
Publication date
Jan 12, 2023
HOFFMANN-LA ROCHE INC.
Jean-Baptiste BLANC
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL HETEROCYCLIC COMPOUNDS
Publication number
20220396565
Publication date
Dec 15, 2022
HOFFMANN-LA ROCHE INC.
Zhanling CHENG
C07 - ORGANIC CHEMISTRY
Information
Patent Application
SUBSTITUTED PYRIMIDINE FOR THE TREATMENT AND PROPHYLAXIS OF HEPATIT...
Publication number
20220396567
Publication date
Dec 15, 2022
HOFFMANN-LA ROCHE INC.
Song FENG
C07 - ORGANIC CHEMISTRY
Information
Patent Application
PAPD5 AND PAPD7 INHIBITORS FOR TREATING A HEPATITIS B INFECTION
Publication number
20220096527
Publication date
Mar 31, 2022
HOFFMANN-LA ROCHE INC.
Xingchun HAN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
DIHYDROPYRIMIDINYLTHIAZOLE FOR THE TREATMENT AND PROPHYLAXIS OF HEP...
Publication number
20210061801
Publication date
Mar 4, 2021
HOFFMANN-LA ROCHE INC.
Xingchun HAN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL TETRAHYDROPYRIDOPYRIMIDINES FOR THE TREATMENT AND PROPHYLAXIS...
Publication number
20200062748
Publication date
Feb 27, 2020
HOFFMANN-LA ROCHE INC.
Zhanling CHENG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL PYRAZOLOPYRAZINE AND TRIAZOLOPYRAZINE COMPOUNDS FOR THE TREAT...
Publication number
20190248792
Publication date
Aug 15, 2019
HOFFMANN-LA ROCHE INC.
Xingchun Han
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL TETRAHYDROPYRAZOLOPYRIDINE COMPOUNDS FOR THE TREATMENT OF INF...
Publication number
20190248786
Publication date
Aug 15, 2019
HOFFMANN-LA ROCHE INC.
Taishan Hu
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL TETRAHYDROPYRIDOPYRIMIDINES FOR THE TREATMENT AND PROPHYLAXIS...
Publication number
20190241559
Publication date
Aug 8, 2019
HOFFMANN-LA ROCHE INC.
Zhanling Cheng
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL DIHYDROPYRROLOPYRIMIDINES FOR THE TREATMENT AND PROPHYLAXIS O...
Publication number
20190241570
Publication date
Aug 8, 2019
HOFFMANN-LA ROCHE INC.
Zhanling Cheng
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
PAPD5 AND PAPD7 INHIBITORS FOR TREATING A HEPATITIS B INFECTION
Publication number
20190194768
Publication date
Jun 27, 2019
HOFFMANN-LA ROCHE INC.
Xingchun HAN
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL PYRAZINE COMPOUNDS FOR THE TREATMENT OF INFECTIOUS DISEASES
Publication number
20180334461
Publication date
Nov 22, 2018
HOFFMANN-LA ROCHE INC.
Taishan Hu
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL TRICYCLIC 4-PYRIDONE-3-CARBOXYLIC ACID DERIVATIVES FOR THE TR...
Publication number
20180134705
Publication date
May 17, 2018
HOFFMANN-LA ROCHE INC.
Zhanling CHENG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL TETRACYCLIC 4-OXO-PYRIDINE-3-CARBOXYLIC ACID DERIVATIVES FOR...
Publication number
20180127416
Publication date
May 10, 2018
HOFFMANN-LA ROCHE INC.
Xingchun HAN
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL 6,7-DIHYDROPYRIDO[2,1-A]PHTHALAZIN-2-ONES FOR THE TREATMENT A...
Publication number
20180127381
Publication date
May 10, 2018
HOFFMANN-LA ROCHE INC.
Zhanling CHENG
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL 2-OXO-6, 7-DIHYDROBENZO[a]QUINOLIZINE-3-CARBOXYLIC ACID DERIV...
Publication number
20170342069
Publication date
Nov 30, 2017
HOFFMANN-LA ROCHE INC.
Xingchun Han
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL DIHYDROQUINOLIZINONES FOR THE TREATMENT AND PROPHYLAXIS OF HE...
Publication number
20170057952
Publication date
Mar 2, 2017
HOFFMANN-LA ROCHE INC.
Song Yang
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel Tetrahydropyridopyrimidines and Tetrahydropyridopyridines for...
Publication number
20160326167
Publication date
Nov 10, 2016
HOFFMANN-LA ROCHE INC.
Zhanling Cheng
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL DIHYDROQUINOLIZINONES FOR THE TREATMENT AND PROPHYLAXIS OF HE...
Publication number
20160296515
Publication date
Oct 13, 2016
HOFFMANN-LA ROCHE INC.
Xingchun Han
A61 - MEDICAL OR VETERINARY SCIENCE HYGIENE
Information
Patent Application
NOVEL PYRAZINE COMPOUNDS FOR THE TREATMENT OF INFECTIOUS DISEASES
Publication number
20160237090
Publication date
Aug 18, 2016
HOFFMANN-LA ROCHE INC.
Taishan HU
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel dihydroquinolizinones for the treatment and prophylaxis of he...
Publication number
20160207914
Publication date
Jul 21, 2016
HOFFMANN-LA ROCHE INC.
Xingchun Han
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel 6,7-dihydrobenzo[a]quinolizin-2-one derivatives for the trea...
Publication number
20160122344
Publication date
May 5, 2016
HOFFMANN-LA ROCHE INC.
Xingchun Han
C07 - ORGANIC CHEMISTRY
Information
Patent Application
NOVEL BI-RING PHENYL-PYRIDINES/PYRAZINES FOR THE TREATMENT OF CANCER
Publication number
20150266878
Publication date
Sep 24, 2015
HOFFMANN-LA ROCHE INC.
Song Yang
C07 - ORGANIC CHEMISTRY
Information
Patent Application
Novel dihydroquinolizinones for the treatment and prophylaxis of he...
Publication number
20150210682
Publication date
Jul 30, 2015
HOFFMANN-LA ROCHE INC.
Xingchun Han
C07 - ORGANIC CHEMISTRY